Brief Information of the Cell Line and Protein
Cell Line ID: CL000026 , CHO-K1
Synonyms
CHO K1
CHOK1
CHO cell clone K1
GM15452
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_0214
Protein ID: PT01711 , Histamine H4 receptor
Gene Name HRH4
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID Q9H3N8
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000026  Protein ID: PT01711
 
Compound ID Compound Name Compound Formula
CP0041262
5-chloro-2-[(4-methylpiperazin-1-yl)carbonyl]-1H-indole
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C14H16ClN3O
 1
1
IC50 = 13 nM
   TI
   LI
   LO
   TS
CP0044460
N-cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide
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C15H24N4S
 1
1
IC50 = 19 nM
   TI
   LI
   LO
   TS
CP0390721
4-(cyclohexylmethyl)-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine
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C15H26N6
 1
1
IC50 = 32 nM
   TI
   LI
   LO
   TS
CP0430105
4-(4-methylpiperazin-1-yl)-6-propyl-1,3,5-triazin-2-amine
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C11H20N6
 1
1
IC50 = 265 nM
   TI
   LI
   LO
   TS
CP0262529
diethyl 2,6-dimethyl-4-[4-(5-piperidin-1-ylpentoxy)phenyl]-1,4-dihydropyridine-3,5-dicarboxylate
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C29H42N2O5
 1
1
IC50 = 1400 nM
   TI
   LI
   LO
   TS
CP0092861
2-(2-(4-tert-Butylphenylthio)ethyl)-1H-imidazole
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C15H20N2S
 1
1
Ki = 1.1 nM
   TI
   LI
   LO
   TS
CP0110239
4-(1H-imidazol-4-ylmethyl)piperidine
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C9H15N3
 1
1
Ki = 22 nM
   TI
   LI
   LO
   TS
CP0438775
4-((1H-Imidazol-4-yl)methyl)-1-(4-(trifluoromethyl)-phenyl)piperidine
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C16H18F3N3
 1
1
Ki = 216 nM
   TI
   LI
   LO
   TS
CP0400519
4-((1H-Imidazol-4-yl)methyl)-1-(4-methoxyphenyl)piperidine
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C16H21N3O
 1
1
Ki = 3100 nM
   TI
   LI
   LO
   TS