| Compound ID |
Compound Name |
Compound Formula |
|
CP0491864
|
US9394273, 15
Show/Hide
|
C26H26O4S
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0418279
|
US9394273, 7
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|
C24H25ClO4
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0529357
|
US9394273, 18
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|
C29H30O5
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0384076
|
US9394273, 16
Show/Hide
|
C29H30O5
|
1
|
| 1 |
EC50 = 728 nM
|
|
|
|
CP0847236
|
5-{(R)-1-[4-(1-Hydroxy-hexyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-thiophene-2-carboxylic acid
Show/Hide
|
C23H29NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0847237
|
5-{3-[(S)-1-(4-Hexanoyl-phenyl)-5-oxo-pyrrolidin-2-yl]-propyl}-thiophene-2-carboxylic acid
Show/Hide
|
C24H29NO4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0847239
|
5-{(R)-1-[4-(1-Hydroxy-propyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-thiophene-2-carboxylic acid
Show/Hide
|
C20H23NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0847241
|
3-[(R)-1-(4-tert-Butyl-phenyl)-5-oxo-pyrrolidin-2-ylmethoxymethyl]-benzoic acid
Show/Hide
|
C23H27NO4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0847242
|
5-[(R)-1-(4-tert-Butyl-phenyl)-5-oxo-pyrrolidin-2-ylmethoxymethyl]-thiophene-2-carboxylic acid
Show/Hide
|
C21H25NO4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0866241
|
5-(3-{(S)-1-[4-(1-Hydroxy-heptyl)-phenyl]-5-oxo-pyrrolidin-2-yl}-propyl)-thiophene-2-carboxylic acid
Show/Hide
|
C25H33NO4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0866744
|
7-[(S)-1-(4-tert-Butyl-phenyl)-5-oxo-pyrrolidin-2-yl]-heptanoic acid
Show/Hide
|
C21H31NO3
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0870431
|
5-(3-{(S)-1-[4-(1-Hydroxy-hexyl)-phenyl]-5-oxo-pyrrolidin-2-yl}-propyl)-thiophene-2-carboxylic acid
Show/Hide
|
C24H31NO4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0883084
|
5-[(R)-1-(4-tert-Butyl-phenyl)-5-oxo-pyrrolidin-2-ylmethoxy]-pentanoic acid
Show/Hide
|
C20H29NO4
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0885328
|
5-[(R)-1-(4-tert-Butyl-phenyl)-5-oxo-pyrrolidin-2-ylmethoxymethyl]-furan-2-carboxylic acid
Show/Hide
|
C21H25NO5
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0055947
|
(15S)-prostaglandin E2
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|
C20H32O5
|
1
|
| 1 |
IC50 = 0.7 nM
|
|
|
|
CP0381433
|
(R)-5-((E)-(S)-3-Hydroxy-4-phenyl-but-1-enyl)-1-[6-(1H-tetrazol-5-yl)-hexyl]-pyrrolidin-2-one
Show/Hide
|
C21H29N5O2
|
2
|
| 1 |
IC50 = 1.4 nM
|
|
|
| 2 |
Ki = 1.2 nM
|
|
|
|
CP0202009
|
