Brief Information of the Cell Line and Protein
Cell Line ID: CL000011 , CHO
Synonyms
Chinese Hamster Ovary
CHO-ori
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_0213
Protein ID: PT01205 , Prostaglandin E2 receptor EP1 subtype
Gene Name PTGER1
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P34995
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000011  Protein ID: PT01205
 
Compound ID Compound Name Compound Formula
CP0847317
2-{(2R,4aR,5R,6R,7aS)-6-hydroxy-5-[(1E,3R)-3-hydroxy-4-phenoxy-1-buten-1-yl]octahydrocyclopenta[b]pyran-2-yl}-1,3-thiazole-4-carboxylic acid
   Show/Hide
C22H25NO6S
 1
1
EC50 = 1.4 nM
   TI
   LI
   LO
   TS
CP0055947
(15S)-prostaglandin E2
   Show/Hide
C20H32O5
 1
1
EC50 = 3.7 nM
   TI
   LI
   LO
   TS
CP0847320
2-[(2R,4aR,5R,6R,7aS)-6-hydroxy-5-(2-phenoxyethyl)octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
   Show/Hide
C20H23NO5S
 1
1
EC50 = 97 nM
   TI
   LI
   LO
   TS
CP0862926
2-{(2R,4aR,5R,6R,7aS)-6-hydroxy-5-[(1E)-4-phenoxy-1-buten-1-yl]octahydrocyclopenta[b]pyran-2-yl}-1,3-thiazole-4-carboxylic acid
   Show/Hide
C22H25NO5S
 1
1
EC50 = 160 nM
   TI
   LI
   LO
   TS
CP0847318
2-{(2R,4aR,5R,6R,7aS)-6-hydroxy-5-[(1E)-3-phenoxy-1-propen-1-yl]octahydrocyclopenta[b]pyran-2-yl}-1,3-thiazole-4-carboxylic acid
   Show/Hide
C21H23NO5S
 1
1
EC50 = 700 nM
   TI
   LI
   LO
   TS
CP0847322
2-{(2R,4aR,5R,6R,7aS)-6-hydroxy-5-[(1E)-5-phenoxy-1-penten-1-yl]octahydrocyclopenta[b]pyran-2-yl}-1,3-thiazole-4-carboxylic acid
   Show/Hide
C23H27NO5S
 1
1
EC50 = 970 nM
   TI
   LI
   LO
   TS
CP0415586
2-[2-[(1R,2R)-2-[(E,4S)-5-cyclopentyl-4-hydroxy-4-methylpent-1-enyl]-5-oxocyclopentyl]ethylsulfanyl]-1,3-thiazole-4-carboxylic acid
   Show/Hide
C22H31NO4S2
 1
1
EC50 = 2000 nM
   TI
   LI
   LO
   TS
CP0870958
2-[(2R,4aR,5R,6R,7aS)-6-hydroxy-5-(3-phenoxypropyl)octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
   Show/Hide
C21H25NO5S
 1
1
EC50 = 4200 nM
   TI
   LI
   LO
   TS
CP0391092
2-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-oxazole-4-carboxylic acid
   Show/Hide
C20H22ClNO6
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0391098
4-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]thiophene-2-carboxylic acid
   Show/Hide
C21H23ClO5S
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0401698
2-[(2R,4aR,5S,6S,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-methoxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
   Show/Hide
C21H24ClNO5S
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0401699
2-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
   Show/Hide
C20H22ClNO5S
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0401700
2-[(2R,4aR,5S,6S,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
   Show/Hide
C20H22ClNO5S
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0401702
2-[(2R,4aR,5S,6S,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-fluoro-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
   Show/Hide
C20H21ClFNO4S
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0407410
4-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]furan-2-carboxylic acid
   Show/Hide
C21H23ClO6
