| Compound ID |
Compound Name |
Compound Formula |
|
CP0229599
|
2-ethyl-N-[1-[(E)-4-[2-(2-ethyl-5-methylpyrazole-3-carbonyl)imino-3-methyl-7-(piperidin-1-ylmethyl)benzimidazol-1-yl]but-2-enyl]-3-methylbenzimidazol-2-ylidene]-5-methylpyrazole-3-carboxamide
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|
C40H49N11O2
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0229600
|
2-ethyl-N-[1-[(E)-4-[2-(2-ethyl-5-methylpyrazole-3-carbonyl)imino-4-(hydroxymethyl)-3-methylbenzimidazol-1-yl]but-2-enyl]-3-methylbenzimidazol-2-ylidene]-5-methylpyrazole-3-carboxamide
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|
C35H40N10O3
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0311616
|
N-[1-[(E)-4-[7-(1,2-dihydroxyethyl)-2-(2-ethyl-5-methylpyrazole-3-carbonyl)imino-3-methylbenzimidazol-1-yl]but-2-enyl]-3-methylbenzimidazol-2-ylidene]-2-ethyl-5-methylpyrazole-3-carboxamide
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|
C36H42N10O4
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0317724
|
2-ethyl-N-[1-[(E)-4-[2-(2-ethyl-5-methylpyrazole-3-carbonyl)imino-3-methyl-7-(morpholin-4-ylmethyl)benzimidazol-1-yl]but-2-enyl]-3-methylbenzimidazol-2-ylidene]-5-methylpyrazole-3-carboxamide
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|
C39H47N11O3
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0543694
|
N-[1-[(E)-4-[7-(azepan-1-ylmethyl)-2-(2-ethyl-5-methylpyrazole-3-carbonyl)imino-3-methylbenzimidazol-1-yl]but-2-enyl]-3-methylbenzimidazol-2-ylidene]-2-ethyl-5-methylpyrazole-3-carboxamide
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|
C41H51N11O2
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0576045
|
2-ethyl-N-[3-[(E)-4-[2-(2-ethyl-5-methylpyrazole-3-carbonyl)imino-7-(3-hydroxypropoxy)-3-methylbenzimidazol-1-yl]but-2-enyl]-4-methoxy-1-methylbenzimidazol-2-ylidene]-5-methylpyrazole-3-carboxamide
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|
C38H46N10O5
|
1
|
| 1 |
EC50 < 1 nM
|
|
|
|
CP0248635
|
1-[(E)-4-[5-carbamoyl-2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-(3-morpholin-4-ylpropoxy)benzimidazol-1-yl]but-2-enyl]-2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-methoxybenzimidazole-5-carboxamide
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|
C42H51N13O7
|
1
|
| 1 |
EC50 = 130 nM
|
|
|
|
CP0243314
|
benzyl N-[3-[5-carbamoyl-2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-(3-morpholin-4-ylpropoxy)benzimidazol-1-yl]propyl]carbamate
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|
C33H42N8O6
|
1
|
| 1 |
EC50 = 1110 nM
|
|
|
|
CP0069029
|
tert-butyl N-[3-[5-carbamoyl-2-[(2-ethyl-5-methylpyrazole-3-carbonyl)amino]-7-methoxybenzimidazol-1-yl]propyl]carbamate
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|
C24H33N7O5
|
1
|
| 1 |
EC50 = 1790 nM
|
|
|
|
CP0345476
|
3-chloro-5-methyl-2-[(pyrazolo[1,5-a]pyrimidine-3-carbonylamino)methyl]-1-benzofuran-7-carboxylic acid
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|
C18H13ClN4O4
|
6
|
| 1 |
EC50 = 5900 nM
|
|
|
| 2 |
EC50 = 11000 nM
|
|
|
| 3 |
EC50 = 15000 nM
|
|
|
| 4 |
EC50 = 21000 nM
|
|
|
| 5 |
EC50 = 34000 nM
|
|
|
| 6 |
EC50 = 35000 nM
|
|
|