(2S)-2-[(5-{[4-(3-acetamidophenyl)phenyl]methyl}-1,3-oxazol-4-yl)formamido]-3-phenylpropanoic acid
Show/Hide
|
C28H25N3O5
|
1
|
| 1 |
IC50 = 24000 nM
|
|
|
|
CP0374156
|
4-(1-(1-(4-(trifluoromethyl)benzyl)-1H-indole-7-carboxamido)cyclopropyl)benzoic acid
Show/Hide
|
C27H21F3N2O3
|
2
|
| 1 |
Ki = 0.23 nM
|
|
|
| 2 |
Ki = 0.34 nM
|
|
|
|
CP0437430
|
(S)-4-(1-(1-(biphenyl-4-ylmethyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C31H28N2O3
|
1
|
| 1 |
Ki = 0.28 nM
|
|
|
|
CP0372255
|
4-(1-(5-chloro-1-(4-(trifluoromethyl)benzyl)-1H-indole-7-carboxamido)cyclopropyl)benzoic acid
Show/Hide
|
C27H20ClF3N2O3
|
1
|
| 1 |
Ki = 0.31 nM
|
|
|
|
CP0379617
|
(S)-4-(1-(1-(3,5-dibromobenzyl)indoline-7-carboxamido)ethyl)benzoic acid
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|
C25H22Br2N2O3
|
1
|
| 1 |
Ki = 0.33 nM
|
|
|
|
CP0473507
|
(S)-4-(1-(1-(3,4-dichlorobenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C25H22Cl2N2O3
|
1
|
| 1 |
Ki = 0.34 nM
|
|
|
|
CP0393826
|
(S)-4-(1-(1-(4-(trifluoromethyl)benzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H23F3N2O3
|
1
|
| 1 |
Ki = 0.37 nM
|
|
|
|
CP0402997
|
(S)-4-(1-(5-fluoro-1-(4-(trifluoromethyl)benzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H22F4N2O3
|
1
|
| 1 |
Ki = 0.37 nM
|
|
|
|
CP0388650
|
(S)-4-(1-(1-(3-chloro-5-(trifluoromethoxy)benzyl)-1H-indole-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H20ClF3N2O4
|
1
|
| 1 |
Ki = 0.38 nM
|
|
|
|
CP0377873
|
(S)-4-(1-(5-chloro-1-(4-(trifluoromethyl)benzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H22ClF3N2O3
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0380631
|
(S)-4-(1-(1-(3-(trifluoromethyl)benzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H23F3N2O3
|
1
|
| 1 |
Ki = 0.4 nM
|
|
|
|
CP0388647
|
(S)-4-(1-(5-chloro-1-(4-(trifluoromethyl)benzyl)-1H-indole-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H20ClF3N2O3
|
1
|
| 1 |
Ki = 0.44 nM
|
|
|
|
CP0379615
|
(S)-4-(1-(1-(3-chlorobenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C25H23ClN2O3
|
1
|
| 1 |
Ki = 0.44 nM
|
|
|
|
CP0468170
|
(S)-4-(1-(1-(4-chlorobenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C25H23ClN2O3
|
1
|
| 1 |
Ki = 0.44 nM
|
|
|
|
CP0452755
|
4-{1-[({2,5-Dimethyl-4-[4-(trifluoromethyl)benzyl]-3-thienyl}-carbonyl)amino]cyclopropyl}benzoic Acid
Show/Hide
|
C25H22F3NO3S
|
2
|
| 1 |
Ki = 0.56 nM
|
|
|
| 2 |
Ki = 0.97 nM
|
|
|
|
CP0411079
|
(S)-4-(1-(1-(4-(trifluoromethyl)benzyl)-1H-indole-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H21F3N2O3
|
1
|
| 1 |
Ki = 0.62 nM
|
|
|
|
CP0469926
|
US8969394, 14
Show/Hide
|
C25H22F3N5OS
|
1
|
| 1 |
Ki = 0.63 nM
|
|
|
|
CP0508827
|
