Brief Information of the Cell Line and Protein
Cell Line ID: CL000352 , HL-60/ADR
Synonyms
HL60/ADR
HL60/Adr
HL60-ADR
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0304
Protein ID: PT02516 , Multidrug resistance-associated protein 1
Gene Name ABCC1
Organism Homo sapiens, Human
Protein Classification Transporter
Uniprot ID P33527
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000352  Protein ID: PT02516
 
Compound ID Compound Name Compound Formula
CP0248788
SCHISANTHERIN A
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C29H30O9
 3
1
IC50 = 0.765477 nM
   TI
   LI
   LO
   TS
2
IC50 = 110.994163 nM
   TI
   LI
   LO
   TS
3
IC50 = 3056.166874 nM
   TI
   LI
   LO
   TS
CP0036379
GOMISIN A
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C23H28O7
 3
1
IC50 = 0.960453 nM
   TI
   LI
   LO
   TS
2
IC50 = 122.4578 nM
   TI
   LI
   LO
   TS
3
IC50 = 7772.468605 nM
   TI
   LI
   LO
   TS
CP0109568
SCHIZANDRIN
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C24H32O7
 3
1
IC50 = 1.156043 nM
   TI
   LI
   LO
   TS
2
IC50 = 124.852605 nM
   TI
   LI
   LO
   TS
3
IC50 = 7248.387321 nM
   TI
   LI
   LO
   TS
CP0287511
3,4,5,19-tetramethoxy-9,10-dimethyl-15,17-dioxatetracyclo[10.7.0.02,7.014,18]nonadeca-1(19),2,4,6,12,14(18)-hexaene
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C23H28O6
 3
1
IC50 = 1.248533 nM
   TI
   LI
   LO
   TS
2
IC50 = 139.835693 nM
   TI
   LI
   LO
   TS
3
IC50 = 4185.082528 nM
   TI
   LI
   LO
   TS
CP0109652
SCHISANDRIN A
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C24H32O6
 3
1
IC50 = 9.843701 nM
   TI
   LI
   LO
   TS
2
IC50 = 141.653262 nM
   TI
   LI
   LO
   TS
3
IC50 = 4888.237977 nM
   TI
   LI
   LO
   TS