Brief Information of the Compound and Protein
Compound Name
N-[3-(4-tert-butylphenyl)-5,6-dichloro-2-oxo-1H-indol-3-yl]-2-(4-methylpiperazin-1-yl)acetamide
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PubChem ID
CID: 71460564
Canonical SMILES
CN1CCN(CC(=O)NC2(C(=O)Nc3cc(Cl)c(Cl)cc23)c2ccc(cc2)C(C)(C)C)CC1
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Compound Formula C25H30Cl2N4O2
Compound Structure
Protein Name
Growth hormone secretagogue receptor type 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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GRP-related receptor
Uniprot ID
Q92847
Gene Name
GHSR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000643 CHO-K1/CRE-Luc Cricetulus griseus (Chinese hamster)  1
1
IC50 = 1470 nM
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