(S)-4-(1-(5-(trifluoromethyl)-1-(4-(trifluoromethyl)benzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C27H22F6N2O3
|
1
|
| 1 |
Ki = 0.66 nM
|
|
|
|
CP0383780
|
4-[({[2,5-Dichloro-4-(3-chlorobenzyl)-3-thienyl]carbonyl}amino)methyl]benzoic acid
Show/Hide
|
C20H14Cl3NO3S
|
1
|
| 1 |
Ki = 0.72 nM
|
|
|
|
CP0421644
|
4-{1-[({2,5-Dimethyl-4-[3-(trifluoromethyl)benzyl]-3-thienyl}-carbonyl)amino]cyclopropyl}benzoic Acid
Show/Hide
|
C25H22F3NO3S
|
1
|
| 1 |
Ki = 0.75 nM
|
|
|
|
CP0474166
|
(S)-4-(1-(1-(4-methylbenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H26N2O3
|
1
|
| 1 |
Ki = 0.78 nM
|
|
|
|
CP0388649
|
(S)-4-(1-(5-chloro-1-(3-chlorobenzyl)-1H-indole-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C25H20Cl2N2O3
|
1
|
| 1 |
Ki = 0.81 nM
|
|
|
|
CP0383779
|
4-[(1R)-1-({[2,5-Dichloro-4-(3-chlorobenzyl)-3-thienyl]carbonyl}amino)ethyl]benzoic acid
Show/Hide
|
C21H16Cl3NO3S
|
1
|
| 1 |
Ki = 0.87 nM
|
|
|
|
CP0393828
|
(S)-N-(1-(4-(2H-tetrazol-5-yl)phenyl)ethyl)-1-(4-(trifluoromethyl)benzyl)indoline-7-carboxamide
Show/Hide
|
C26H23F3N6O
|
1
|
| 1 |
Ki = 1 nM
|
|
|
|
CP0469928
|
4-[(1S)-1-({[2,5-Dichloro-4-(3-chlorobenzyl)-3-thienyl]carbonyl}-amino)ethyl]benzoic Acid
Show/Hide
|
C21H16Cl3NO3S
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0489160
|
4-{(1S)-1-[({2,5-Dimethyl-4-[4-(trifluoromethyl)benzyl]-3-thienyl}-carbonyl)amino]ethyl}benzoic acid
Show/Hide
|
C24H22F3NO3S
|
1
|
| 1 |
Ki = 1.4 nM
|
|
|
|
CP0380630
|
(S)-4-(1-(1-(4-(trifluoromethoxy)benzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H23F3N2O4
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0477213
|
(S)-4-(1-(1-(4-fluorobenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C25H23FN2O3
|
1
|
| 1 |
Ki = 1.8 nM
|
|
|
|
CP0475979
|
(S)-4-(1-(1-(2-bromo-4-chlorobenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C25H22BrClN2O3
|
1
|
| 1 |
Ki = 2.3 nM
|
|
|
|
CP0372247
|
(S)-4-(1-(1-(3-chlorobenzyl)-5-fluoro-1H-indole-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C25H20ClFN2O3
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
|
CP0847359
|
(R)-5-((E)-(S)-3-Hydroxy-4-phenyl-but-1-enyl)-1-[6-(1H-tetrazol-5-yl)-hexyl]-pyrrolidin-2-one; compound with (R)-5-((E)-(R)-3-hydroxy-4-phenyl-but-1-enyl)-1-[6-(1H-tetrazol-5-yl)-hexyl]-pyrrolidin-2-one
Show/Hide
|
C42H58N10O4
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0447496
|
4-{(1S)-1-[({2,5-Dimethyl-4-[3-(trifluoromethyl)benzyl]-3-thienyl}carbonyl)amino]ethyl}benzoic Acid
Show/Hide
|
C24H22F3NO3S
|
1
|
| 1 |
Ki = 2.5 nM
|
|
|
|
CP0257412
|
7-[(R)-2-((E)-3-Hydroxy-4-phenyl-but-1-enyl)-5-oxo-pyrrolidin-1-yl]-heptanoic acid
Show/Hide
|
C21H29NO4
|
1
|
| 1 |
Ki = 2.6 nM
|
|
|
|
CP0377878
|
