Compound ID |
Compound Name |
Compound Formula |
CP0372534
|
(S)-6-amino-2-((S)-2-amino-3-(1H-indol-3-yl)propanamido)-N-((5R,8S,11S,14S)-5-carbamoyl-15-(4-hydroxyphenyl)-8-isopropyl-11-(2-(methylthio)ethyl)-7,10,13-trioxo-2-thia-6,9,12-triazapentadecan-14-yl)hexanamide
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|
C41H61N9O7S2
|
1
|
1 |
EC50 = 10 nM
|
|
|
CP0046087
|
(S)-2-[(S)-2-((S)-2-Formylamino-4-methylsulfanyl-butyrylamino)-4-methyl-pentanoylamino]-3-phenyl-propionic acid
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|
C21H31N3O5S
|
1
|
1 |
EC50 = 1900 nM
|
|
|
CP0394900
|
N-(4-bromophenyl)-2-[3-methyl-6-oxo-5-(thiophen-2-ylmethyl)pyridazin-1-yl]acetamide
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|
C18H16BrN3O2S
|
1
|
1 |
EC50 = 10200 nM
|
|
|
CP0387583
|
N-(4-iodophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
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|
C21H20IN3O3
|
1
|
1 |
EC50 = 13000 nM
|
|
|
CP0382870
|
N-(4-bromophenyl)-2-[5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide
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|
C20H18BrN3O3
|
1
|
1 |
EC50 = 14600 nM
|
|
|
CP0396522
|
N-(4-bromophenyl)-2-[5-[(3-methoxyphenyl)methyl]-6-oxo-3-propan-2-ylpyridazin-1-yl]acetamide
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|
C23H24BrN3O3
|
1
|
1 |
EC50 = 17400 nM
|
|
|
CP0382862
|
2-(5-benzyl-3-methyl-6-oxopyridazin-1-yl)-N-(4-fluorophenyl)acetamide
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|
C20H18FN3O2
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0382863
|
N-(4-fluorophenyl)-2-[3-(4-fluorophenyl)-5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide
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|
C26H21F2N3O3
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0382864
|
N-(1,3-benzodioxol-5-yl)-2-[3-(4-fluorophenyl)-5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide
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|
C27H22FN3O5
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0382865
|
N-(1,3-benzodioxol-5-yl)-2-[5-[(3-methoxyphenyl)methyl]-6-oxo-3-phenylpyridazin-1-yl]acetamide
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|
C27H23N3O5
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0382866
|
N-(4-bromophenyl)-2-[5-[(3-bromophenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
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|
C20H17Br2N3O2
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0382867
|
2-[3-benzyl-5-[(4-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]-N-(4-bromophenyl)acetamide
Show/Hide
|
C27H24BrN3O3
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0387809
|
N-(4-bromophenyl)-2-[5-[(3,5-dimethoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
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|
C22H22BrN3O4
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0387810
|
2-[3-(4-chlorophenyl)-5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]-N-(4-fluorophenyl)acetamide
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|
C26H21ClFN3O3
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0387812
|
2-[3-ethyl-5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]-N-(4-iodophenyl)acetamide
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|
C22H22IN3O3
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0387813
|
N-(4-bromophenyl)-2-[5-[(4-methoxyphenyl)methyl]-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
Show/Hide
|
C24H20BrN3O3S
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0387815
|
N-(4-bromophenyl)-2-[5-[(4-cyanophenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
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|
C21H17BrN4O2
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0387817
|
N-(4-bromophenyl)-2-[5-[(4-methoxyphenyl)methyl]-3-(4-methylphenyl)-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C27H24BrN3O3
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0387818
|
N-(1,3-benzodioxol-5-yl)-2-[5-[(3-methoxyphenyl)methyl]-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
Show/Hide
|
C25H21N3O5S
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0387819
|
2-[5-[(3,5-dimethoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]-N-(4-iodophenyl)acetamide
Show/Hide
|
C22H22IN3O4
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0387820
|
N-(4-bromophenyl)-2-[5-(3-methoxybenzoyl)-3-methyl-6-oxopyridazin-1-yl]acetamide
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|
C21H18BrN3O4
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0387821
|
N-[2-[2-(4-bromoanilino)-2-oxoethyl]-6-methyl-3-oxopyridazin-4-yl]-3-methoxybenzamide
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|
C21H19BrN4O4
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0394901
|
N-(1,3-benzodioxol-5-yl)-2-(5-benzyl-3-methyl-6-oxopyridazin-1-yl)acetamide
Show/Hide
|
C21H19N3O4
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0394902
|
