| Compound ID |
Compound Name |
Compound Formula |
|
CP0450865
|
N-[(2R,3S)-1-[5-[(dimethylamino)methyl]-2-(trifluoromethoxy)anilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(4-fluoro-2-methylphenyl)-3-oxopiperazine-1-carboxamide
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|
C34H36F4N6O4
|
1
|
| 1 |
IC50 = 0.17 nM
|
|
|
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CP0396326
|
N-[(2R,3S)-1-[5-[(dimethylamino)methyl]-2-ethoxyanilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(4-fluorophenyl)piperazine-1-carboxamide
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|
C34H41FN6O3
|
1
|
| 1 |
IC50 = 0.2 nM
|
|
|
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CP0412209
|
N-[(2R,3S)-1-[5-[(dimethylamino)methyl]-2-ethoxyanilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(4-fluoro-2-methylphenyl)-3-oxopiperazine-1-carboxamide
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|
C35H41FN6O4
|
1
|
| 1 |
IC50 = 0.2 nM
|
|
|
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CP0471779
|
N-[(2R,3S)-1-[5-[(dimethylamino)methyl]-2-ethoxyanilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(4-fluorophenyl)-3-oxopiperazine-1-carboxamide
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|
C34H39FN6O4
|
1
|
| 1 |
IC50 = 0.2 nM
|
|
|
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CP0568697
|
N-[(2R,3S)-1-[5-[(dimethylamino)methyl]-2-ethoxyanilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-phenylpiperidine-1-carboxamide
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|
C35H43N5O3
|
1
|
| 1 |
IC50 = 0.2 nM
|
|
|
|
CP0534134
|
N-[(2R,3S)-1-[2-acetyl-5-[(dimethylamino)methyl]anilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(4-fluoro-2-methylphenyl)-3-oxopiperazine-1-carboxamide
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|
C35H39FN6O4
|
1
|
| 1 |
IC50 = 0.24 nM
|
|
|
|
CP0471778
|
N-[(2R,3S)-1-[2-acetyl-5-[(dimethylamino)methyl]anilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(4-fluorophenyl)-3-oxopiperazine-1-carboxamide
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|
C34H37FN6O4
|
1
|
| 1 |
IC50 = 0.31 nM
|
|
|
|
CP0450866
|
N-[(2R,3S)-1-[5-[(dimethylamino)methyl]-2-(trifluoromethoxy)anilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(4-fluorophenyl)-3-oxopiperazine-1-carboxamide
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|
C33H34F4N6O4
|
1
|
| 1 |
IC50 = 0.53 nM
|
|
|
|
CP0408515
|
N-[(2R,3S)-1-[5-[(dimethylamino)methyl]-2-ethoxyanilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(thiophene-2-carbonyl)piperidine-1-carboxamide
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|
C34H41N5O4S
|
1
|
| 1 |
IC50 = 0.58 nM
|
|
|
|
CP0389174
|
4-(cyclobutanecarbonyl)-N-[(2R,3S)-1-[5-[(dimethylamino)methyl]-2-ethoxyanilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]piperidine-1-carboxamide
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|
C34H45N5O4
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
|
CP0486208
|
N-[(2R,3S)-1-[2-acetyl-5-[(dimethylamino)methyl]anilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(thiophene-2-carbonyl)piperidine-1-carboxamide
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|
C34H39N5O4S
|
1
|
| 1 |
IC50 = 0.68 nM
|
|
|
|
CP0412208
|
N-[(2R,3S)-1-[2-acetyl-5-[(dimethylamino)methyl]anilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(cyclobutanecarbonyl)piperidine-1-carboxamide
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|
C34H43N5O4
|
1
|
| 1 |
IC50 = 0.69 nM
|
|
|
|
CP0548218
|
N-[(2R,3S)-1-[5-[(dimethylamino)methyl]-2-ethoxyanilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(3-methylbutanoyl)piperidine-1-carboxamide
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|
C34H47N5O4
|
1
|
| 1 |
IC50 = 0.89 nM
|
|
|
|
CP0571253
|
N-[(2R,3S)-1-[2-acetyl-5-[(dimethylamino)methyl]anilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(2,2-dimethylpropanoyl)piperazine-1-carboxamide
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|
C33H44N6O4
|
1
|
| 1 |
IC50 = 0.98 nM
|
|
|
|
CP0474746
|
N-[(2R,3S)-1-[5-[(dimethylamino)methyl]-2-ethoxyanilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(2-methylpropanoyl)piperidine-1-carboxamide
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|
C33H45N5O4
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0571254
|
N-[(2R,3S)-1-[2-acetyl-5-[(dimethylamino)methyl]anilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(cyclobutanecarbonyl)piperazine-1-carboxamide
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|
C33H42N6O4
|
1
|
| 1 |
IC50 = 1.8 nM
|
|
|
|
CP0396325
|
N-[(2R,3S)-1-[2-acetyl-5-[(dimethylamino)methyl]anilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(2-methylpropanoyl)piperidine-1-carboxamide
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|
C33H43N5O4
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0476993
|
N-[(2R,3S)-1-[5-[(dimethylamino)methyl]-2-ethoxyanilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(1,3-thiazole-2-carbonyl)piperidine-1-carboxamide
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|
C33H40N6O4S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0571255
|
4-(cyclobutanecarbonyl)-N-[(2R,3S)-1-[5-[(dimethylamino)methyl]-2-ethoxyanilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]piperazine-1-carboxamide
Show/Hide
|
C33H44N6O4
|
1
|
| 1 |
IC50 = 2.1 nM
|
|
|
|
CP0471722
|
N-[(2R,3S)-1-[5-[(dimethylamino)methyl]-2-ethoxyanilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(2,2-dimethylpropanoyl)piperazine-1-carboxamide
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|
C33H46N6O4
|
1
|
| 1 |
IC50 = 2.3 nM
|
|
|
|
CP0568698
|
N-[(2R,3S)-1-[5-[(dimethylamino)methyl]-2-ethoxyanilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(furan-2-carbonyl)piperidine-1-carboxamide
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|
C34H41N5O5
|
1
|
| 1 |
IC50 = 2.3 nM
|
|
|
|
CP0412210
|
N-[(2R,3S)-1-[5-[(dimethylamino)methyl]-2-ethoxyanilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(pyridine-2-carbonyl)piperidine-1-carboxamide
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|
C35H42N6O4
|
1
|
| 1 |
IC50 = 2.6 nM
|
|
|
|
CP0568696
|
N-[(2R,3S)-1-[5-[(dimethylamino)methyl]-2-(trifluoromethoxy)anilino]-3-(1H-indol-3-yl)-1-oxobutan-2-yl]-4-(2,2-dimethylpropanoyl)piperazine-1-carboxamide
Show/Hide
|
C32H41F3N6O4
|
1
|
| 1 |
IC50 = 2.8 nM
|
|
|
