General Information of the Compound
Compound ID
CP0564257
Compound Name
3-[(2S)-6-[3-(difluoromethoxy)phenyl]-4-[3-(trifluoromethyl)phenyl]sulfonyl-2,3-dihydro-1,4-benzoxazin-2-yl]propanoic acid
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Structure
Formula
C25H20F5NO6S
Molecular Weight
557.493
Canonical SMILES
OC(=O)CC[C@H]1CN(c2cc(ccc2O1)-c1cccc(OC(F)F)c1)S(=O)(=O)c1cccc(c1)C(F)(F)F
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InChI
InChI=1S/C25H20F5NO6S/c26-24(27)37-18-5-1-3-15(11-18)16-7-9-22-21(12-16)31(14-19(36-22)8-10-23(32)33)38(34,35)20-6-2-4-17(13-20)25(28,29)30/h1-7,9,11-13,19,24H,8,10,14H2,(H,32,33)/t19-/m0/s1
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InChIKey
UZTBXPPLLTXTNE-IBGZPJMESA-N
Physicochemical Property
logP
5.7949
Rotatable Bonds
8
Heavy Atom Count
38
Polar Areas
93.14
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
5
Complexity
38

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 124133617
ChEMBL ID
CHEMBL4859796
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT02663, Nuclear receptor ROR-gamma
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000013 Sf9 Spodoptera frugiperda (Fall armyworm)  1
1
EC50 = 10 nM
   TI
   LI
   LO
   TS
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 278 nM
   TI
   LI
   LO
   TS
Protein ID: PT01552, Nuclear receptor subfamily 1 group I member 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS