Brief Information of the Cell Line and Protein
Cell Line ID: CL001056 , MEF-1 [Mouse fibroblast]
Synonyms
MEF1
Mouse Embryo Fibroblast-1
Category Transformed cell line
Organism
Mus musculus (Mouse)
Protein ID: PT04536 , Lysophosphatidic acid receptor 2
Gene Name LPAR2
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID Q9HBW0
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL001056  Protein ID: PT04536
 
Compound ID Compound Name Compound Formula
CP0379813
2-[4-(1,3-dioxobenzo[de]isoquinolin-2-yl)butylsulfamoyl]-5-fluorobenzoic acid
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C23H19FN2O6S
 1
1
EC50 = 0.15 nM
   TI
   LI
   LO
   TS
CP0125579
(R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-propyl ester
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C21H41O7P
 1
1
EC50 = 2 nM
   TI
   LI
   LO
   TS
CP0482104
(2-hydroxy-3-phosphonooxypropyl) (Z)-octadec-9-enoate
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C21H41O7P
 1
1
EC50 = 3 nM
   TI
   LI
   LO
   TS
CP0415360
4-bromo-2-[4-(1,3-dioxobenzo[de]isoquinolin-2-yl)butylsulfamoyl]benzoic acid
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C23H19BrN2O6S
 1
1
EC50 = 50 nM
   TI
   LI
   LO
   TS
CP0480547
5-bromo-2-[4-(1,3-dioxobenzo[de]isoquinolin-2-yl)butylsulfamoyl]benzoic acid
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C23H19BrN2O6S
 1
1
EC50 = 60 nM
   TI
   LI
   LO
   TS
CP0410868
2-[4-(1,3-dioxobenzo[de]isoquinolin-2-yl)butylsulfamoyl]benzoic acid
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C23H20N2O6S
 1
1
EC50 = 110 nM
   TI
   LI
   LO
   TS
CP0415517
2-[5-(1,3-dioxobenzo[de]isoquinolin-2-yl)pentylsulfamoyl]benzoic acid
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C24H22N2O6S
 1
1
EC50 = 1420 nM
   TI
   LI
   LO
   TS
CP0375203
2-[3-(1,3-dioxobenzo[de]isoquinolin-2-yl)propylsulfamoyl]benzoic acid
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C22H18N2O6S
 1
1
EC50 = 2160 nM
   TI
   LI
   LO
   TS
CP0410869
2-[3-(1,3-dioxobenzo[de]isoquinolin-2-yl)propylsulfanyl]benzoic acid
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C22H17NO4S
 1
1
EC50 = 3300 nM
   TI
   LI
   LO
   TS
CP0480548
2-[4-(1,3-dioxobenzo[de]isoquinolin-2-yl)butyl]-1,1,3-trioxo-1,2-benzothiazole-6-carboxylic acid
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C24H18N2O7S
 1
1
EC50 = 3600 nM
   TI
   LI
   LO
   TS