Compound ID |
Compound Name |
Compound Formula |
CP0847317
|
2-{(2R,4aR,5R,6R,7aS)-6-hydroxy-5-[(1E,3R)-3-hydroxy-4-phenoxy-1-buten-1-yl]octahydrocyclopenta[b]pyran-2-yl}-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C22H25NO6S
|
1
|
1 |
EC50 = 1.4 nM
|
|
|
CP0055947
|
(15S)-prostaglandin E2
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|
C20H32O5
|
1
|
1 |
EC50 = 3.7 nM
|
|
|
CP0847320
|
2-[(2R,4aR,5R,6R,7aS)-6-hydroxy-5-(2-phenoxyethyl)octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C20H23NO5S
|
1
|
1 |
EC50 = 97 nM
|
|
|
CP0862926
|
2-{(2R,4aR,5R,6R,7aS)-6-hydroxy-5-[(1E)-4-phenoxy-1-buten-1-yl]octahydrocyclopenta[b]pyran-2-yl}-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C22H25NO5S
|
1
|
1 |
EC50 = 160 nM
|
|
|
CP0847318
|
2-{(2R,4aR,5R,6R,7aS)-6-hydroxy-5-[(1E)-3-phenoxy-1-propen-1-yl]octahydrocyclopenta[b]pyran-2-yl}-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C21H23NO5S
|
1
|
1 |
EC50 = 700 nM
|
|
|
CP0847322
|
2-{(2R,4aR,5R,6R,7aS)-6-hydroxy-5-[(1E)-5-phenoxy-1-penten-1-yl]octahydrocyclopenta[b]pyran-2-yl}-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C23H27NO5S
|
1
|
1 |
EC50 = 970 nM
|
|
|
CP0415586
|
2-[2-[(1R,2R)-2-[(E,4S)-5-cyclopentyl-4-hydroxy-4-methylpent-1-enyl]-5-oxocyclopentyl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C22H31NO4S2
|
1
|
1 |
EC50 = 2000 nM
|
|
|
CP0870958
|
2-[(2R,4aR,5R,6R,7aS)-6-hydroxy-5-(3-phenoxypropyl)octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C21H25NO5S
|
1
|
1 |
EC50 = 4200 nM
|
|
|
CP0391092
|
2-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-oxazole-4-carboxylic acid
Show/Hide
|
C20H22ClNO6
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0391098
|
4-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]thiophene-2-carboxylic acid
Show/Hide
|
C21H23ClO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0401698
|
2-[(2R,4aR,5S,6S,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-methoxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C21H24ClNO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0401699
|
2-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C20H22ClNO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0401700
|
2-[(2R,4aR,5S,6S,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C20H22ClNO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0401702
|
2-[(2R,4aR,5S,6S,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-fluoro-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C20H21ClFNO4S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0407410
|
4-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]furan-2-carboxylic acid
Show/Hide
|
C21H23ClO6
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0434444
|
5-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]furan-2-carboxylic acid
Show/Hide
|
C21H23ClO6
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0380278
|
2-[(2R,4aR,5S,6R,7aS)-6-hydroxy-5-(phenoxymethyl)-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C19H21NO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0928357
|
sodium 1-(5-bromo-2-(2,4-dichlorobenzyloxy)phenyl)-5-methyl-1H-pyrazole-3-carboxylate
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|
C19H14BrCl2N2NaO3
|
1
|
1 |
IC50 = 0.1288 nM
|
|
|
CP0209434
|
3-acetamido-5-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C27H21BrF2N2O4
|
2
|
1 |
IC50 = 0.3981 nM
|
|
|
2 |
Ki = 0.1 nM
|
|
|
CP0456738
|
3-amino-5-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C25H19BrF2N2O3
|
1
|
1 |
IC50 = 0.5012 nM
|
|
|
CP0541607
|
3-acetamido-5-[2-[5-bromo-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C27H22BrFN2O4
|
1
|
1 |
IC50 = 0.7943 nM
|
|
|
CP0920199
|
3-(2-(2-(2,6-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C25H18BrF2NO3
|
1
|
1 |
IC50 = 1 nM
|
|
|
CP0427628
|
3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-5-(2-oxopiperidin-1-yl)benzoic acid
Show/Hide
|
C30H25BrF2N2O4
|
1
|
1 |
IC50 = 1.259 nM
|
|
|
CP0427630
|
3-acetamido-5-[2-methyl-5-[2-phenylmethoxy-5-(trifluoromethyl)phenyl]pyrrol-1-yl]benzoic acid
Show/Hide
|
C28H23F3N2O4
|
1
|
1 |
IC50 = 1.259 nM
|
|
|
CP0434068
|
3-acetamido-5-[2-(5-bromo-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C27H23BrN2O4
|
1
|
1 |
IC50 = 1.259 nM
|
|
|
CP0456737
|
3-[acetyl(methyl)amino]-5-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C28H23BrF2N2O4
|
1
|
1 |
IC50 = 1.259 nM
|
|
|
CP0880014
|
3-(2-(2-(2,4,6-trifluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C25H17BrF3NO3
|
1
|
1 |
IC50 = 1.585 nM
|
|
|
CP0427632
|
3-acetamido-5-[2-[2-[(2,4-difluorophenyl)methoxy]-5-iodophenyl]-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C27H21F2IN2O4
|
1
|
1 |
IC50 = 1.585 nM
|
|
|
CP0434067
|
3-[2-[5-chloro-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-5-(methanesulfonamido)benzoic acid
Show/Hide
|
C26H22ClFN2O5S
|
1
|
1 |
IC50 = 1.585 nM
|
|
|
CP0462923
|
4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-[(1R)-1-phenylethyl]benzamide
Show/Hide
|
C33H29ClN2O2
|
1
|
1 |
IC50 = 1.585 nM
|
|
|
CP0427634
|
3-acetamido-5-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C27H23ClN2O4
|
1
|
1 |
IC50 = 1.995 nM
|
|
|
CP0456736
|
3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-5-(2-oxopyrrolidin-1-yl)benzoic acid
Show/Hide
|
C29H23BrF2N2O4
|
1
|
1 |
IC50 = 1.995 nM
|
|
|
CP0167117
|
6-(2-(2-(2,4-difluorobenzyloxy)-5-chlorophenyl)cyclopent-1-enyl)picolinic acid
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|
C24H18ClF2NO3
|
1
|
1 |
IC50 = 2.512 nM
|
|
|
CP0869607
|
3-{2-[5-Bromo-2-(4-methyl-benzyloxy)-phenyl]-5-methyl-pyrrol-1-yl}-benzoic acid
Show/Hide
|
C26H22BrNO3
|
1
|
1 |
IC50 = 2.512 nM
|
|
|
CP0522274
|
3-acetamido-5-[2-[5-chloro-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C27H22ClFN2O4
|
1
|
1 |
IC50 = 2.512 nM
|
|
|
CP0444761
|
N-(benzenesulfonyl)-3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzamide
Show/Hide
|
C31H25ClN2O4S
|
1
|
1 |
IC50 = 2.512 nM
|
|
|
CP0497527
|
4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-(pyridin-2-ylmethyl)benzamide
Show/Hide
|
C31H26ClN3O2
|
1
|
1 |
IC50 = 2.512 nM
|
|
|
CP0538704
|
N-(benzenesulfonyl)-3-[2-methyl-5-(2-phenylmethoxyphenyl)pyrrol-1-yl]benzamide
Show/Hide
|
C31H26N2O4S
|
1
|
1 |
IC50 = 2.512 nM
|
|
|
CP0876752
|
N-((5-(4-ethoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(2,3-dichlorophenyl)-4-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C25H20Cl2F3N3O4S
|
2
|
1 |
IC50 = 2.512 nM
|
|
|
2 |
Ki = 6.31 nM
|
|
|
CP0910939
|
3-(2-(2-(2-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C25H19BrFNO3
|
1
|
1 |
IC50 = 3.162 nM
|
|
|
CP0439617
|
3-amino-5-[2-(5-bromo-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C25H21BrN2O3
|
1
|
1 |
IC50 = 3.162 nM
|
|
|
CP0862538
|
3-(2-(2-(2,4-difluorobenzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C25H18ClF2NO3
|
1
|
1 |
IC50 = 3.981 nM
|
|
|
CP0456739
|
3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-5-chlorobenzoic acid
Show/Hide
|
C25H17BrClF2NO3
|
1
|
1 |
IC50 = 3.981 nM
|
|
|
CP0485040
|
3-acetamido-5-[2-[5-fluoro-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C27H22F2N2O4
|
1
|
1 |
IC50 = 3.981 nM
|
|
|
CP0524522
|
3-chloro-5-[2-[5-chloro-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C25H17Cl2F2NO3
|
1
|
1 |
IC50 = 3.981 nM
|
|
|
CP0562586
|
3-amino-5-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C25H21ClN2O3
|
1
|
1 |
IC50 = 3.981 nM
|
|
|
CP0485321
|
4-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-N-methylbenzamide
Show/Hide
|
C26H21BrF2N2O2
|
1
|
1 |
IC50 = 3.981 nM
|
|
|
CP0538705
|
3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-N-methylsulfonylbenzamide
Show/Hide
|
C26H21BrF2N2O4S
|
1
|
1 |
IC50 = 3.981 nM
|
|
|
CP0942622
|
N-((5-(4-ethoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
Show/Hide
|
C26H26ClN3O4S
|
2
|
1 |
IC50 = 3.981 nM
|
|
|
2 |
Ki = 50.12 nM
|
|
|
CP0192211
|
3-[2-[5-chloro-2-(2-methylpropoxy)phenyl]-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C22H22ClNO3
|
1
|
1 |
IC50 = 5.012 nM
|
|
|
CP0851033
|
3-(2-(5-bromo-2-isobutoxyphenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C22H22BrNO3
|
1
|
1 |
IC50 = 5.012 nM
|
|
|
CP0862528
|