(S)-4-(1-(1-(3-chlorobenzyl)-1H-indole-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C25H21ClN2O3
|
1
|
| 1 |
Ki = 2.7 nM
|
|
|
|
CP0447789
|
4-[(1S)-1-({[4-(4-Chlorobenzyl)-2,5-dimethyl-3-thienyl]carbonyl}-amino)ethyl]benzoicAcid
Show/Hide
|
C23H22ClNO3S
|
1
|
| 1 |
Ki = 2.9 nM
|
|
|
|
CP0371889
|
4-[(1S)-1-({[4-(3-Chlorobenzyl)-2,5-dimethyl-3-thienyl]carbonyl}-amino)ethyl]benzoic Acid
Show/Hide
|
C23H22ClNO3S
|
1
|
| 1 |
Ki = 3.1 nM
|
|
|
|
CP0522152
|
(S)-4-(1-(1-(4-cyanobenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H23N3O3
|
1
|
| 1 |
Ki = 3.1 nM
|
|
|
|
CP0378243
|
7-{(R)-2-[(E)-3-Hydroxy-4-(3-methoxymethyl-phenyl)-but-1-enyl]-5-oxo-pyrrolidin-1-yl}-heptanoic acid
Show/Hide
|
C23H33NO5
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0388651
|
(S)-4-(1-(1-(3-(trifluoromethyl)benzyl)-1H-indole-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H21F3N2O3
|
1
|
| 1 |
Ki = 4.8 nM
|
|
|
|
CP0480400
|
7-[(R)-2-((E)-3-Hydroxy-oct-1-enyl)-5-oxo-pyrrolidin-1-yl]-heptanoic acid
Show/Hide
|
C19H33NO4
|
1
|
| 1 |
Ki = 6 nM
|
|
|
|
CP0481524
|
4-[(1S)-1-({[4-(3-Chlorobenzyl)-3-thienyl]carbonyl}amino)ethyl]-benzoic Acid
Show/Hide
|
C21H18ClNO3S
|
1
|
| 1 |
Ki = 6.4 nM
|
|
|
|
CP0393829
|
(S)-4-(1-(1-(2-bromo-4-(trifluoromethyl)benzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H22BrF3N2O3
|
1
|
| 1 |
Ki = 6.7 nM
|
|
|
|
CP0380405
|
(S)-4-(1-(1-(3-cyanobenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H23N3O3
|
1
|
| 1 |
Ki = 7.5 nM
|
|
|
|
CP0084755
|
7-{(R)-2-[(E)-3-Hydroxy-3-(1-phenyl-cyclopropyl)-propenyl]-5-oxo-pyrrolidin-1-yl}-heptanoic acid
Show/Hide
|
C23H31NO4
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0378479
|
2-[4-[(2R)-2-[(E)-3-hydroxy-4-phenylbut-1-enyl]-5-oxopyrrolidin-1-yl]butylsulfanyl]acetic acid
Show/Hide
|
C20H27NO4S
|
1
|
| 1 |
Ki = 13 nM
|
|
|
|
CP0477214
|
(S)-4-(1-(1-(4-tert-butylbenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C29H32N2O3
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0388652
|
(S)-4-(1-(3-chloro-1-(3-chlorobenzyl)-1H-indole-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C25H20Cl2N2O3
|
1
|
| 1 |
Ki = 20.1 nM
|
|
|
|
CP0377110
|
7-[(S)-2-(3-Hydroxy-octyl)-5-oxo-pyrrolidin-1-yl]-heptanoic acid
Show/Hide
|
C19H35NO4
|
1
|
| 1 |
Ki = 28 nM
|
|
|
|
CP0402996
|
(S)-4-(1-(1-(3-carbamoylbenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H25N3O4
|
1
|
| 1 |
Ki = 30 nM
|
|
|
|
CP0474165
|
(S)-4-(1-(1-(4-carbamoylbenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H25N3O4
|
1
|
| 1 |
Ki = 30 nM
|
|
|
|
CP0377281
|
7-[2-(3-Hydroxy-octyl)-5-oxo-pyrrolidin-1-yl]-heptanoic acid
Show/Hide
|
C19H35NO4
|
1
|
| 1 |
Ki = 35 nM