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0434444
5-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]furan-2-carboxylic acid
   Show/Hide
C21H23ClO6
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0380278
2-[(2R,4aR,5S,6R,7aS)-6-hydroxy-5-(phenoxymethyl)-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
   Show/Hide
C19H21NO5S
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0928357
sodium 1-(5-bromo-2-(2,4-dichlorobenzyloxy)phenyl)-5-methyl-1H-pyrazole-3-carboxylate
   Show/Hide
C19H14BrCl2N2NaO3
 1
1
IC50 = 0.1288 nM
   TI
   LI
   LO
   TS
CP0209434
3-acetamido-5-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C27H21BrF2N2O4
 2
1
IC50 = 0.3981 nM
   TI
   LI
   LO
   TS
2
Ki = 0.1 nM
   TI
   LI
   LO
   TS
CP0456738
3-amino-5-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C25H19BrF2N2O3
 1
1
IC50 = 0.5012 nM
   TI
   LI
   LO
   TS
CP0541607
3-acetamido-5-[2-[5-bromo-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C27H22BrFN2O4
 1
1
IC50 = 0.7943 nM
   TI
   LI
   LO
   TS
CP0920199
3-(2-(2-(2,6-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H18BrF2NO3
 1
1
IC50 = 1 nM
   TI
   LI
   LO
   TS
CP0427628
3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-5-(2-oxopiperidin-1-yl)benzoic acid
   Show/Hide
C30H25BrF2N2O4
 1
1
IC50 = 1.259 nM
   TI
   LI
   LO
   TS
CP0427630
3-acetamido-5-[2-methyl-5-[2-phenylmethoxy-5-(trifluoromethyl)phenyl]pyrrol-1-yl]benzoic acid
   Show/Hide
C28H23F3N2O4
 1
1
IC50 = 1.259 nM
   TI
   LI
   LO
   TS
CP0434068
3-acetamido-5-[2-(5-bromo-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C27H23BrN2O4
 1
1
IC50 = 1.259 nM
   TI
   LI
   LO
   TS
CP0456737
3-[acetyl(methyl)amino]-5-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C28H23BrF2N2O4
 1
1
IC50 = 1.259 nM
   TI
   LI
   LO
   TS
CP0880014
3-(2-(2-(2,4,6-trifluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H17BrF3NO3
 1
1
IC50 = 1.585 nM
   TI
   LI
   LO
   TS
CP0427632
3-acetamido-5-[2-[2-[(2,4-difluorophenyl)methoxy]-5-iodophenyl]-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C27H21F2IN2O4
 1
1
IC50 = 1.585 nM
   TI
   LI
   LO
   TS
CP0434067
3-[2-[5-chloro-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-5-(methanesulfonamido)benzoic acid
   Show/Hide
C26H22ClFN2O5S
 1
1
IC50 = 1.585 nM
   TI
   LI
   LO
   TS
CP0462923
4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-[(1R)-1-phenylethyl]benzamide
   Show/Hide
C33H29ClN2O2
 1
1
IC50 = 1.585 nM
   TI
   LI
   LO
   TS
CP0427634
3-acetamido-5-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C27H23ClN2O4
 1
1
IC50 = 1.995 nM
   TI
   LI
   LO
   TS
CP0456736
3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-5-(2-oxopyrrolidin-1-yl)benzoic acid
   Show/Hide
C29H23BrF2N2O4
 1
1
IC50 = 1.995 nM
   TI
   LI
   LO
   TS
CP0167117
6-(2-(2-(2,4-difluorobenzyloxy)-5-chlorophenyl)cyclopent-1-enyl)picolinic acid
   Show/Hide
C24H18ClF2NO3
 1
1
IC50 = 2.512 nM
   TI
   LI
   LO
   TS
CP0869607
3-{2-[5-Bromo-2-(4-methyl-benzyloxy)-phenyl]-5-methyl-pyrrol-1-yl}-benzoic acid
   Show/Hide
C26H22BrNO3
 1
1
IC50 = 2.512 nM
   TI
   LI
   LO
   TS
CP0522274
3-acetamido-5-[2-[5-chloro-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C27H22ClFN2O4
