| Compound ID |
Compound Name |
Compound Formula |
|
CP0860990
|
3-(Diphenylphosphorothioyl)-2-methyl-1-(3-phenylpropyl)-imidazo[1,2-a]pyridin-1-ium Trifluoroacetate
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|
C31H28F3N2O2PS
|
2
|
| 1 |
IC50 < 0.5 nM
|
|
|
| 2 |
IC50 = 110 nM
|
|
|
|
CP0933738
|
SID99368032
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|
C30H30BrN2PS
|
3
|
| 1 |
IC50 < 0.5 nM
|
|
|
| 2 |
IC50 = 15 nM
|
|
|
| 3 |
IC50 = 940 nM
|
|
|
|
CP0467442
|
MLS002703109
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|
C29H26N2PS+
|
4
|
| 1 |
IC50 = 0.96 nM
|
|
|
| 2 |
IC50 = 1.3 nM
|
|
|
| 3 |
IC50 = 3.5 nM
|
|
|
| 4 |
IC50 = 45 nM
|
|
|
|
CP0321401
|
N-(3-methyl-1-morpholin-4-ylpentan-3-yl)-N-[(1-methyl-2-oxoquinolin-3-yl)methyl]cyclohexanecarboxamide
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|
C28H41N3O3
|
4
|
| 1 |
IC50 = 1.2 nM
|
|
|
| 2 |
IC50 = 6.7 nM
|
|
|
| 3 |
IC50 = 11 nM
|
|
|
| 4 |
IC50 = 55 nM
|
|
|
|
CP0942690
|
(E)-1-(3-(4-Chlorophenyl)allyl)-3-(diphenylphosphorothioyl)-2-methylimidazo[1,2-a]pyridin-1-iumTrifluoroacetate
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|
C31H25ClF3N2O2PS
|
2
|
| 1 |
IC50 = 2.2 nM
|
|
|
| 2 |
IC50 = 120 nM
|
|
|
|
CP0933710
|
(E)-3-(Diphenylphosphorothioyl)-1-(3-(3-methoxyphenyl)allyl)-2-methylimidazo[1,2-a]pyridin-1-iumTrifluoroacetate
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|
C32H28F3N2O3PS
|
2
|
| 1 |
IC50 = 3.2 nM
|
|
|
| 2 |
IC50 = 110 nM
|
|
|
|
CP0855742
|
(E)-1-(3-(2-Chlorophenyl)allyl)-3-(diphenylphosphorothioyl)-2-methylimidazo[1,2-a]pyridin-1-iumTrifluoroacetate
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|
C31H25ClF3N2O2PS
|
2
|
| 1 |
IC50 = 3.4 nM
|
|
|
| 2 |
IC50 = 94 nM
|
|
|
|
CP0903634
|
(E)-3-(Diphenylphosphorothioyl)-1-(3-(4-fluorophenyl)allyl)-2-methylimidazo[1,2-a]pyridin-1-iumTrifluoroacetate
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|
C31H25F4N2O2PS
|
2
|
| 1 |
IC50 = 3.4 nM
|
|
|
| 2 |
IC50 = 71 nM
|
|
|
|
CP0938258
|
(E)-3-(Diphenylphosphorothioyl)-2-methyl-1-(3-(4-(trifluoromethyl)phenyl)allyl)imidazo[1,2-a]pyridin-1-iumTrifluoroacetate
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|
C32H25F6N2O2PS
|
2
|
| 1 |
IC50 = 4.5 nM
|
|
|
| 2 |
IC50 = 400 nM
|
|
|
|
CP0334232
|
N-[(4-fluorophenyl)methyl]-3-oxo-1,1-diphenyl-5,6,8,8a-tetrahydro-[1,3]oxazolo[3,4-a]pyrazine-7-carboxamide
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|
C26H24FN3O3
|
4
|
| 1 |
IC50 = 5.3 nM
|
|
|
| 2 |
IC50 = 14 nM
|
|
|
| 3 |
IC50 = 25 nM
|
|
|
| 4 |
IC50 = 420 nM
|
|
|
|
CP0855738
|
(E)-1-(3-(4-Bromophenyl)allyl)-3-(diphenylphosphorothioyl)-2-methylimidazo[1,2-a]pyridin-1-iumTrifluoroacetate
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|
C31H25BrF3N2O2PS
|
2
|
| 1 |
IC50 = 5.7 nM
|
|
|
| 2 |
IC50 = 170 nM
|
|
|
|
CP0903784
|
SID99368034
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|
C33H32F3N2O2PS
|
3
|
| 1 |
IC50 = 6.2 nM
|
|
|
| 2 |
IC50 = 13 nM
|
|
|
| 3 |
IC50 = 710 nM
|
|
|
|
CP0899575
|
(E)-3-(Diphenylphosphorothioyl)-2-methyl-1-(3-p-tolylallyl)-imidazo[1,2-a]pyridin-1-iumBromide
