Brief Information of the Cell Line and Protein
Cell Line ID: CL000886 , HL60/MRP
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0002
Protein ID: PT02516 , Multidrug resistance-associated protein 1
Gene Name ABCC1
Organism Homo sapiens, Human
Protein Classification Transporter
Uniprot ID P33527
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000886  Protein ID: PT02516
 
Compound ID Compound Name Compound Formula
CP0248788
SCHISANTHERIN A
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C29H30O9
 3
1
IC50 = 6.315185 nM
   TI
   LI
   LO
   TS
2
IC50 = 162.66386 nM
   TI
   LI
   LO
   TS
3
IC50 = 1636.207062 nM
   TI
   LI
   LO
   TS
CP0109652
SCHISANDRIN A
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C24H32O6
 3
1
IC50 = 6.962618 nM
   TI
   LI
   LO
   TS
2
IC50 = 153.657775 nM
   TI
   LI
   LO
   TS
3
IC50 = 2336.078365 nM
   TI
   LI
   LO
   TS
CP0109568
SCHIZANDRIN
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C24H32O7
 3
1
IC50 = 8.092298 nM
   TI
   LI
   LO
   TS
2
IC50 = 217.336015 nM
   TI
   LI
   LO
   TS
3
IC50 = 3239.231463 nM
   TI
   LI
   LO
   TS
CP0036379
GOMISIN A
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C23H28O7
 3
1
IC50 = 9.36442 nM
   TI
   LI
   LO
   TS
2
IC50 = 182.486133 nM
   TI
   LI
   LO
   TS
3
IC50 = 2763.704469 nM
   TI
   LI
   LO
   TS
CP0287511
3,4,5,19-tetramethoxy-9,10-dimethyl-15,17-dioxatetracyclo[10.7.0.02,7.014,18]nonadeca-1(19),2,4,6,12,14(18)-hexaene
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C23H28O6
 3
1
IC50 = 9.488851 nM
   TI
   LI
   LO
   TS
2
IC50 = 204.759408 nM
   TI
   LI
   LO
   TS
3
IC50 = 2249.856419 nM
   TI
   LI
   LO
   TS