| Compound ID |
Compound Name |
Compound Formula |
|
CP0357968
|
CHEBI:77317
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C24H42O7P2
|
1
|
| 1 |
EC50 = 80 nM
|
|
|
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CP0003740
|
N-[4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)phenyl]-N-(2,2,2-trifluoroethyl)benzenesulfonamide
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C17H12F9NO3S
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
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CP0053566
|
N-[5-(2-chlorobenzoyl)-4-(3-chlorophenyl)-1,3-thiazol-2-yl]-2-(4-ethylsulfonylphenyl)acetamide
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|
C26H20Cl2N2O4S2
|
1
|
| 1 |
EC50 = 260 nM
|
|
|
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CP0385671
|
N-[4-[hydroxy(dimethyl)silyl]phenyl]-N-(2,2,2-trifluoroethyl)benzenesulfonamide
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C16H18F3NO3SSi
|
1
|
| 1 |
EC50 = 630 nM
|
|
|
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CP0389947
|
methyl 2-[N-(benzenesulfonyl)-4-[hydroxy(dimethyl)silyl]anilino]acetate
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C17H21NO5SSi
|
1
|
| 1 |
EC50 = 1400 nM
|
|
|
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CP0466299
|
N-ethyl-N-[4-[hydroxy(dimethyl)silyl]phenyl]benzenesulfonamide
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|
C16H21NO3SSi
|
1
|
| 1 |
EC50 = 1900 nM
|
|
|
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CP0071702
|
BA-41166E
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|
C43H58N4O12
|
1
|
| 1 |
EC50 = 2000 nM
|
|
|
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CP0138637
|
3-[(2S)-6-[(E)-2-[2-chloro-6-(trifluoromethyl)phenyl]ethenyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
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|
C27H20ClF6NO5S
|
1
|
| 1 |
EC50 = 2000 nM
|
|
|
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CP0396596
|
N-[4-[hydroxy(dimethyl)silyl]phenyl]benzenesulfonamide
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|
C14H17NO3SSi
|
1
|
| 1 |
EC50 = 2400 nM
|
|
|
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CP0396600
|
N-benzyl-N-[4-[hydroxy(dimethyl)silyl]phenyl]benzenesulfonamide
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|
C21H23NO3SSi
|
1
|
| 1 |
EC50 = 3200 nM
|
|
|
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CP0396598
|
N-[4-[hydroxy(dimethyl)silyl]phenyl]-N-methylbenzenesulfonamide
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|
C15H19NO3SSi
|
1
|
| 1 |
EC50 = 3400 nM
|
|
|
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CP0389948
|
N-[4-[hydroxy(dimethyl)silyl]phenyl]-N-(2-methoxyethyl)benzenesulfonamide
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|
C17H23NO4SSi
|
1
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| 1 |
EC50 = 4200 nM
|
|
|
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CP0534098
|
3-[(2S)-6-[(E)-2-(2-methylphenyl)prop-1-enyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
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|
C28H26F3NO5S
|
1
|
| 1 |
EC50 = 5000 nM
|
|
|
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CP0420013
|
3-[[(2S)-6-[3-(difluoromethoxy)-5-fluorophenyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]methyl]oxetane-3-carboxylic acid
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|
C27H21F6NO7S
|
1
|
| 1 |
EC50 = 5460 nM
|
|
|
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CP0550332
|
3-[(2S)-6-[(E)-2-(2-chloro-6-fluorophenyl)prop-1-enyl]-4-[4-fluoro-3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
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|
C27H21ClF5NO5S
|
1
|
| 1 |
EC50 = 6000 nM
|
|
|
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CP0390984
|
N-butyl-N-[4-[hydroxy(dimethyl)silyl]phenyl]benzenesulfonamide
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|
C18H25NO3SSi
|
1
|
| 1 |
EC50 = 6500 nM
|
|
|
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CP0552371
|
3-[(2S)-6-[(E)-2-(2-chloro-6-fluorophenyl)prop-1-enyl]-4-(3-cyclopropyl-4-fluorophenyl)sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
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|
C29H26ClF2NO5S
|
1
|
| 1 |
EC50 = 6700 nM
|
|
|
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CP0060756
|
3-[(2S)-6-[3-(difluoromethoxy)-5-fluorophenyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]-2,2-dimethylpropanoic acid
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|
C27H23F6NO6S
|
1
|
| 1 |
EC50 = 8000 nM
|
|
|
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CP0471271
|
3-[(2S)-6-[(E)-2-(2-chloro-6-fluorophenyl)prop-1-enyl]-4-[3-(difluoromethoxy)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
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|
C27H23ClF3NO6S
|
1
|
| 1 |
EC50 = 9100 nM
|
|
|
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CP0138557
|
3-[(2S)-6-[(E)-2-(2-chloro-6-fluorophenyl)prop-1-enyl]-4-[[2-(2-hydroxyethoxy)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl]sulfonyl]-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
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|
C29H31ClFN3O7S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0138560
|
4-[[(2S)-6-(3-chloro-2-fluorophenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]methyl]oxane-4-carboxylic acid
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|
C28H24ClF4NO6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0138638
|
3-[(2S)-6-(4-propan-2-ylphenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
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|
C27H26F3NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0138639
|
3-[(2S)-6-[(E)-2-(2-methoxyphenyl)prop-1-enyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
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|
C28H26F3NO6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0189594
|
3-[(2S)-6-[(E)-2-(2-chlorophenyl)prop-1-enyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
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|
C27H23ClF3NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0189596
|
3-[(2S)-6-[(E)-2-(2-chloro-6-fluorophenyl)prop-1-enyl]-4-[(2-ethoxy-4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)sulfonyl]-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
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|
C29H31ClFN3O6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0351090
