| Compound ID |
Compound Name |
Compound Formula |
|
CP0534919
|
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(4-methylcyclohexyl)-N-[(2S)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]propanamide
Show/Hide
|
C37H50N6O5
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 11 nM
|
|
|
|
CP0045910
|
(S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2-methyloxiran-2-yl)-1-oxopentan-2-ylamino)-1-oxo-3-phenylpropan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)-3-phenylpropanamide
Show/Hide
|
C36H42N6O5
|
2
|
| 1 |
IC50 = 2.1 nM
|
|
|
| 2 |
IC50 = 5.5 nM
|
|
|
|
CP0446489
|
(2S)-2-[[(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(4-methoxyphenyl)propanoyl]amino]-N-[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]-3-phenylpropanamide
Show/Hide
|
C37H44N6O6
|
2
|
| 1 |
IC50 = 2.1 nM
|
|
|
| 2 |
IC50 = 7.8 nM
|
|
|
|
CP0455723
|
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(4-methoxycyclohexyl)-N-[(2S)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]propanamide
Show/Hide
|
C37H50N6O6
|
2
|
| 1 |
IC50 = 2.1 nM
|
|
|
| 2 |
IC50 = 22 nM
|
|
|
|
CP0475289
|
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-N-[(2S)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]-4-phenylbutanamide
Show/Hide
|
C37H44N6O5
|
2
|
| 1 |
IC50 = 3 nM
|
|
|
| 2 |
IC50 = 5.1 nM
|
|
|
|
CP0455719
|
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]-3-(4-phenylcyclohexyl)propanamide
Show/Hide
|
C39H46N6O5
|
2
|
| 1 |
IC50 = 3.8 nM
|
|
|
| 2 |
IC50 = 8560 nM
|
|
|
|
CP0420041
|
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(4-cyclohexylcyclohexyl)-N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]propanamide
Show/Hide
|
C39H52N6O5
|
2
|
| 1 |
IC50 = 4.9 nM
|
|
|
| 2 |
IC50 = 13200 nM
|
|
|
|
CP0420035
|
(2S)-3-(1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalen-2-yl)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-N-[(2S)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]propanamide
Show/Hide
|
C40H54N6O5
|
2
|
| 1 |
IC50 < 10 nM
|
|
|
| 2 |
IC50 = 25 nM
|
|
|
|
CP0420037
|
(2S)-2-[[(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-2-phenylacetyl]amino]-N-[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]-3-phenylpropanamide
Show/Hide
|
C35H40N6O5
|
2
|
| 1 |
IC50 < 10 nM
|
|
|
| 2 |
IC50 > 10 nM
|
|
|
|
CP0446490
|
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(2-bicyclo[2.2.1]heptanyl)-N-[(2S)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]propanamide
Show/Hide
|
C37H48N6O5
|
2
|
| 1 |
IC50 < 10 nM
|
|
|
| 2 |
IC50 = 33 nM
|
|
|
|
CP0490362
|
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-cyclohexyl-N-[(2S)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]propanamide
Show/Hide
|
C36H48N6O5
|
2
|
| 1 |
IC50 < 10 nM
|
|
|
| 2 |
IC50 = 50 nM
|
|
|
|
CP0534915
|
(2S)-2-[[(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(4-methylphenyl)propanoyl]amino]-N-[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]-3-phenylpropanamide
Show/Hide
|
C37H44N6O5
|
1
|
| 1 |
IC50 < 10 nM
|
|
|
|
CP0534916
|
(2S)-2-[[(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(4-phenylphenyl)propanoyl]amino]-N-[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]-3-phenylpropanamide
Show/Hide
|
C39H40N6O5
|
2
|
| 1 |
IC50 < 10 nM
|
|
|
| 2 |
IC50 = 134 nM
|
|
|
|
CP0540693
|
(2S)-2-[[(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(4-phenylphenyl)propanoyl]amino]-N-[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]-3-phenylpropanamide
Show/Hide
|
C42H46N6O5
|
1
|
| 1 |
IC50 < 10 nM
|
|
|
|
CP0550476
|
(2S)-3-(1,2,3,4,4a,5,6,7,8,8a-decahydronaphthalen-1-yl)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-N-[(2S)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]propanamide
Show/Hide
|
C40H54N6O5
|
2
|
| 1 |
IC50 < 10 nM
|
|
|
| 2 |
IC50 = 15 nM
|
|
|
|
CP0420036
|
(2S)-2-[[(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-naphthalen-2-ylpropanoyl]amino]-N-[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]-3-phenylpropanamide
Show/Hide
|
C40H44N6O5
|
1
|
| 1 |
IC50 < 10 nM
|
|
|
|
CP0420038
|
(2S)-2-[[(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-naphthalen-1-ylpropanoyl]amino]-N-[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]-3-phenylpropanamide
Show/Hide
|
C40H44N6O5
|
1
|
| 1 |
IC50 < 10 nM
|
|
|
|
CP0420039
|
(2S)-N-[(2S)-3-(4-methoxyphenyl)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]-2-[(2-morpholin-4-ylacetyl)amino]-3-(4-phenylphenyl)propanamide