3-(2-(2-(2,4-dichlorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C25H18BrCl2NO3
|
1
|
1 |
IC50 = 5.012 nM
|
|
|
CP0916321
|
3-(2-(2-(3,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C25H18BrF2NO3
|
1
|
1 |
IC50 = 5.012 nM
|
|
|
CP0941236
|
3-(2-(2-(benzyloxy)-5-(trifluoromethyl)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C26H20F3NO3
|
1
|
1 |
IC50 = 5.012 nM
|
|
|
CP0464233
|
3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-5-(methoxycarbonylamino)benzoic acid
Show/Hide
|
C27H23ClN2O5
|
1
|
1 |
IC50 = 5.012 nM
|
|
|
CP0464235
|
3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-5-(1,1-dioxo-1,2-thiazolidin-2-yl)benzoic acid
Show/Hide
|
C28H25ClN2O5S
|
1
|
1 |
IC50 = 5.012 nM
|
|
|
CP0493623
|
3-bromo-5-[2-[5-chloro-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C25H17BrClF2NO3
|
1
|
1 |
IC50 = 5.012 nM
|
|
|
CP0562587
|
3-bromo-5-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C25H19BrClNO3
|
1
|
1 |
IC50 = 5.012 nM
|
|
|
CP0462931
|
N-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-[2-methyl-5-(2-phenylmethoxyphenyl)pyrrol-1-yl]benzamide
Show/Hide
|
C30H27N3O5S
|
1
|
1 |
IC50 = 5.012 nM
|
|
|
CP0497525
|
4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-[(1S)-1-phenylethyl]benzamide
Show/Hide
|
C33H29ClN2O2
|
1
|
1 |
IC50 = 5.012 nM
|
|
|
CP0082063
|
3-(2-(2-(4-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C25H19BrFNO3
|
1
|
1 |
IC50 = 6.31 nM
|
|
|
CP0942294
|
3-(2-(2-(4-fluorobenzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C25H19ClFNO3
|
1
|
1 |
IC50 = 6.31 nM
|
|
|
CP0942298
|
3-(2-(2-(2,3-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C25H18BrF2NO3
|
1
|
1 |
IC50 = 6.31 nM
|
|
|
CP0439618
|
3-[2-[5-bromo-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-4-fluorobenzoic acid
Show/Hide
|
C25H18BrF2NO3
|
1
|
1 |
IC50 = 6.31 nM
|
|
|
CP0485043
|
3-[2-[5-chloro-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-4-fluorobenzoic acid
Show/Hide
|
C25H17ClF3NO3
|
1
|
1 |
IC50 = 6.31 nM
|
|
|
CP0554333
|
4-fluoro-3-[2-methyl-5-[2-phenylmethoxy-5-(trifluoromethyl)phenyl]pyrrol-1-yl]benzoic acid
Show/Hide
|
C26H19F4NO3
|
1
|
1 |
IC50 = 6.31 nM
|
|
|
CP0876749
|
N-((5-(4-ethoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(2,3-dichlorophenyl)-4-methylbenzenesulfonamide
Show/Hide
|
C25H23Cl2N3O4S
|
2
|
1 |
IC50 = 6.31 nM
|
|
|
2 |
Ki = 31.62 nM
|
|
|
CP0945566
|
N-((5-(4-methoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
Show/Hide
|
C25H24ClN3O4S
|
2
|
1 |
IC50 = 6.31 nM
|
|
|
2 |
Ki = 39.81 nM
|
|
|
CP0109778
|
3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C25H20ClNO3
|
2
|
1 |
IC50 = 7.943 nM
|
|
|
2 |
Ki = 0.7079 nM
|
|
|
CP0110250
|
3-(2-(2-(benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C25H20BrNO3
|
1
|
1 |
IC50 = 7.943 nM
|
|
|
CP0893530
|
3-(2-(2-(2,5-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C25H18BrF2NO3
|
1
|
1 |
IC50 = 7.943 nM
|
|
|
CP0485039
|
3-(1,1-dioxo-1,2-thiazolidin-2-yl)-5-[2-[2-[(4-fluorophenyl)methoxy]-5-(trifluoromethyl)phenyl]-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C29H24F4N2O5S
|
1
|
1 |
IC50 = 7.943 nM
|
|
|
CP0540242
|
N-[4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]phenyl]sulfonylbenzamide
Show/Hide
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C31H25ClN2O4S
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1
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1 |
IC50 = 7.943 nM
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CP0551265
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4-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzamide
Show/Hide
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C25H19BrF2N2O2
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1
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1 |
IC50 = 7.943 nM
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CP0897850
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N-(3,4-dimethoxyphenethyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
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C27H32N2O5S
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2
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1 |
IC50 = 7.943 nM
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2 |
Kd = 5.012 nM
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CP0920137
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N-((5-(4-methoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(2,3-dichlorophenyl)-4-methylbenzenesulfonamide
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C24H21Cl2N3O4S
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2
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1 |
IC50 = 7.943 nM
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2 |
Ki = 39.81 nM
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CP0922170
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N-(2,3-dichlorophenyl)-N-((5-(4-methoxyphenylamino)-1,3,4-oxadiazol-2-yl)methyl)-4-(trifluoromethyl)benzenesulfonamide
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C23H17Cl2F3N4O4S
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2
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1 |
IC50 = 7.943 nM
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2 |
Ki = 63.1 nM
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CP0370068
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5-(2-(2-(benzyloxy)-5-(trifluoromethyl)phenyl)cyclopent-1-enyl)nicotinic acid
Show/Hide
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C25H20F3NO3
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1
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1 |
IC50 = 10 nM
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CP0645644
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sodium 6-(5-chloro-2-(2,4-dichlorobenzyloxy)benzyl)picolinate
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C20H13Cl3NNaO3
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2
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1 |
IC50 = 10 nM
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2 |
Ki = 25.12 nM
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CP0192990
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3-(2-(2-(benzyloxy)-5-chlorophenyl)-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C24H18ClNO3
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1
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1 |
IC50 = 10 nM
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CP0932566
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3-(2-(2-(4-chlorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C25H19BrClNO3
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1
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1 |
IC50 = 10 nM
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CP0941231
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3-(2-(2-(3-chlorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C25H19BrClNO3
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1
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1 |
IC50 = 10 nM
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CP0434069
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3-[2-[5-chloro-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-5-(trifluoromethyl)benzoic acid
Show/Hide
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C26H17ClF5NO3
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1
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1 |
IC50 = 10 nM
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CP0439448
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3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-N,N-dimethylbenzamide
Show/Hide
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C27H23BrF2N2O2
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1
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1 |
IC50 = 10 nM
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CP0675883
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sodium 6-(5-chloro-2-(2-chloro-4-fluorobenzyloxy)benzyl)picolinate
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C20H13Cl2FNNaO3
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2
