Brief Information of the Cell Line and Protein
Cell Line ID: CL000102 , U-87MG ATCC
Synonyms
U-87MG
U-87 MG
U87 MG
U-87-MG
U87-MG
U87MG
U-87
U87
87 MG
87MG
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0022
Protein ID: PT03648 , Isocitrate dehydrogenase [NADP], mitochondrial
Gene Name IDH2
Organism Homo sapiens, Human
Protein Classification Enzyme
Uniprot ID P48735
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000102  Protein ID: PT03648
 
Compound ID Compound Name Compound Formula
CP0476930
US10028961, Compound 149
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C17H15F7N6
 1
1
IC50 = 3 nM
   TI
   LI
   LO
   TS
CP0551346
US10028961, Compound 45
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C18H23ClN6
 1
1
IC50 = 4 nM
   TI
   LI
   LO
   TS
CP0387438
US10028961, Compound 113
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C18H19ClF4N6
 1
1
IC50 = 6 nM
   TI
   LI
   LO
   TS
CP0420686
US10028961, Compound 142
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C14H13ClF6N6
 1
1
IC50 = 7 nM
   TI
   LI
   LO
   TS
CP0401743
US10028961, Compound 130
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C14H13ClF6N6
 1
1
IC50 = 8 nM
   TI
   LI
   LO
   TS
CP0412010
US10028961, Compound 31
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C19H19F7N6
 1
1
IC50 = 9 nM
   TI
   LI
   LO
   TS
CP0455814
US10028961, Compound 41
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C21H23F7N6
 1
1
IC50 = 9 nM
   TI
   LI
   LO
   TS
CP0387387
US10028961, Compound 110
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C20H27ClN6
 1
1
IC50 = 14 nM
   TI
   LI
   LO
   TS
CP0424115
US10028961, Compound 2
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C19H23F3N6
 1
1
IC50 = 14 nM
   TI
   LI
   LO
   TS
CP0427569
US10028961, Compound 1
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C17H19F3N6
 1
1
IC50 = 22 nM
   TI
   LI
   LO
   TS
CP0477111
US10028961, Compound 212
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C20H23ClF4N6
 1
1
IC50 = 22 nM
   TI
   LI
   LO
   TS