Compound ID |
Compound Name |
Compound Formula |
CP0573769
|
(2R)-N-(1H-indazol-4-yl)-1-[1-(4-methoxyphenyl)cyclohexanecarbonyl]pyrrolidine-2-carboxamide
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|
C26H30N4O3
|
1
|
1 |
IC50 = 420 nM
|
|
|
CP0574532
|
(4S)-N-(1H-indazol-4-yl)-3-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-1,1-dioxo-1,3-thiazolidine-4-carboxamide
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|
C24H26N4O5S
|
1
|
1 |
IC50 = 450 nM
|
|
|
CP0579345
|
(2R,4R)-4-fluoro-N-(1H-indazol-4-yl)-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]pyrrolidine-2-carboxamide
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|
C25H27FN4O3
|
1
|
1 |
IC50 = 460 nM
|
|
|
CP0571169
|
[6-(1H-indazol-4-ylmethyl)-1,4-oxazepan-4-yl]-[1-(4-methoxyphenyl)cyclohexyl]methanone
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|
C27H33N3O3
|
1
|
1 |
IC50 = 610 nM
|
|
|
CP0573770
|
(2R)-N-(1H-indazol-4-yl)-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]pyrrolidine-2-carboxamide
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|
C25H28N4O3
|
1
|
1 |
IC50 = 690 nM
|
|
|
CP0570129
|
N-[2-(1H-indazol-4-ylamino)-2-oxoethyl]-1-(4-methoxyphenyl)-N-methylcyclohexane-1-carboxamide
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|
C24H28N4O3
|
1
|
1 |
IC50 = 1010 nM
|
|
|
CP0577523
|
(2R,4R)-4-hydroxy-N-(1H-indazol-4-yl)-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]pyrrolidine-2-carboxamide
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|
C25H28N4O4
|
1
|
1 |
IC50 = 1030 nM
|
|
|
CP0576758
|
(2R,4S)-4-hydroxy-N-(1H-indazol-4-yl)-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]pyrrolidine-2-carboxamide
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|
C25H28N4O4
|
1
|
1 |
IC50 = 1450 nM
|
|
|
CP0576361
|
[6-(1H-indazol-4-ylmethyl)-1,4-oxazepan-4-yl]-[4-(4-methoxyphenyl)oxan-4-yl]methanone
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|
C26H31N3O4
|
1
|
1 |
IC50 = 2240 nM
|
|
|
CP0572251
|
N-[(2R)-1-(1H-indazol-4-ylamino)-1-oxopropan-2-yl]-1-(4-methoxyphenyl)-N-methylcyclopentane-1-carboxamide
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|
C24H28N4O3
|
1
|
1 |
IC50 = 5020 nM
|
|
|