 1
1
IC50 = 2.512 nM
   TI
   LI
   LO
   TS
CP0444761
N-(benzenesulfonyl)-3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzamide
   Show/Hide
C31H25ClN2O4S
 1
1
IC50 = 2.512 nM
   TI
   LI
   LO
   TS
CP0497527
4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-(pyridin-2-ylmethyl)benzamide
   Show/Hide
C31H26ClN3O2
 1
1
IC50 = 2.512 nM
   TI
   LI
   LO
   TS
CP0538704
N-(benzenesulfonyl)-3-[2-methyl-5-(2-phenylmethoxyphenyl)pyrrol-1-yl]benzamide
   Show/Hide
C31H26N2O4S
 1
1
IC50 = 2.512 nM
   TI
   LI
   LO
   TS
CP0876752
N-((5-(4-ethoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(2,3-dichlorophenyl)-4-(trifluoromethyl)benzenesulfonamide
   Show/Hide
C25H20Cl2F3N3O4S
 2
1
IC50 = 2.512 nM
   TI
   LI
   LO
   TS
2
Ki = 6.31 nM
   TI
   LI
   LO
   TS
CP0910939
3-(2-(2-(2-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H19BrFNO3
 1
1
IC50 = 3.162 nM
   TI
   LI
   LO
   TS
CP0439617
3-amino-5-[2-(5-bromo-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C25H21BrN2O3
 1
1
IC50 = 3.162 nM
   TI
   LI
   LO
   TS
CP0862538
3-(2-(2-(2,4-difluorobenzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H18ClF2NO3
 1
1
IC50 = 3.981 nM
   TI
   LI
   LO
   TS
CP0456739
3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-5-chlorobenzoic acid
   Show/Hide
C25H17BrClF2NO3
 1
1
IC50 = 3.981 nM
   TI
   LI
   LO
   TS
CP0485040
3-acetamido-5-[2-[5-fluoro-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C27H22F2N2O4
 1
1
IC50 = 3.981 nM
   TI
   LI
   LO
   TS
CP0524522
3-chloro-5-[2-[5-chloro-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C25H17Cl2F2NO3
 1
1
IC50 = 3.981 nM
   TI
   LI
   LO
   TS
CP0562586
3-amino-5-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C25H21ClN2O3
 1
1
IC50 = 3.981 nM
   TI
   LI
   LO
   TS
CP0485321
4-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-N-methylbenzamide
   Show/Hide
C26H21BrF2N2O2
 1
1
IC50 = 3.981 nM
   TI
   LI
   LO
   TS
CP0538705
3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-N-methylsulfonylbenzamide
   Show/Hide
C26H21BrF2N2O4S
 1
1
IC50 = 3.981 nM
   TI
   LI
   LO
   TS
CP0942622
N-((5-(4-ethoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
   Show/Hide
C26H26ClN3O4S
 2
1
IC50 = 3.981 nM
   TI
   LI
   LO
   TS
2
Ki = 50.12 nM
   TI
   LI
   LO
   TS
CP0192211
3-[2-[5-chloro-2-(2-methylpropoxy)phenyl]-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C22H22ClNO3
 1
1
IC50 = 5.012 nM
   TI
   LI
   LO
   TS
CP0851033
3-(2-(5-bromo-2-isobutoxyphenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C22H22BrNO3
 1
1
IC50 = 5.012 nM
   TI
   LI
   LO
   TS
CP0862528
3-(2-(2-(2,4-dichlorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H18BrCl2NO3
 1
1
IC50 = 5.012 nM
   TI
   LI
   LO
   TS
CP0916321
3-(2-(2-(3,4-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H18BrF2NO3
 1
1
IC50 = 5.012 nM
   TI
   LI
   LO
   TS
CP0941236
3-(2-(2-(benzyloxy)-5-(trifluoromethyl)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C26H20F3NO3
 1
1
IC50 = 5.012 nM
   TI
   LI
   LO
   TS
CP0464233
3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-5-(methoxycarbonylamino)benzoic acid
