Brief Information of the Compound and Protein
Compound Name
(2R,4S)-4-hydroxy-N-(1H-indazol-4-yl)-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]pyrrolidine-2-carboxamide
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PubChem ID
CID: 168271390
Canonical SMILES
COc1ccc(cc1)C1(CCCC1)C(=O)N1C[C@@H](O)C[C@@H]1C(=O)Nc1cccc2[nH]ncc12
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Compound Formula C25H28N4O4
Compound Structure
Protein Name
Histone acetyltransferase p300
Protein Classification
Epigenetic regulator
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Bromodomain
Uniprot ID
Q09472
Gene Name
EP300
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000715 LK2 Homo sapiens (Human)  1
1
IC50 = 1450 nM
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