Show/Hide
|
C40H50N4O7
|
1
|
| 1 |
IC50 < 10 nM
|
|
|
|
CP0482497
|
(2S)-3-(4-methoxyphenyl)-N-[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]-2-[[(2S)-2-[(2-morpholin-4-ylacetyl)amino]-3-naphthalen-1-ylpropanoyl]amino]propanamide
Show/Hide
|
C38H48N4O7
|
1
|
| 1 |
IC50 < 10 nM
|
|
|
|
CP0534918
|
(2S)-2-[[(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-N-[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]-3-phenylpropanamide
Show/Hide
|
C38H43N7O5
|
1
|
| 1 |
IC50 < 10 nM
|
|
|
|
CP0549256
|
(2S)-3-(4-methoxyphenyl)-N-[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]-2-[[(2S)-2-[(2-morpholin-4-ylacetyl)amino]-3-naphthalen-2-ylpropanoyl]amino]propanamide
Show/Hide
|
C38H48N4O7
|
1
|
| 1 |
IC50 < 10 nM
|
|
|
|
CP0868641
|
N-((R)-1-((S)-1-((S)-3-cyclohexyl-1-((R)-2-methyloxiran-2-yl)-1-oxopropan-2-ylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-3-methyl-1H-indene-2-carboxamide
Show/Hide
|
C37H44N4O5
|
2
|
| 1 |
IC50 = 16 nM
|
|
|
| 2 |
IC50 > 1000 nM
|
|
|
|
CP0420040
|
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(4-cyclohexylcyclohexyl)-N-[(2S)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]propanamide
Show/Hide
|
C42H58N6O5
|
2
|
| 1 |
IC50 = 17 nM
|
|
|
| 2 |
IC50 = 439 nM
|
|
|
|
CP0549209
|
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-4,4-dimethyl-N-[(2S)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]pentanamide
Show/Hide
|
C34H46N6O5
|
2
|
| 1 |
IC50 = 18 nM
|
|
|
| 2 |
IC50 = 68 nM
|
|
|
|
CP0455722
|
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(4-cyclohexylcyclohexyl)-N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]propanamide
Show/Hide
|
C39H52N6O5
|
2
|
| 1 |
IC50 = 20 nM
|
|
|
| 2 |
IC50 > 10000 nM
|
|
|
|
CP0482909
|
(2S)-N-[(2S)-3-(4-cyclohexylcyclohexyl)-1-[[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-1-oxopropan-2-yl]-4-methyl-2-[(2-morpholin-4-ylacetyl)amino]pentanamide
Show/Hide
|
C42H65N5O7
|
2
|
| 1 |
IC50 = 28 nM
|
|
|
| 2 |
IC50 = 22800 nM
|
|
|
|
CP0446491
|
(2S)-2-[[(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-2-cyclohexylacetyl]amino]-N-[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]-3-phenylpropanamide
Show/Hide
|
C35H46N6O5
|
2
|
| 1 |
IC50 = 33 nM
|
|
|
| 2 |
IC50 = 72 nM
|
|
|
|
CP0530760
|
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-4-cyclohexyl-N-[(2S)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]butanamide
Show/Hide
|
C37H50N6O5
|
2
|
| 1 |
IC50 = 35 nM
|
|
|
| 2 |
IC50 = 36 nM
|
|
|
|
CP0549255
|
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-cyclohexyl-N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]propanamide
Show/Hide
|
C33H42N6O5
|
2
|
| 1 |
IC50 = 57 nM
|
|
|
| 2 |
IC50 > 10000 nM
|
|
|
|
CP0446492
|
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]-3-(4-phenylcyclohexyl)propanamide
Show/Hide
|
C39H46N6O5
|
2
|
| 1 |
IC50 = 71 nM
|
|
|
| 2 |
IC50 = 11700 nM
|
|
|
|
CP0540677
|
(2S)-3-cyclohexyl-N-[(2S)-3-(4-methoxyphenyl)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxopropan-2-yl]-2-[(2-morpholin-4-ylacetyl)amino]propanamide
Show/Hide
|
C34H52N4O7
|
2
|
| 1 |
IC50 = 119 nM
|
|
|
| 2 |
IC50 = 274 nM
|
|
|
|
CP0540676
|
(2S)-2-[[(2S)-3-(1-adamantyl)-2-[(2-morpholin-4-ylacetyl)amino]propanoyl]amino]-3-(4-methoxyphenyl)-N-[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]propanamide
Show/Hide
|
C38H56N4O7
|
2
|
| 1 |
IC50 = 638 nM
|
|
|
| 2 |
IC50 = 853 nM
|
|
|
|
CP0475291
|
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(4-cyclohexylcyclohexyl)-N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]propanamide
Show/Hide
|
C39H52N6O5
|
2
|
| 1 |
IC50 = 710 nM
|
|
|
| 2 |
IC50 = 21600 nM
|
|
|
|
CP0544673
|
(2S)-2-[[(2S)-3-(1-adamantyl)-2-[(2-morpholin-4-ylacetyl)amino]propanoyl]amino]-3-(4-methoxyphenyl)-N-[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]propanamide
Show/Hide
|
C35H50N4O7
|
2
|
| 1 |
IC50 = 853 nM
|
|
|
| 2 |
IC50 > 10000 nM
|
|
|
|
CP0490363
|
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]-3-[(2-methylpropan-2-yl)oxy]butanamide
Show/Hide
|
C32H42N6O6
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0529457
|
(2S)-3-(4-cyclohexylcyclohexyl)-N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]-2-[(2-morpholin-4-ylacetyl)amino]propanamide
Show/Hide
|
C36H54N4O6
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