   Show/Hide
C27H23ClN2O5
 1
1
IC50 = 5.012 nM
   TI
   LI
   LO
   TS
CP0464235
3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-5-(1,1-dioxo-1,2-thiazolidin-2-yl)benzoic acid
   Show/Hide
C28H25ClN2O5S
 1
1
IC50 = 5.012 nM
   TI
   LI
   LO
   TS
CP0493623
3-bromo-5-[2-[5-chloro-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C25H17BrClF2NO3
 1
1
IC50 = 5.012 nM
   TI
   LI
   LO
   TS
CP0562587
3-bromo-5-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C25H19BrClNO3
 1
1
IC50 = 5.012 nM
   TI
   LI
   LO
   TS
CP0462931
N-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-[2-methyl-5-(2-phenylmethoxyphenyl)pyrrol-1-yl]benzamide
   Show/Hide
C30H27N3O5S
 1
1
IC50 = 5.012 nM
   TI
   LI
   LO
   TS
CP0497525
4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-[(1S)-1-phenylethyl]benzamide
   Show/Hide
C33H29ClN2O2
 1
1
IC50 = 5.012 nM
   TI
   LI
   LO
   TS
CP0082063
3-(2-(2-(4-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H19BrFNO3
 1
1
IC50 = 6.31 nM
   TI
   LI
   LO
   TS
CP0942294
3-(2-(2-(4-fluorobenzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H19ClFNO3
 1
1
IC50 = 6.31 nM
   TI
   LI
   LO
   TS
CP0942298
3-(2-(2-(2,3-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H18BrF2NO3
 1
1
IC50 = 6.31 nM
   TI
   LI
   LO
   TS
CP0439618
3-[2-[5-bromo-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-4-fluorobenzoic acid
   Show/Hide
C25H18BrF2NO3
 1
1
IC50 = 6.31 nM
   TI
   LI
   LO
   TS
CP0485043
3-[2-[5-chloro-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-4-fluorobenzoic acid
   Show/Hide
C25H17ClF3NO3
 1
1
IC50 = 6.31 nM
   TI
   LI
   LO
   TS
CP0554333
4-fluoro-3-[2-methyl-5-[2-phenylmethoxy-5-(trifluoromethyl)phenyl]pyrrol-1-yl]benzoic acid
   Show/Hide
C26H19F4NO3
 1
1
IC50 = 6.31 nM
   TI
   LI
   LO
   TS
CP0876749
N-((5-(4-ethoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(2,3-dichlorophenyl)-4-methylbenzenesulfonamide
   Show/Hide
C25H23Cl2N3O4S
 2
1
IC50 = 6.31 nM
   TI
   LI
   LO
   TS
2
Ki = 31.62 nM
   TI
   LI
   LO
   TS
CP0945566
N-((5-(4-methoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
   Show/Hide
C25H24ClN3O4S
 2
1
IC50 = 6.31 nM
   TI
   LI
   LO
   TS
2
Ki = 39.81 nM
   TI
   LI
   LO
   TS
CP0109778
3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H20ClNO3
 2
1
IC50 = 7.943 nM
   TI
   LI
   LO
   TS
2
Ki = 0.7079 nM
   TI
   LI
   LO
   TS
CP0110250
3-(2-(2-(benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H20BrNO3
 1
1
IC50 = 7.943 nM
   TI
   LI
   LO
   TS
CP0893530
3-(2-(2-(2,5-difluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H18BrF2NO3
 1
1
IC50 = 7.943 nM
   TI
   LI
   LO
   TS
CP0485039
3-(1,1-dioxo-1,2-thiazolidin-2-yl)-5-[2-[2-[(4-fluorophenyl)methoxy]-5-(trifluoromethyl)phenyl]-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C29H24F4N2O5S
 1
1
IC50 = 7.943 nM
   TI
   LI
   LO
   TS
CP0540242
N-[4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]phenyl]sulfonylbenzamide
   Show/Hide
C31H25ClN2O4S
 1
1
IC50 = 7.943 nM
   TI
   LI
   LO
   TS
CP0551265
4-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzamide
   Show/Hide
C25H19BrF2N2O2
