| Compound ID |
Compound Name |
Compound Formula |
|
CP0039984
|
CGP 71683
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|
C26H29N5O2S
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
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CP0431012
|
N-[[4-[[(4-aminoquinazolin-2-yl)amino]methyl]cyclohexyl]methyl]-4-bromo-2-(trifluoromethoxy)benzenesulfonamide
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|
C23H25BrF3N5O3S
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0404813
|
4-Bromo-N-{4-[(4-dimethylamino-quinazolin-2-ylamino)-methyl]-cyclohexyl}-2-trifluoromethoxy-benzenesulfonamide
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|
C24H27BrF3N5O3S
|
1
|
| 1 |
IC50 = 2.5 nM
|
|
|
|
CP0871069
|
4-Bromo-N-{4-[(4-dimethylamino-quinazolin-2-ylamino)-methyl]-cyclohexylmethyl}-2-trifluoromethoxy-benzenesulfonamide hydrochloride
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|
C25H30BrClF3N5O3S
|
1
|
| 1 |
IC50 = 2.7 nM
|
|
|
|
CP0404808
|
4-Bromo-N-{4-[(4-dimethylamino-quinazolin-2-ylamino)-methyl]-cyclohexylmethyl}-2-trifluoromethoxy-benzenesulfonamide
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|
C25H29BrF3N5O3S
|
1
|
| 1 |
IC50 = 2.7 nM
|
|
|
|
CP0466919
|
Butane-1-sulfonic acid {4-[(4-dimethylamino-quinazolin-2-ylamino)-methyl]-cyclohexylmethyl}-amide
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|
C22H35N5O2S
|
1
|
| 1 |
IC50 = 4.9 nM
|
|
|
|
CP0495240
|
4-Bromo-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-2-trifluoromethoxy-benzenesulfonamide
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|
C23H25BrF3N5O3S
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0493156
|
N-[[4-[[[4-(dimethylamino)quinazolin-2-yl]amino]methyl]cyclohexyl]methyl]methanesulfonamide
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|
C19H29N5O2S
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
|
CP0404811
|
4-Bromo-N-[4-(quinazolin-2-ylaminomethyl)-cyclohexylmethyl]-2-trifluoromethoxy-benzenesulfonamide
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|
C23H24BrF3N4O3S
|
1
|
| 1 |
IC50 = 78 nM
|
|
|
|
CP0378340
|
4-Bromo-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexylmethyl]-2-trifluoromethoxy-benzenesulfonamide
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|
C24H27BrF3N5O3S
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0409350
|
4-Bromo-N-[4-(quinazolin-2-ylamino)-cyclohexylmethyl]-2-trifluoromethoxy-benzenesulfonamide
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|
C22H22BrF3N4O3S
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0431015
|
4-Bromo-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexylmethyl]-2-trifluoromethoxy-benzenesulfonamide
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|
C24H27BrF3N5O3S
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0494619
|
4-bromo-N-[[4-[[[4-(dimethylamino)quinazolin-2-yl]amino]methyl]cyclohexyl]methyl]-N-methyl-2-(trifluoromethoxy)benzenesulfonamide
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|
C26H31BrF3N5O3S
|
1
|
| 1 |
IC50 = 460 nM
|
|
|
|
CP0500756
|
4-bromo-N-[[4-[[[4-(dimethylamino)quinazolin-2-yl]amino]methyl]cyclohexyl]methyl]-2-(trifluoromethoxy)benzamide
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|
C26H29BrF3N5O2
|
1
|
| 1 |
IC50 = 470 nM
|
|
|
|
CP0464467
|
2-N-[[4-[[[4-bromo-2-(trifluoromethoxy)phenyl]methylamino]methyl]cyclohexyl]methyl]-4-N,4-N-dimethylquinazoline-2,4-diamine
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|
C26H31BrF3N5O
|
1
|
| 1 |
IC50 = 560 nM
|
|
|
|
CP0392292
|
4-Bromo-N-[4-(4-dimethylamino-quinazolin-2-ylamino)-cyclohexyl]-2-trifluoromethoxy-benzenesulfonamide
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|
C23H25BrF3N5O3S
|
1
|
| 1 |
IC50 = 880 nM
|
|
|
|
CP0409351
|
4-Bromo-N-[4-(quinazolin-2-ylamino)-cyclohexyl]-2-trifluoromethoxy-benzenesulfonamide
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|
C21H20BrF3N4O3S
|
1
|
| 1 |
IC50 = 880 nM
|
|
|
|
CP0436964
|
4-bromo-N-[[4-[[4-(dimethylamino)quinazolin-2-yl]amino]cyclohexyl]methyl]-2-(trifluoromethoxy)benzamide
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|
C25H27BrF3N5O2
|
1
|
| 1 |
IC50 = 1800 nM
|
|
|
|
CP0431371
|
2-N-[4-[[[4-bromo-2-(trifluoromethoxy)phenyl]methylamino]methyl]cyclohexyl]-4-N,4-N-dimethylquinazoline-2,4-diamine
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|
C25H29BrF3N5O
|
1
|
| 1 |
IC50 = 2400 nM
|
|
|
|
CP0043469
|
ATC0175
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|
C23H25F2N5O
|
1
|
| 1 |
IC50 = 2700 nM
|
|
|
|
CP0503845
|
2-N-[[1-[4-bromo-2-(trifluoromethoxy)phenyl]sulfonylpiperidin-4-yl]methyl]-4-N,4-N-dimethylquinazoline-2,4-diamine
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|
C23H25BrF3N5O3S
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
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CP0440289
|
2-N-[1-[4-bromo-2-(trifluoromethoxy)phenyl]sulfonylpiperidin-4-yl]-4-N,4-N-dimethylquinazoline-2,4-diamine
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|
C22H23BrF3N5O3S
|
1
|
| 1 |
IC50 = 8900 nM
|
|
|
|
CP0379328
|
2-N-[4-[[4-bromo-2-(trifluoromethoxy)phenyl]methylamino]cyclohexyl]-4-N,4-N-dimethylquinazoline-2,4-diamine
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|
C24H27BrF3N5O
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0392299
|
4-bromo-N-[4-[[4-(dimethylamino)quinazolin-2-yl]amino]cyclohexyl]-2-(trifluoromethoxy)benzamide
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|
C24H25BrF3N5O2
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
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CP0392533
|
2-N-[[4-[[[4-bromo-2-(trifluoromethoxy)phenyl]methyl-methylamino]methyl]cyclohexyl]methyl]-4-N,4-N-dimethylquinazoline-2,4-diamine
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|
C27H33BrF3N5O
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
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CP0424935
|
2-N-[1-[[4-bromo-2-(trifluoromethoxy)phenyl]methyl]piperidin-4-yl]-4-N,4-N-dimethylquinazoline-2,4-diamine
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|
C23H25BrF3N5O
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