N-(4-bromophenyl)-2-[3-methyl-5-(naphthalen-1-ylmethyl)-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C24H20BrN3O2
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0394903
|
N-(4-bromophenyl)-2-[3-methyl-6-oxo-5-(pyridin-3-ylmethyl)pyridazin-1-yl]acetamide
Show/Hide
|
C19H17BrN4O2
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0396516
|
N-(1,3-benzodioxol-5-yl)-2-[3-(4-chlorophenyl)-5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C27H22ClN3O5
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0396517
|
N-(4-fluorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide
Show/Hide
|
C24H20FN3O3S
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0396518
|
N-(4-bromophenyl)-2-[3-cyclohexyl-5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C26H28BrN3O3
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0396519
|
N-(4-bromophenyl)-2-[3-(4-chlorophenyl)-5-[(4-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C26H21BrClN3O3
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0396520
|
N-(4-fluorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-6-oxo-3-phenylpyridazin-1-yl]acetamide
Show/Hide
|
C26H22FN3O3
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0396524
|
N-(4-bromophenyl)-2-[3-methyl-6-oxo-5-(thiophen-3-ylmethyl)pyridazin-1-yl]acetamide
Show/Hide
|
C18H16BrN3O2S
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0396525
|
2-[4-acetyl-5-(4-methoxyanilino)-3-methyl-6-oxopyridazin-1-yl]-N-(4-bromophenyl)acetamide
Show/Hide
|
C22H21BrN4O4
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0396526
|
N-(4-bromophenyl)-2-[5-[(3-methoxyphenyl)methyl]-6-oxo-3-phenylpyridazin-1-yl]acetamide
Show/Hide
|
C26H22BrN3O3
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0396527
|
2-(5-benzyl-3-methyl-6-oxopyridazin-1-yl)-N-(4-bromophenyl)acetamide
Show/Hide
|
C20H18BrN3O2
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0396528
|
2-[5-[(3-chlorophenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]-N-(4-iodophenyl)acetamide
Show/Hide
|
C20H17ClIN3O2
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0396530
|
N-(4-bromophenyl)-2-[5-[(3-fluorophenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C20H17BrFN3O2
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0396662
|
N-(4-bromophenyl)-2-[5-(furan-3-ylmethyl)-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C18H16BrN3O3
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0407624
|
4-bromo-N-[2-[2-(4-bromoanilino)-2-oxoethyl]-6-methyl-3-oxopyridazin-4-yl]benzamide
Show/Hide
|
C20H16Br2N4O3
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0413860
|
N-(4-bromophenyl)-2-[3-methyl-6-oxo-5-[[4-(trifluoromethyl)phenyl]methyl]pyridazin-1-yl]acetamide
Show/Hide
|
C21H17BrF3N3O2
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0413862
|
N-(4-fluorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-(4-methylphenyl)-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C27H24FN3O3
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0413863
|
N-(4-iodophenyl)-2-(3-methyl-6-oxo-4,5-dihydropyridazin-1-yl)acetamide
Show/Hide
|
C13H14IN3O2
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0413864
|
N-(1,3-benzodioxol-5-yl)-2-[3-(4-methoxyphenyl)-5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C28H25N3O6
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0413865
|
N-(4-bromophenyl)-2-[3-(4-methoxyphenyl)-5-[(4-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C27H24BrN3O4
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0423047
|
N-(4-bromophenyl)-2-[5-(4-methoxyanilino)-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C20H19BrN4O3
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0423063
|
2-(5-amino-3-methyl-6-oxopyridazin-1-yl)-N-(4-bromophenyl)acetamide
Show/Hide
|
C13H13BrN4O2
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0423064
|
4-[[2-[2-(4-bromoanilino)-2-oxoethyl]-6-methyl-3-oxopyridazin-4-yl]methyl]benzamide
Show/Hide
|
C21H19BrN4O3
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0432405
|
N-(4-iodophenyl)-2-(3-methyl-6-oxopyridazin-1-yl)acetamide
Show/Hide
|
C13H12IN3O2
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0433041
|
N-(4-bromophenyl)-2-[3-(4-fluorophenyl)-5-[(4-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C26H21BrFN3O3
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0435699
|
N-(1,3-benzodioxol-5-yl)-2-[5-[(3-methoxyphenyl)methyl]-3-(4-methylphenyl)-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C28H25N3O5
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0482517
|
N-(4-bromophenyl)-2-[5-(4-methoxyphenyl)-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C20H18BrN3O3
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0482518
|
N-(4-bromophenyl)-2-[5-[(3-chlorophenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C20H17BrClN3O2
|
1
|
1 |
EC50 > 50000 nM
|
|
|
CP0482519
|
N-(4-fluorophenyl)-2-[3-(4-methoxyphenyl)-5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide
Show/Hide
|
C27H24FN3O4
|
1
|
1 |
EC50 > 50000 nM
|
|
|