Brief Information of the Compound and Protein
Compound Name
CGP 71683
    Show/Hide
PubChem ID
SID: 24739773
Canonical SMILES
Nc1nc(NC[C@H]2CC[C@H](CNS(=O)(=O)c3cccc4ccccc34)CC2)nc2ccccc12
    Show/Hide
Compound Formula C26H29N5O2S
Compound Structure
Protein Name
Neuropeptide Y receptor type 5
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
>
Short peptide receptor (family A GPCR)
>
Neuropeptide Y receptor
Uniprot ID
Q15761
Gene Name
NPY5R
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000109 COS-1 Chlorocebus aethiops (Green monkey)  1
1
IC50 = 1.3 nM
   TI
   LI
   LO
   TS
CL000101 L-M(TK-) Mus musculus (Mouse)  1
1
IC50 = 2.9 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 2.9 nM