| Compound ID |
Compound Name |
Compound Formula |
|
CP0116207
|
CHEMBL3717769
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|
C19H22F5N5
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0390422
|
5-[5-[1-(oxetan-3-yl)piperidin-4-yl]-1-propan-2-ylpyrazol-3-yl]-3-(trifluoromethyl)-1H-pyrrolo[2,3-b]pyridine
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|
C22H26F3N5O
|
1
|
| 1 |
Ki = 2.3 nM
|
|
|
|
CP0016719
|
5-[5-[(1R,5S)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]-1-propan-2-ylpyrazol-3-yl]-3-(trifluoromethoxy)pyridin-2-amine
Show/Hide
|
C20H24F3N5O2
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0477225
|
CHEMBL4125721
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|
C21H24F3N5O2
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0477226
|
CHEMBL4128619
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|
C21H26F3N5O
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0552526
|
5-[1-ethyl-5-[(1S,5R)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]pyrazol-3-yl]-3-(trifluoromethyl)pyridin-2-amine
Show/Hide
|
C19H22F3N5O
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0023938
|
CHEMBL3715238
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|
C21H24F3N5O
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0261263
|
3-methyl-5-[5-[1-(oxetan-3-yl)piperidin-4-yl]-1-propan-2-ylpyrazol-3-yl]-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C22H29N5O
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0389292
|
CHEMBL4128889
Show/Hide
|
C20H26F3N5O
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0396483
|
5-[5-[(1S,5R)-3-(oxetan-3-ylmethyl)-3-azabicyclo[3.1.0]hexan-6-yl]-1-propan-2-ylpyrazol-3-yl]-3-(trifluoromethyl)pyridin-2-amine
Show/Hide
|
C21H26F3N5O
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0122104
|
CHEMBL3718265
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|
C19H22F3N5O
|
1
|
| 1 |
Ki = 6 nM
|
|
|
|
CP0133222
|
CHEMBL3717481
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|
C20H24F3N5O
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0555734
|
CHEMBL3715469
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|
C20H27N5O2
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0074414
|
CHEMBL3714987
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|
C20H25F2N5O2
|
1
|
| 1 |
Ki = 8 nM
|
|
|
|
CP0478051
|
5-[1-(cyclopentylmethyl)-5-[(1R,5S)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]pyrazol-3-yl]-3-(trifluoromethyl)pyridin-2-amine
Show/Hide
|
C23H28F3N5O
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0538682
|
5-[5-[(1S,5R)-3-(2-methoxyethyl)-3-azabicyclo[3.1.0]hexan-6-yl]-1-propan-2-ylpyrazol-3-yl]-3-(trifluoromethyl)pyridin-2-amine
Show/Hide
|
C20H26F3N5O
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0122103
|
5-[1-(cyclobutylmethyl)-5-[(1S,5R)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]pyrazol-3-yl]-3-(trifluoromethyl)pyridin-2-amine
Show/Hide
|
C22H26F3N5O
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0552789
|
3-chloro-5-[5-[1-(oxetan-3-yl)piperidin-4-yl]-1-propan-2-ylpyrazol-3-yl]-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C21H26ClN5O
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0224284
|
CHEMBL3718522
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|
C19H19F6N5O
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0456375
|
CHEMBL4127238
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|
C21H26F3N5O2
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0210720
|
CHEMBL3717627
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|
C20H25F2N5O
|
1
|
| 1 |
Ki = 35 nM
|
|
|
|
CP0538684
|
CHEMBL4127922
Show/Hide
|
C18H20F3N5O2
|
1
|
| 1 |
Ki = 67 nM
|
|
|
|
CP0550383
|
CHEMBL4126530
Show/Hide
|
C18H20F3N5O
|
1
|
| 1 |
Ki = 82 nM
|
|
|
|
CP0332421
|
3-fluoro-5-[5-[1-(oxetan-3-yl)piperidin-4-yl]-1-propan-2-ylpyrazol-3-yl]-1H-pyrrolo[2,3-b]pyridine
Show/Hide
|
C21H26FN5O
|
1
|
| 1 |
Ki = 96 nM
|
|
|
|
CP0304367
|
3-methoxy-5-[5-[1-(oxetan-3-yl)piperidin-4-yl]-1-propan-2-ylpyrazol-3-yl]pyridin-2-amine
Show/Hide
|
C20H29N5O2
|
1
|
| 1 |
Ki = 142 nM
|
|
|
|
CP0088424
|
5-[5-[1-(oxetan-3-yl)piperidin-4-yl]-1-propan-2-ylpyrazol-3-yl]-3-(trifluoromethyl)pyridin-2-amine
Show/Hide
|
C20H26F3N5O
|
1
|
| 1 |
Ki = 154 nM
|
|
|
|
CP0088423
|
3-chloro-5-[5-[1-(oxetan-3-yl)piperidin-4-yl]-1-propan-2-ylpyrazol-3-yl]pyridin-2-amine
Show/Hide
|
C19H26ClN5O
|
1
|
| 1 |
Ki = 1000 nM
|
|
|
|
CP0332420
|
3-methyl-5-[5-[1-(oxetan-3-yl)piperidin-4-yl]-1-propan-2-ylpyrazol-3-yl]pyridin-2-amine
Show/Hide
|
C20H29N5O
|
1
|
| 1 |
Ki > 1600 nM
|
|
|