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1 |
IC50 = 12.59 nM
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2 |
Ki = 100 nM
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CP0709887
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sodium 6-(5-chloro-2-(4-chloro-2-fluorobenzyloxy)benzyl)picolinate
Show/Hide
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C20H13Cl2FNNaO3
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3
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1 |
IC50 = 12.59 nM
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2 |
Kd = 7.943 nM
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3 |
Ki = 7.943 nM
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CP0897821
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3-(2-(2-(2-chlorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C25H19BrClNO3
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1
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1 |
IC50 = 12.59 nM
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CP0899685
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3-(2-(2-(2-fluoro-4-(trifluoromethyl)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C26H18BrF4NO3
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1
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1 |
IC50 = 12.59 nM
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CP0920198
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3-(2-(2-(2-chloro-6-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C25H18BrClFNO3
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1
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1 |
IC50 = 12.59 nM
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CP0466792
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3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-5-(trifluoromethyl)benzoic acid
Show/Hide
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C26H17BrF5NO3
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1
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1 |
IC50 = 12.59 nM
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CP0462924
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4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-(pyridin-3-ylmethyl)benzamide
Show/Hide
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C31H26ClN3O2
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1
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1 |
IC50 = 12.59 nM
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CP0876737
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N-((5-(4-(dimethylamino)benzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
Show/Hide
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C26H27ClN4O3S
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2
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1 |
IC50 = 12.59 nM
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2 |
Ki = 19.95 nM
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CP0648581
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sodium 6-(5'-chloro-2'-isobutoxybiphenyl-2-yl)picolinate
Show/Hide
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C22H19ClNNaO3
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1
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1 |
IC50 = 15.85 nM
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CP0875503
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3-(2-(2-(2-chloro-4-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C25H18BrClFNO3
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1
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1 |
IC50 = 15.85 nM
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CP0897819
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3-(2-(5-bromo-2-(cyclopentylmethoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C24H24BrNO3
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1
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1 |
IC50 = 15.85 nM
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CP0899684
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3-(2-(2-(4-(trifluoromethoxy)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C26H19BrF3NO4
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1
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1 |
IC50 = 15.85 nM
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CP0462925
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4-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-N-tert-butylbenzamide
Show/Hide
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C29H27BrF2N2O2
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1
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1 |
IC50 = 15.85 nM
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CP0540240
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4-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-N,N-dimethylbenzamide
Show/Hide
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C27H23BrF2N2O2
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1
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1 |
IC50 = 15.85 nM
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CP0862530
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3-{2-[5-Bromo-2-(2-methyl-benzyloxy)-phenyl]-5-methyl-pyrrol-1-yl}-benzoic acid
Show/Hide
|
C26H22BrNO3
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1
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1 |
IC50 = 19.95 nM
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CP0862539
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3-(2-(2-(benzyloxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C25H21NO3
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1
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1 |
IC50 = 19.95 nM
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CP0444760
|
2-(5-chloro-2-phenylmethoxyphenyl)-5-methyl-1-(4-methylsulfonylphenyl)pyrrole
Show/Hide
|
C25H22ClNO3S
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1
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1 |
IC50 = 19.95 nM
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CP0462927
|
4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzenesulfonamide
Show/Hide
|
C24H21ClN2O3S
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1
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1 |
IC50 = 19.95 nM
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CP0538700
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3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-N-methylbenzamide
Show/Hide
|
C26H21BrF2N2O2
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1
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1 |
IC50 = 19.95 nM
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CP0920132
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N-((5-(4-methoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-4-chloro-N-(2,3-dichlorophenyl)benzenesulfonamide
Show/Hide
|
C23H18Cl3N3O4S
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2
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1 |
IC50 = 19.95 nM
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2 |
Ki = 63.1 nM
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CP0932499
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N-(3-chloro-2-methylphenyl)-N-((5-((4-methoxyphenylamino)methyl)-1,3,4-oxadiazol-2-yl)methyl)-4-methylbenzenesulfonamide
Show/Hide
|
C25H25ClN4O4S
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2
|
1 |
IC50 = 19.95 nM
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2 |
Ki = 79.43 nM
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CP0867891
|
sodium 6-(5-chloro-2-(2,4-difluorobenzyloxy)benzyl)picolinate
Show/Hide
|
C20H13ClF2NNaO3
|
1
|
1 |
IC50 = 25.12 nM
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CP0851030
|
3-(2-(5-bromo-2-((5-methylisoxazol-3-yl)methoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C23H19BrN2O4
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1
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1 |
IC50 = 25.12 nM
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CP0869609
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3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-chloro-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C24H17Cl2NO3
|
1
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1 |
IC50 = 25.12 nM
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CP0918358
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3-(2-(5-chloro-2-(cyclopentylmethoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C24H24ClNO3
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1
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1 |
IC50 = 25.12 nM
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CP0920194
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3-(2-(2-(benzyloxy)-5-(methylsulfonyl)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C26H23NO5S
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1
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1 |
IC50 = 25.12 nM
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CP0444759
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N-benzyl-4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzamide
Show/Hide
|
C32H27ClN2O2
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1
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1 |
IC50 = 25.12 nM
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CP0524536
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N-benzyl-3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzamide
Show/Hide
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C32H27ClN2O2
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1
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1 |
IC50 = 25.12 nM
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CP0540241
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2-[3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]phenyl]-1,1,1,3,3,3-hexafluoropropan-2-ol
Show/Hide
|
C27H18BrF8NO2
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1
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1 |
IC50 = 25.12 nM
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CP0551264
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5-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-2H-benzotriazole
Show/Hide
|
C24H19ClN4O
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1
|
1 |
IC50 = 25.12 nM
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CP0876729
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N-(2-ethylphenyl)-N-((5-((4-methoxyphenoxy)methyl)-1,3,4-oxadiazol-2-yl)methyl)-4-methylbenzenesulfonamide
Show/Hide
|
C26H27N3O5S
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2
|
1 |
IC50 = 25.12 nM
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2 |
Ki = 125.89 nM
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CP0867850
|
sodium 6-(5-chloro-2-(cyclopentylmethoxy)benzyl)picolinate
Show/Hide
|
C19H19ClNNaO3
|
1
|
1 |
IC50 = 31.62 nM
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CP0942293
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3-(2-(2-(cyclohexylmethoxy)-5-(trifluoromethyl)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C26H26F3NO3
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1
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1 |
IC50 = 31.62 nM
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CP0462929
|
2-(5-bromo-2-phenylmethoxyphenyl)-5-methyl-1-(4-methylsulfonylphenyl)pyrrole
Show/Hide
|
C25H22BrNO3S
|
1
|
1 |
IC50 = 31.62 nM
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CP0876751
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N-(3-chloro-2-methylphenyl)-N-((5-(4-methoxyphenylamino)-1,3,4-oxadiazol-2-yl)methyl)-4-methylbenzenesulfonamide
Show/Hide
|
C24H23ClN4O4S
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2
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1 |
IC50 = 31.62 nM
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2 |
Ki = 79.43 nM
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CP0867849
|
sodium 6-(5-chloro-2-(2-chlorobenzyloxy)benzyl)picolinate
Show/Hide
|
C20H14Cl2NNaO3
|
1
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1 |
IC50 = 39.81 nM
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CP0890928
|
sodium 6-(5-chloro-2-isobutoxybenzyl)picolinate
Show/Hide
|
C17H17ClNNaO3
|
1
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1 |
IC50 = 39.81 nM
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CP0946776
|
sodium 6-(5-chloro-2-(4-chlorobenzyloxy)benzyl)picolinate
Show/Hide
|
C20H14Cl2NNaO3
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1
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1 |
IC50 = 39.81 nM
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CP0916323
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3-(2-(2-(4-(trifluoromethyl)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C26H19BrF3NO3
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1
|
1 |
IC50 = 39.81 nM
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CP0916448
|
3-(2-(5-bromo-2-(cyclohexylmethoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C25H26BrNO3
|
1
|
1 |
IC50 = 39.81 nM
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CP0941234
|
3-(2-(5-chloro-2-((tetrahydrofuran-2-yl)methoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C23H22ClNO4
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1
|
1 |
IC50 = 39.81 nM
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CP0942292
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3-(2-(5-chloro-2-((tetrahydro-2H-pyran-4-yl)methoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C24H24ClNO4
|
1
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1 |
IC50 = 39.81 nM
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CP0439539
|
6-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-1H-indazole
Show/Hide
|
C25H20ClN3O
|
1
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1 |
IC50 = 39.81 nM
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CP0484290
|
2-[3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]phenyl]-5-methyl-1,3,4-oxadiazole
Show/Hide
|
C27H20BrF2N3O2
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1
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1 |
IC50 = 39.81 nM
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CP0485320
|
5-[4-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]phenyl]-1H-imidazole
Show/Hide
|
C27H20BrF2N3O
|
1
|
1 |
IC50 = 39.81 nM
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CP0510800
|
3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-[(1R)-1-phenylethyl]benzamide
Show/Hide
|
C33H29ClN2O2
|
1
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1 |
IC50 = 39.81 nM
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CP0538699
|
5-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-1H-indazole
Show/Hide
|
C25H20ClN3O
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1
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1 |
IC50 = 39.81 nM
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CP0942621
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N-(2,3-dichlorophenyl)-N-((5-(4-methoxyphenylamino)-1,3,4-oxadiazol-2-yl)methyl)-4-methylbenzenesulfonamide
Show/Hide
|
C23H20Cl2N4O4S
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2
|
1 |
IC50 = 39.81 nM
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2 |
Ki = 50.12 nM
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CP0855112
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3-(2-(2-(4-methoxybenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C26H22BrNO4
|
1
|
1 |
IC50 = 50.12 nM
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CP0916322
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3-(2-(2-(3-methoxybenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C26H22BrNO4
|
1
|
1 |
IC50 = 50.12 nM
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CP0394640
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3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-(pyridin-2-ylmethyl)benzamide
Show/Hide
|
C31H26ClN3O2
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1
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1 |
IC50 = 50.12 nM
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CP0538701
|
4-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-N,N-diethylbenzamide
Show/Hide
|
C29H27BrF2N2O2
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1
|
1 |
IC50 = 50.12 nM
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CP0910970
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N-((5-(4-(trifluoromethyl)benzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
Show/Hide
|
C25H21ClF3N3O3S
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2
|
1 |
IC50 = 50.12 nM
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2 |
Ki = 158.49 nM
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CP0394728
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7-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-4-methyl-1H-quinolin-2-one
Show/Hide
|
C28H23ClN2O2
|
1
|
1 |
IC50 = 63.1 nM
|
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CP0439445
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2-[3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]phenyl]-1H-benzimidazole
Show/Hide
|
C31H22BrF2N3O
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1
|
1 |
IC50 = 63.1 nM
|
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CP0439447
|
3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-(pyridin-3-ylmethyl)benzamide
Show/Hide
|
C31H26ClN3O2
|
1
|
1 |
IC50 = 63.1 nM
|
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CP0439540
|
4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-(pyridin-4-ylmethyl)benzamide
Show/Hide
|
C31H26ClN3O2
|
1
|
1 |
IC50 = 63.1 nM
|
|
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CP0484293
|
3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-(pyridin-4-ylmethyl)benzamide
Show/Hide
|
C31H26ClN3O2
|
1
|
1 |
IC50 = 63.1 nM
|
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CP0505267
|
3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzamide
Show/Hide
|
C25H21ClN2O2
|
1
|
1 |
IC50 = 63.1 nM
|
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CP0540237
|
N-[3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]phenyl]acetamide
Show/Hide
|
C26H23ClN2O2
|
1
|
1 |
IC50 = 63.1 nM
|
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CP0879922
|
N-((5-(4-methoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-4-methyl-N-(2-methyl-3-(trifluoromethyl)phenyl)benzenesulfonamide
Show/Hide
|
C26H24F3N3O4S
|
2
|
1 |
IC50 = 63.1 nM
|
|
|
2 |
Ki = 398.11 nM
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CP0920139
|
N-((5-(2,6-dichlorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
Show/Hide
|
C24H20Cl3N3O3S
|
2
|
1 |
IC50 = 63.1 nM
|
|
|
2 |
Ki = 501.19 nM
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CP0947170
|
N-((5-(2,4-dichlorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
Show/Hide
|
C24H20Cl3N3O3S
|
2
|
1 |
IC50 = 63.1 nM
|
|
|
2 |
Ki = 1000 nM
|
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CP0867890
|
sodium 6-(5-chloro-2-(2-fluorobenzyloxy)benzyl)picolinate
Show/Hide
|
C20H14ClFNNaO3
|
1
|
1 |
IC50 = 79.43 nM
|
|
|
CP0928358
|
sodium 6-(5-chloro-2-(2,4,6-trifluorobenzyloxy)benzyl)picolinate
Show/Hide
|
C20H12ClF3NNaO3
|
1
|
1 |
IC50 = 79.43 nM
|
|
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CP0851021
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3-(2-(2-(benzyloxy)-5-bromophenyl)-5-ethyl-1H-pyrrol-1-yl)benzoic acid
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C26H22BrNO3
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1
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1 |
IC50 = 79.43 nM
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CP0853242
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3-(2-(2-(3-(difluoromethoxy)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
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C26H20BrF2NO4
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1
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1 |
IC50 = 79.43 nM
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CP0538703
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N-[3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]phenyl]sulfonylbenzamide
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C31H25ClN2O4S
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1
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1 |
IC50 = 79.43 nM
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CP0876754
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N-((5-(2-chlorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
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C24H21Cl2N3O3S
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2
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1 |
IC50 = 79.43 nM
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2 |
Ki = 398.11 nM
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CP0906801
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sodium 6-(5-chloro-2-(cyclohexylmethoxy)benzyl)picolinate
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C20H21ClNNaO3
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1
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1 |
IC50 = 100 nM
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CP0935423
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sodium 6-(5-chloro-2-(4-fluorobenzyloxy)benzyl)picolinate
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C20H14ClFNNaO3
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1
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1 |
IC50 = 100 nM
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CP0862527
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3-(2-(2-(3,4-dichlorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
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C25H18BrCl2NO3
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1
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1 |
IC50 = 100 nM
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CP0916446
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3-(2-(2-(2-fluoro-6-(trifluoromethyl)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C26H18BrF4NO3
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1
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1 |
IC50 = 100 nM
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CP0921558
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3-(2-(2-(2,4-difluorobenzyloxy)-5-chlorophenyl)-5-(trifluoromethyl)-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C25H15ClF5NO3
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1
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1 |
IC50 = 100 nM
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CP0922210
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3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-ethyl-1H-pyrrol-1-yl)benzoic acid
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C26H22ClNO3
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1
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1 |
IC50 = 100 nM
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CP0853249
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3-(2-(5-chloro-2-(cyclohexylmethoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
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C25H26ClNO3
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1
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1 |
IC50 = 125.89 nM
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CP0485041
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3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-4-ethoxybenzoic acid
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C27H24ClNO4
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1
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1 |
IC50 = 125.89 nM
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CP0400069
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2-(5-chloro-2-phenylmethoxyphenyl)-5-methyl-1-(3-methylsulfonylphenyl)pyrrole
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C25H22ClNO3S
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1
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1 |
IC50 = 125.89 nM
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CP0524535
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3-[3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]phenyl]pyridine
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C29H21BrF2N2O
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1
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1 |
IC50 = 125.89 nM
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CP0540238
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2-[3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]phenyl]pyrimidine
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C28H20BrF2N3O
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1
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1 |
IC50 = 125.89 nM
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CP0935660
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N-((5-(4-ethoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(2-ethylphenyl)-4-methylbenzenesulfonamide
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C27H29N3O4S
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2
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1 |
IC50 = 125.89 nM
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2 |
Ki = 39.81 nM
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CP0878525
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sodium 6-(2-(benzyloxy)-5-chlorobenzyl)picolinate
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C20H15ClNNaO3
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1
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1 |
IC50 = 158.49 nM
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CP0562588
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4-chloro-3-[2-[5-chloro-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
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C25H17Cl2F2NO3
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1
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1 |
IC50 = 158.49 nM
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CP0439444
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5-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]isoindole-1,3-dione
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C26H17BrF2N2O3
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1
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1 |
IC50 = 158.49 nM
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CP0918609
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N-((5-(3-chlorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
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C24H21Cl2N3O3S
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2
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1 |
IC50 = 158.49 nM
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2 |
Ki = 1995.26 nM
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CP0891913
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sodium 6-(5-chloro-2-(cyclopropylmethoxy)benzyl)picolinate
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C17H15ClNNaO3
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1
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1 |
IC50 = 199.53 nM
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CP0851031
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3-(2-(5-bromo-2-((3,5-dimethylisoxazol-4-yl)methoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C24H21BrN2O4
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1
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1 |
IC50 = 199.53 nM
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CP0918718
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3-(2-(2-(4-fluorobenzyloxy)-5-chlorophenyl)-5-(trifluoromethyl)-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C25H16ClF4NO3
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1
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1 |
IC50 = 199.53 nM
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CP0538698
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3-[3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]phenyl]-5-methyl-1,2,4-oxadiazole
Show/Hide
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C27H20BrF2N3O2
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1
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1 |
IC50 = 199.53 nM
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CP0538702
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2-(5-bromo-2-phenylmethoxyphenyl)-5-methyl-1-(3-methylsulfonylphenyl)pyrrole
Show/Hide
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C25H22BrNO3S
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1
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1 |
IC50 = 199.53 nM
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CP0858980
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N-((5-(4-fluorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
Show/Hide
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C24H21ClFN3O3S
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2
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1 |
IC50 = 199.53 nM
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2 |
Ki = 501.19 nM
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CP0851029
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3-(2-(2-(3-(trifluoromethyl)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C26H19BrF3NO3
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1
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1 |
IC50 = 251.19 nM
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CP0485412
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3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-4-methoxybenzoic acid
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C26H22ClNO4
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1
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1 |
IC50 = 251.19 nM
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CP0505265
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2-[3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]phenyl]pyridine
Show/Hide
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C29H21BrF2N2O
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1
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1 |
IC50 = 251.19 nM
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CP0652436
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N-(4-chlorophenethyl)-2-(4-methyl-N-o-tolylphenylsulfonamido)acetamide
Show/Hide
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C24H25ClN2O3S
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1
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1 |
IC50 = 251.19 nM
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CP0434071
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4-chloro-3-[2-[5-chloro-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
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C25H18Cl2FNO3
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1
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1 |
IC50 = 316.23 nM
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CP0505266
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3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-[(1S)-1-phenylethyl]benzamide
Show/Hide
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C33H29ClN2O2
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1
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1 |
IC50 = 316.23 nM
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CP0949627
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N-((5-(3-fluorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
Show/Hide
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C24H21ClFN3O3S
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2
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1 |
IC50 = 316.23 nM
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2 |
Ki = 501.19 nM
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CP0910942
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3-[2-(4-Benzyloxy-biphenyl-3-yl)-5-methyl-pyrrol-1-yl]-benzoic acid
