| Compound ID |
Compound Name |
Compound Formula |
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CP0958942
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N-((2S)-3-hydroxy-1-((2S)-1-hydroxy-1-((R)-2-methyloxiran-2-yl)-3-phenylpropan-2-ylamino)-1-oxopropan-2-yl)-6-oxo-1,6-dihydropyridine-2-carboxamide
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C21H25N3O6
|
2
|
| 1 |
IC50 = 28 nM
|
|
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| 2 |
IC50 = 204.4 nM
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CP0075994
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(2S)-1-(2-acetamidoacetyl)-N-[(2S)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]pyrrolidine-2-carboxamide
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|
C27H38N4O6
|
2
|
| 1 |
IC50 = 30.9 nM
|
|
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| 2 |
IC50 = 213 nM
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CP0418920
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(3S,6S)-N-[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxo-3-phenylpropan-2-yl]-5,11-dioxo-19-oxa-4,10-diazatricyclo[18.2.2.06,10]tetracosa-1(23),20(24),21-triene-3-carboxamide
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|
C34H43N3O6
|
2
|
| 1 |
IC50 = 32.7 nM
|
|
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| 2 |
IC50 = 105.6 nM
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|
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CP0576198
|
(3S,6S)-N-[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]-5,11-dioxo-19-oxa-4,10-diazatricyclo[18.2.2.06,10]tetracosa-1(23),20(24),21-triene-3-carboxamide
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|
C31H45N3O6
|
2
|
| 1 |
IC50 = 33.9 nM
|
|
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| 2 |
IC50 = 160.7 nM
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|
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CP0573254
|
(10S,13S)-N-[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]-2,12-dioxo-8-oxa-1,11-diazabicyclo[11.3.0]hexadecane-10-carboxamide
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|
C23H37N3O6
|
2
|
| 1 |
IC50 = 35.8 nM
|
|
|
| 2 |
IC50 = 146.8 nM
|
|
|
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CP0475672
|
(2S)-1-[(2S)-2-[(2-azidoacetyl)amino]propanoyl]-N-[(2S)-1-[[(2S)-3-cyclohexyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-1-oxohexan-2-yl]-4,4-difluoropyrrolidine-2-carboxamide
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|
C28H43F2N7O6
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0399509
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(2S)-1-[(2S)-2-[(2-azidoacetyl)amino]propanoyl]-N-[(2S)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]pyrrolidine-2-carboxamide
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|
C25H41N7O6
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0062987
|
(2S)-3-(4-methoxyphenyl)-N-[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxo-3-phenylpropan-2-yl]-2-[[(2S)-2-[(2-morpholin-4-ylacetyl)amino]propanoyl]amino]propanamide
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|
C31H40N4O7
|
1
|
| 1 |
IC50 = 340 nM
|
|
|
|
CP0885679
|
(S)-N-((S)-3-cyclohexyl-1-((R)-2-methyloxiran-2-yl)-1-oxopropan-2-yl)-3-(4-methoxyphenyl)-2-((S)-2-(2-morpholinoacetamido)propanamido)propanamide
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|
C31H46N4O7
|
1
|
| 1 |
IC50 = 370 nM
|
|
|
|
CP0847941
|
N-((R)-1-((S)-3-(1H-indol-3-yl)-1-((S)-1-((R)-2-methyloxiran-2-yl)-1-oxo-3-phenylpropan-2-ylamino)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-3-methyl-1H-indene-2-carboxamide
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|
C37H38N4O5
|
1
|
| 1 |
IC50 = 3500 nM
|
|
|
|
CP0864816
|
(S)-N-((S)-3-cyclohexyl-1-((R)-2-methyloxiran-2-yl)-1-oxopropan-2-yl)-3-(1H-indol-3-yl)-2-((R)-2-(2-morpholinoacetamido)propanamido)propanamide
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|
C32H45N5O6
|
1
|
| 1 |
IC50 = 6200 nM
|
|
|
|
CP0386861
|
(2S)-N-[(2S)-3-cyclohexyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]-3-(4-methoxyphenyl)-2-[[(2R)-2-[(2-morpholin-4-ylacetyl)amino]propanoyl]amino]propanamide
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|
C31H46N4O7
|
1
|
| 1 |
IC50 = 7300 nM
|
|
|
|
CP0576199
|
(13S,16S)-N-[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]-2,5,15-trioxo-11-oxa-1,4,14-triazabicyclo[14.3.0]nonadecane-13-carboxamide
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|
C25H40N4O7
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0351150
|
(14S,17S)-N-[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]-2,5,16-trioxo-12-oxa-1,4,15-triazabicyclo[15.3.0]icosane-14-carboxamide
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|
C26H42N4O7
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0868641
|
N-((R)-1-((S)-1-((S)-3-cyclohexyl-1-((R)-2-methyloxiran-2-yl)-1-oxopropan-2-ylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-3-methyl-1H-indene-2-carboxamide
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|
C37H44N4O5
|
1
|
| 1 |
IC50 = 16000 nM
|
|
|
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CP0411613
|
N-[(2R)-1-[[(2S)-1-[[(2S)-3-cyclohexyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-3-(4-methoxyphenyl)-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]-3-methyl-1H-indene-2-carboxamide
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|
C36H45N3O6
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
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CP0850423
|
N-((R)-1-((S)-3-(1H-indol-3-yl)-1-((S)-4-(methylsulfonyl)-1-phenylbut-3-en-2-ylamino)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-3-methyl-1H-indene-2-carboxamide
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|
C36H38N4O5S
|
1
|
| 1 |
IC50 > 100000 nM
|
|
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