|
|
|
|
CP0372254
|
(S)-4-(1-(1-(3-chlorobenzyl)-3-methyl-1H-indole-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H23ClN2O3
|
1
|
| 1 |
Ki = 39.5 nM
|
|
|
|
CP0468171
|
(S)-4-(1-(1-(4-carboxybenzyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H24N2O5
|
1
|
| 1 |
Ki = 54 nM
|
|
|
|
CP0388648
|
(S)-4-(1-(1-(3-chlorobenzyl)-2-methyl-1H-indole-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C26H23ClN2O3
|
1
|
| 1 |
Ki = 56 nM
|
|
|
|
CP0383825
|
7-[(R)-2-((E)-3-Hydroxy-4-methyl-4-phenyl-pent-1-enyl)-5-oxo-pyrrolidin-1-yl]-heptanoic acid
Show/Hide
|
C23H33NO4
|
1
|
| 1 |
Ki = 62 nM
|
|
|
|
CP0377605
|
(R)-5-((E)-3-Hydroxy-4-phenyl-but-1-enyl)-1-[4-(1H-tetrazol-5-ylmethylsulfanyl)-butyl]-pyrrolidin-2-one
Show/Hide
|
C20H27N5O2S
|
1
|
| 1 |
Ki = 66 nM
|
|
|
|
CP0380632
|
(S)-4-(1-(1-(pyridin-3-ylmethyl)indoline-7-carboxamido)ethyl)benzoic acid
Show/Hide
|
C24H23N3O3
|
1
|
| 1 |
Ki = 76 nM
|
|
|
|
CP0409541
|
7-[(R)-2-((E)-3-Hydroxy-5-phenyl-pent-1-enyl)-5-oxo-pyrrolidin-1-yl]-heptanoic acid
Show/Hide
|
C22H31NO4
|
1
|
| 1 |
Ki = 102 nM
|
|
|
|
CP0381345
|
3-{4-[(R)-2-((E)-3-Hydroxy-4-phenyl-but-1-enyl)-5-oxo-pyrrolidin-1-yl]-butylsulfanyl}-propionic acid
Show/Hide
|
C21H29NO4S
|
1
|
| 1 |
Ki = 140 nM
|
|
|
|
CP0406235
|
(R)-5-((E)-(R)-3-Hydroxy-4-phenyl-but-1-enyl)-1-[6-(1H-tetrazol-5-yl)-hexyl]-pyrrolidin-2-one
Show/Hide
|
C21H29N5O2
|
1
|
| 1 |
Ki = 230 nM
|
|
|
|
CP0377295
|
(R)-5-((E)-3-Hydroxy-4-phenyl-but-1-enyl)-1-[4-(1H-tetrazol-5-ylsulfanyl)-butyl]-pyrrolidin-2-one
Show/Hide
|
C19H25N5O2S
|
1
|
| 1 |
Ki = 243 nM
|
|
|
|
CP0378767
|
methyl 2-[4-[(2R)-2-[(E)-3-hydroxy-4-phenylbut-1-enyl]-5-oxopyrrolidin-1-yl]butylsulfanyl]acetate
Show/Hide
|
C21H29NO4S
|
1
|
| 1 |
Ki = 443 nM
|
|
|
|
CP0377111
|
7-[(R)-2-(3-Hydroxy-octyl)-5-oxo-pyrrolidin-1-yl]-heptanoic acid
Show/Hide
|
C19H35NO4
|
1
|
| 1 |
Ki = 1110 nM
|
|
|
|
CP0377113
|
7-[(S)-2-((E)-3-Hydroxy-oct-1-enyl)-5-oxo-pyrrolidin-1-yl]-heptanoic acid
Show/Hide
|
C19H33NO4
|
1
|
| 1 |
Ki = 1410 nM
|
|
|
|
CP0404807
|
7-[(R)-2-((E)-3-Hydroxy-3-methyl-4-phenyl-but-1-enyl)-5-oxo-pyrrolidin-1-yl]-heptanoic acid
Show/Hide
|
C22H31NO4
|
1
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| 1 |
Ki = 2100 nM
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CP0407744
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7-[(R)-2-((E)-3-Cyclohexyl-3-hydroxy-propenyl)-5-oxo-pyrrolidin-1-yl]-heptanoic acid
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C20H33NO4
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1
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| 1 |
Ki = 3500 nM
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