Brief Information of the Cell Line and Protein
Cell Line ID: CL000100 , U-937
Synonyms
U937
U 937
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0007
Protein ID: PT01801 , Leukotriene B4 receptor 1
Gene Name LTB4R
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID Q15722
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000100  Protein ID: PT01801
 
Compound ID Compound Name Compound Formula
CP0044090
7-[3-(4-Acetyl-3-methoxy-2-propyl-phenoxy)-propoxy]-8-propyl-chroman-2-carboxylic acid
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C28H36O7
 1
1
Ki = 220 nM
   TI
   LI
   LO
   TS
CP0041794
(E)-3-{3-(2-Carboxy-ethyl)-4-[6-(4-methoxy-phenyl)-hex-5-enyloxy]-benzoyl}-benzoic acid
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C30H30O7
 1
1
Ki = 360 nM
   TI
   LI
   LO
   TS
CP0554918
4-[4-(2-Amino-5-benzyl-1-methyl-1H-imidazol-4-ylmethyl)-phenyl]-butan-1-ol
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C22H27N3O
 1
1
Ki = 2400 nM
   TI
   LI
   LO
   TS
CP0468064
4,5-Bis-benzo[1,3]dioxol-5-ylmethyl-1-methyl-1H-imidazol-2-ylamine
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C20H19N3O4
 1
1
Ki = 3500 nM
   TI
   LI
   LO
   TS
CP0374374
4,5-Dibenzyl-1H-imidazol-2-ylamine
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C17H17N3
 1
1
Ki = 9000 nM
   TI
   LI
   LO
   TS
CP0540927
4,5-Dibenzyl-1-methyl-1H-imidazol-2-ylamine
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C18H19N3
 1
1
Ki = 19000 nM
   TI
   LI
   LO
   TS
CP0464954
5-Benzyl-4-(3-methoxy-benzyl)-1-methyl-1H-imidazol-2-ylamine
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C19H21N3O
 1
1
Ki = 27000 nM
   TI
   LI
   LO
   TS