|
(2R)-3-[(2S)-6-(2,5-difluorophenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]-2-methylpropanoic acid
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|
C25H20F5NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0420011
|
3-[(2S)-6-[3-(difluoromethoxy)-5-fluorophenyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
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|
C25H19F6NO6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0471263
|
3-[(2S)-6-[(E)-2-(2-chloro-6-fluorophenyl)prop-1-enyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C27H22ClF4NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0471264
|
(2S)-4-[(2S)-6-(2,5-difluorophenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]-2-hydroxybutanoic acid
Show/Hide
|
C25H20F5NO6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0471267
|
3-[(2S)-6-(3-methoxyphenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C25H22F3NO6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0471268
|
3-[(2S)-6-(2-chloro-3,5-difluorophenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C24H17ClF5NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0471273
|
3-[(2S)-6-(2,5-difluorophenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]-2,2-dimethylpropanoic acid
Show/Hide
|
C26H22F5NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0487451
|
3-[(2S)-6-(3-chloro-2-fluorophenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]-2,2-dimethylpropanoic acid
Show/Hide
|
C26H22ClF4NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0487452
|
3-[(2S)-6-[(E)-2-(2-chloro-6-fluorophenyl)prop-1-enyl]-4-(4-fluoro-3-methoxyphenyl)sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C27H24ClF2NO6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0527539
|
4-[[(2S)-6-(2,5-difluorophenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]methyl]oxane-4-carboxylic acid
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|
C28H24F5NO6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0527541
|
3-[(2S)-6-[(E)-2-(2,6-dichlorophenyl)prop-1-enyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C27H22Cl2F3NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0534099
|
3-[(2S)-6-(2,5-difluorophenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C24H18F5NO5S
|
1
|
| 1 |
EC50 > 10000 nM
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|
|
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CP0534360
|
3-[(2S)-6-[(E)-2-phenylprop-1-enyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C27H24F3NO5S
|
1
|
| 1 |
EC50 > 10000 nM
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|
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CP0539745
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3-[(2S)-6-(3-fluorophenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
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|
C24H19F4NO5S
|
1
|
| 1 |
EC50 > 10000 nM
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|
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CP0546382
|
3-[(2S)-6-[(E)-2-(4-methylphenyl)ethenyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C27H24F3NO5S
|
1
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| 1 |
EC50 > 10000 nM
|
|
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CP0546383
|
3-[(2S)-6-(3-chlorophenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C24H19ClF3NO5S
|
1
|
| 1 |
EC50 > 10000 nM
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|
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CP0546458
|
3-[(2S)-6-[3-(2-hydroxyethoxy)phenyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C26H24F3NO7S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0546643
|
3-[(2S)-6-[(E)-2-(4-chloro-2-fluorophenyl)ethenyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C26H20ClF4NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0549139
|
3-[(2S)-6-(3,5-difluorophenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C24H18F5NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0550333
|
3-[(2S)-6-[(E)-2-(2-chloro-6-fluorophenyl)ethenyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C26H20ClF4NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0552370
|
(2R)-4-[(2S)-6-(2,5-difluorophenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]-2-hydroxybutanoic acid
Show/Hide
|
C25H20F5NO6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0552372
|
3-[(2S)-6-[(E)-2-[2-(trifluoromethyl)phenyl]prop-1-enyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C28H23F6NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0552378
|
3-[(2S)-6-(2-chloro-5-fluorophenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C24H18ClF4NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0552379
|
3-[(2S)-6-(3-fluoro-5-methoxyphenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C25H21F4NO6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0552384
|
3-[(2S)-6-(2-chlorophenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C24H19ClF3NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0553547
|
3-[(2S)-6-(2-chloro-3-fluorophenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C24H18ClF4NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0557795
|
(2S)-3-[(2S)-6-(2,5-difluorophenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]-2-methylpropanoic acid
Show/Hide
|
C25H20F5NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0562991
|
[3-[[(2S)-6-bromo-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]methyl]oxetan-3-yl]methanol
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|
C20H19BrF3NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0564257
|
3-[(2S)-6-[3-(difluoromethoxy)phenyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
Show/Hide
|
C25H20F5NO6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0534361
|
4-[[(2S)-6-[3-(difluoromethoxy)-5-fluorophenyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]methyl]oxane-4-carboxylic acid
Show/Hide
|
C29H25F6NO7S
|
1
|
| 1 |
EC50 = 13000 nM
|
|
|
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CP0396599
|
N-[4-[hydroxy(dimethyl)silyl]phenyl]-N-(2-phenylethyl)benzenesulfonamide
Show/Hide
|
C22H25NO3SSi
|
1
|
| 1 |
EC50 = 14000 nM
|
|
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CP0471269
|
3-[[(2S)-6-(2,5-difluorophenyl)-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]methyl]oxetane-3-carboxylic acid
Show/Hide
|
C26H20F5NO6S
|
1
|
| 1 |
EC50 = 18000 nM
|
|
|