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|
C30H28BrN2PS
|
2
|
| 1 |
IC50 = 9 nM
|
|
|
| 2 |
IC50 = 330 nM
|
|
|
|
CP0406002
|
(2-methylimidazo[1,2-a]pyridin-3-yl)-diphenyl-sulfanylidene-lambda5-phosphane
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|
C20H17N2PS
|
3
|
| 1 |
IC50 = 9.1 nM
|
|
|
| 2 |
IC50 = 1000 nM
|
|
|
| 3 |
IC50 = 18000 nM
|
|
|
|
CP0860977
|
(E)-1-(3-(3-Chlorophenyl)allyl)-3-(diphenylphosphorothioyl)-2-methylimidazo[1,2-a]pyridin-1-iumTrifluoroacetate
Show/Hide
|
C31H25ClF3N2O2PS
|
2
|
| 1 |
IC50 = 9.2 nM
|
|
|
| 2 |
IC50 = 220 nM
|
|
|
|
CP0894046
|
3-(Diphenylphosphorothioyl)-2-methyl-1-(1-oxo-2-phenylethyl)-imidazo[1,2-a]pyridin-1-ium Bromide
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|
C28H24BrN2OPS
|
3
|
| 1 |
IC50 = 13 nM
|
|
|
| 2 |
IC50 = 80 nM
|
|
|
| 3 |
IC50 = 2100 nM
|
|
|
|
CP0855747
|
SID87796315
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|
C28H26BrN2PS
|
3
|
| 1 |
IC50 = 16 nM
|
|
|
| 2 |
IC50 = 73 nM
|
|
|
| 3 |
IC50 = 2100 nM
|
|
|
|
CP0855748
|
1-Benzyl-3-(diphenylphosphorothioyl)-2-methylimidazo[1,2-a]-pyridin-1-ium Trifluoroacetate
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|
C29H24F3N2O2PS
|
3
|
| 1 |
IC50 = 16 nM
|
|
|
| 2 |
IC50 = 32 nM
|
|
|
| 3 |
IC50 = 1300 nM
|
|
|
|
CP0938260
|
(E)-1-(3-(3-Bromophenyl)allyl)-3-(diphenylphosphorothioyl)-2-methylimidazo[1,2-a]pyridin-1-iumTrifluoroacetate
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|
C31H25BrF3N2O2PS
|
2
|
| 1 |
IC50 = 23 nM
|
|
|
| 2 |
IC50 = 670 nM
|
|
|
|
CP0842124
|
3-(diphenylphosphorothioyl)-1,2-dimethylimidazo[1,2-a]pyridin-1-ium
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|
C21H20IN2PS
|
3
|
| 1 |
IC50 = 30 nM
|
|
|
| 2 |
IC50 = 51 nM
|
|
|
| 3 |
IC50 = 1700 nM
|
|
|
|
CP0938257
|
(E)-1-(3-(3-Bromo-4-fluorophenyl)allyl)-3-(diphenylphosphorothioyl)-2-methylimidazo[1,2-a]pyridin-1-iumTrifluoroacetate
Show/Hide
|
C31H24BrF4N2O2PS
|
2
|
| 1 |
IC50 = 45 nM
|
|
|
| 2 |
IC50 = 840 nM
|
|
|
|
CP0860976
|
(E)-3-(Diphenylphosphorothioyl)-2-methyl-1-(3-(naphthalen-2-yl)allyl)imidazo[1,2-a]pyridin-1-iumBromide
Show/Hide
|
C33H28BrN2PS
|
2
|
| 1 |
IC50 = 64 nM
|
|
|
| 2 |
IC50 = 1300 nM
|
|
|
|
CP0899743
|
3-(Diphenylphosphorothioyl)-1-methylimidazo[1,2-a]-pyridin-1-iumMethylSulfate
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|
C21H21N2O4PS2
|
2
|
| 1 |
IC50 = 2500 nM
|
|
|
| 2 |
IC50 = 39000 nM
|
|
|
|
CP0942689
|
SID87796301
Show/Hide
|
C22H20NPS
|
1
|
| 1 |
IC50 = 2800 nM
|
|
|
|
CP0487769
|
imidazo[1,2-a]pyridin-3-yl-diphenyl-sulfanylidene-lambda5-phosphane
Show/Hide
|
C19H15N2PS
|
2
|
| 1 |
IC50 = 4030 nM
|
|
|
| 2 |
IC50 = 63000 nM
|
|
|
|
CP0855750
|
SID87796306
Show/Hide
|
C21H18NPS
|
1
|
| 1 |
IC50 = 7300 nM
|
|
|
|
CP0461904
|
3-diphenylphosphoryl-2-methylimidazo[1,2-a]pyridine
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|
C20H17N2OP
|
1
|
| 1 |
IC50 = 27000 nM
|
|
|
|
CP0470453
|
imidazo[1,2-a]pyridin-3-yl(diphenyl)phosphane
Show/Hide
|
C19H15N2P
|
1
|
| 1 |
IC50 = 35000 nM
|
|
|