Show/Hide
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C31H25NO3
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1
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1 |
IC50 = 398.11 nM
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CP0920138
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N-((5-(4-chlorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(2-ethylphenyl)-4-methylbenzenesulfonamide
Show/Hide
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C25H24ClN3O3S
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2
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1 |
IC50 = 398.11 nM
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2 |
Ki = 316.23 nM
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CP0485319
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1-[4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]phenyl]-1,2,4-triazole
Show/Hide
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C26H21ClN4O
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1
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1 |
IC50 = 501.19 nM
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CP0497528
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2-methyl-1-(4-methylsulfonylphenyl)-5-(2-phenylmethoxyphenyl)pyrrole
Show/Hide
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C25H23NO3S
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1
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1 |
IC50 = 501.19 nM
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CP0522232
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3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-N-phenylbenzamide
Show/Hide
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C31H23BrF2N2O2
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1
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1 |
IC50 = 501.19 nM
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CP0540239
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3-[2-[2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzamide
Show/Hide
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C25H20F2N2O2
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1
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1 |
IC50 = 501.19 nM
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CP0876731
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N-(2-ethylphenyl)-N-((5-((4-methoxyphenylamino)methyl)-1,3,4-oxadiazol-2-yl)methyl)-4-methylbenzenesulfonamide
Show/Hide
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C26H28N4O4S
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2
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1 |
IC50 = 501.19 nM
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2 |
Ki = 794.33 nM
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CP0945695
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N-((5-(2-fluorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
Show/Hide
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C24H21ClFN3O3S
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2
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1 |
IC50 = 501.19 nM
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2 |
Ki = 630.96 nM
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CP0875506
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3-(2-(2-(benzyloxy)-5-(thiophen-3-yl)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C29H23NO3S
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1
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1 |
IC50 = 630.96 nM
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CP0497524
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5-[2-[2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-2H-benzotriazole
Show/Hide
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C24H18F2N4O
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1
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1 |
IC50 = 630.96 nM
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CP0862536
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3-(5-(2-(benzyloxy)-5-chlorophenyl)-3-bromo-2-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C25H19BrClNO3
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1
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1 |
IC50 = 794.33 nM
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CP0916164
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N-((5-benzyl-1,3,4-oxadiazol-2-yl)methyl)-N-(2-ethylphenyl)-4-methylbenzenesulfonamide
Show/Hide
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C25H25N3O3S
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2
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1 |
IC50 = 1000 nM
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2 |
Ki = 398.11 nM
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CP0427396
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4-[(1S)-1-[[5-phenyl-3-[[4-(trifluoromethyl)phenyl]methyl]triazole-4-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C26H21F3N4O3
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1
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1 |
IC50 > 10000 nM
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CP0427397
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4-[(1S)-1-[[5-(cyclopenten-1-yl)-3-[[4-(trifluoromethyl)phenyl]methyl]triazole-4-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C25H23F3N4O3
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1
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1 |
IC50 > 10000 nM
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CP0435681
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US8686018, 107
Show/Hide
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C22H18F5N3O4
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1
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1 |
IC50 > 10000 nM
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CP0438577
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4-[(1S)-1-[[5-phenyl-3-[2-[3-(trifluoromethyl)phenoxy]ethyl]triazole-4-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C27H23F3N4O4
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1
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1 |
IC50 > 10000 nM
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CP0438580
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4-[(1S)-1-[[5-(furan-3-yl)-3-[[4-(trifluoromethyl)phenyl]methyl]triazole-4-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C24H19F3N4O4
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1
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1 |
IC50 > 10000 nM
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CP0473341
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4-[(1S)-1-[[5-(5-methylthiophen-2-yl)-3-[[4-(trifluoromethyl)phenyl]methyl]triazole-4-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C25H21F3N4O3S
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1
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1 |
IC50 > 10000 nM
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CP0473342
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4-[(1S)-1-[[5-thiophen-3-yl-3-[[4-(trifluoromethyl)phenyl]methyl]triazole-4-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C24H19F3N4O3S
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1
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1 |
IC50 > 10000 nM
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CP0473344
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4-[(1S)-1-[[5-[(E)-prop-1-enyl]-3-[[4-(trifluoromethyl)phenyl]methyl]triazole-4-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C23H21F3N4O3
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1
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1 |
IC50 > 10000 nM
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CP0477510
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4-[(1S)-1-[[5-prop-1-ynyl-3-[[4-(trifluoromethyl)phenyl]methyl]triazole-4-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C23H19F3N4O3
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1
