Brief Information of the Compound and Protein
Compound Name
(4S)-N-(1H-indazol-4-yl)-3-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-1,1-dioxo-1,3-thiazolidine-4-carboxamide
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Canonical SMILES
COc1ccc(cc1)C1(CCCC1)C(=O)N1CS(=O)(=O)C[C@@H]1C(=O)Nc1cccc2[nH]ncc12
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Compound Formula C24H26N4O5S
Compound Structure
Protein Name
Histone acetyltransferase p300
Protein Classification
Epigenetic regulator
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Bromodomain
Uniprot ID
Q09472
Gene Name
EP300
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000715 LK2 Homo sapiens (Human)  1
1
IC50 = 450 nM
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