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1 |
IC50 > 10000 nM
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CP0477511
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4-[(1S)-1-[[3-[2-(4-fluorophenoxy)ethyl]-5-phenyltriazole-4-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C26H23FN4O4
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1
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1 |
IC50 > 10000 nM
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CP0853250
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3-(5-(2-(benzyloxy)-5-chlorophenyl)-2-methyl-3-phenyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C31H24ClNO3
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1
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1 |
IC50 < 1000 nM
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CP0875505
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3-(5-(2-(benzyloxy)-5-chlorophenyl)-3-chloro-2-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
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C25H19Cl2NO3
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1
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1 |
IC50 < 1000 nM
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CP0910605
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2-(2-(benzyloxy)phenyl)-5-methyl-1-(3-(methylsulfonyl)phenyl)-1H-pyrrole
Show/Hide
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C25H23NO3S
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1
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1 |
IC50 < 1000 nM
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CP0882825
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N-((5-(4-methoxyphenoxy)-1,3,4-oxadiazol-2-yl)methyl)-N-(2-ethylphenyl)-4-methylbenzenesulfonamide
Show/Hide
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C25H25N3O5S
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2
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1 |
IC50 < 1000 nM
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2 |
Ki = 100 nM
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CP0383448
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5-[2-[5-chloro-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-2-methylbenzoic acid
Show/Hide
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C26H21ClFNO3
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1
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1 |
Ki = 1 nM
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CP0035659
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N-[(4-chlorophenyl)methyl]-2-(2-ethyl-N-(4-methylphenyl)sulfonylanilino)acetamide
Show/Hide
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C24H25ClN2O3S
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1
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1 |
Ki = 10 nM
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CP0484317
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2-(2-ethyl-N-(4-methylphenyl)sulfonylanilino)-N-[(4-methoxyphenyl)methyl]acetamide
Show/Hide
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C25H28N2O4S
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1
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1 |
Ki = 25.12 nM
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CP0915923
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N-(3,4-dimethoxybenzyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
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C26H30N2O5S
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1
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1 |
Ki = 25.12 nM
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CP0897849
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N-benzyl-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
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C24H26N2O3S
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1
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1 |
Ki = 63.1 nM
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CP0882726
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N-(3-methoxybenzyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
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C25H28N2O4S
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1
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1 |
Ki = 79.43 nM
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CP0915906
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N-(4-chlorobenzyl)-2-(N-(1-ethyl-1H-pyrazol-5-yl)-4-methylphenylsulfonamido)acetamide
Show/Hide
|
C21H23ClN4O3S
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1
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1 |
Ki = 158.49 nM
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CP0844852
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N-(4-chlorobenzyl)-2-(4-methyl-N-(2-methylpyridin-3-yl)phenylsulfonamido)acetamide
Show/Hide
|
C22H22ClN3O3S
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1
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1 |
Ki = 199.53 nM
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CP0939750
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N-(3-chlorobenzyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
|
C24H25ClN2O3S
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1
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1 |
Ki = 251.19 nM
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CP0844860
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N-(4-chlorobenzyl)-2-(4-methyl-N-(1-methyl-1H-pyrazol-5-yl)phenylsulfonamido)acetamide
Show/Hide
|
C20H21ClN4O3S
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1
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1 |
Ki = 398.11 nM
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CP0427199
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N-(2-ethylphenyl)-N-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]methyl]-4-methylbenzenesulfonamide
Show/Hide
|
C26H27N3O4S
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1
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1 |
Ki = 630.96 nM
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CP0942223
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N-(4-chlorobenzyl)-2-(4-methyl-N-(3-methylpyridin-2-yl)phenylsulfonamido)acetamide
Show/Hide
|
C22H22ClN3O3S
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1
|
1 |
Ki = 794.33 nM
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CP0895712
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N-(4-chlorobenzyl)-2-(4-methyl-N-(6-methylpyridin-3-yl)phenylsulfonamido)acetamide
Show/Hide
|
C22H22ClN3O3S
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1
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1 |
Ki < 1000 nM
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CP0902805
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N-(4-chlorobenzyl)-2-(4-methyl-N-(6-methylpyridin-2-yl)phenylsulfonamido)acetamide
Show/Hide
|
C22H22ClN3O3S
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1
|
1 |
Ki < 1000 nM
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CP0915907
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N-(4-chlorobenzyl)-2-(4-methyl-N-(pyridin-2-yl)phenylsulfonamido)acetamide
Show/Hide
|
C21H20ClN3O3S
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1
|
1 |
Ki < 1000 nM
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CP0918668
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N-(4-chlorobenzyl)-2-(4-methyl-N-(pyridin-3-yl)phenylsulfonamido)acetamide
Show/Hide
|
C21H20ClN3O3S
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1
|
1 |
Ki < 1000 nM
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CP0918673
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N-(4-chlorobenzyl)-2-(4-methyl-N-(5-methylpyridin-2-yl)phenylsulfonamido)acetamide
Show/Hide
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C22H22ClN3O3S
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1
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1 |
Ki < 1000 nM
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