 1
1
IC50 = 7.943 nM
   TI
   LI
   LO
   TS
CP0897850
N-(3,4-dimethoxyphenethyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
   Show/Hide
C27H32N2O5S
 2
1
IC50 = 7.943 nM
   TI
   LI
   LO
   TS
2
Kd = 5.012 nM
   TI
   LI
   LO
   TS
CP0920137
N-((5-(4-methoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(2,3-dichlorophenyl)-4-methylbenzenesulfonamide
   Show/Hide
C24H21Cl2N3O4S
 2
1
IC50 = 7.943 nM
   TI
   LI
   LO
   TS
2
Ki = 39.81 nM
   TI
   LI
   LO
   TS
CP0922170
N-(2,3-dichlorophenyl)-N-((5-(4-methoxyphenylamino)-1,3,4-oxadiazol-2-yl)methyl)-4-(trifluoromethyl)benzenesulfonamide
   Show/Hide
C23H17Cl2F3N4O4S
 2
1
IC50 = 7.943 nM
   TI
   LI
   LO
   TS
2
Ki = 63.1 nM
   TI
   LI
   LO
   TS
CP0370068
5-(2-(2-(benzyloxy)-5-(trifluoromethyl)phenyl)cyclopent-1-enyl)nicotinic acid
   Show/Hide
C25H20F3NO3
 1
1
IC50 = 10 nM
   TI
   LI
   LO
   TS
CP0645644
sodium 6-(5-chloro-2-(2,4-dichlorobenzyloxy)benzyl)picolinate
   Show/Hide
C20H13Cl3NNaO3
 2
1
IC50 = 10 nM
   TI
   LI
   LO
   TS
2
Ki = 25.12 nM
   TI
   LI
   LO
   TS
CP0192990
3-(2-(2-(benzyloxy)-5-chlorophenyl)-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C24H18ClNO3
 1
1
IC50 = 10 nM
   TI
   LI
   LO
   TS
CP0932566
3-(2-(2-(4-chlorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H19BrClNO3
 1
1
IC50 = 10 nM
   TI
   LI
   LO
   TS
CP0941231
3-(2-(2-(3-chlorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H19BrClNO3
 1
1
IC50 = 10 nM
   TI
   LI
   LO
   TS
CP0434069
3-[2-[5-chloro-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-5-(trifluoromethyl)benzoic acid
   Show/Hide
C26H17ClF5NO3
 1
1
IC50 = 10 nM
   TI
   LI
   LO
   TS
CP0439448
3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-N,N-dimethylbenzamide
   Show/Hide
C27H23BrF2N2O2
 1
1
IC50 = 10 nM
   TI
   LI
   LO
   TS
CP0675883
sodium 6-(5-chloro-2-(2-chloro-4-fluorobenzyloxy)benzyl)picolinate
   Show/Hide
C20H13Cl2FNNaO3
 2
1
IC50 = 12.59 nM
   TI
   LI
   LO
   TS
2
Ki = 100 nM
   TI
   LI
   LO
   TS
CP0709887
sodium 6-(5-chloro-2-(4-chloro-2-fluorobenzyloxy)benzyl)picolinate
   Show/Hide
C20H13Cl2FNNaO3
 3
1
IC50 = 12.59 nM
   TI
   LI
   LO
   TS
2
Kd = 7.943 nM
   TI
   LI
   LO
   TS
3
Ki = 7.943 nM
   TI
   LI
   LO
   TS
CP0897821
3-(2-(2-(2-chlorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H19BrClNO3
 1
1
IC50 = 12.59 nM
   TI
   LI
   LO
   TS
CP0899685
3-(2-(2-(2-fluoro-4-(trifluoromethyl)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C26H18BrF4NO3
 1
1
IC50 = 12.59 nM
   TI
   LI
   LO
   TS
CP0920198
3-(2-(2-(2-chloro-6-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H18BrClFNO3
 1
1
IC50 = 12.59 nM
   TI
   LI
   LO
   TS
CP0466792
3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-5-(trifluoromethyl)benzoic acid
   Show/Hide
C26H17BrF5NO3
 1
1
IC50 = 12.59 nM
   TI
   LI
   LO
   TS
CP0462924
4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-(pyridin-3-ylmethyl)benzamide
   Show/Hide
C31H26ClN3O2
 1
1
IC50 = 12.59 nM
   TI
   LI
   LO
   TS
CP0876737
N-((5-(4-(dimethylamino)benzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
   Show/Hide
C26H27ClN4O3S
 2
1
IC50 = 12.59 nM
   TI
   LI
   LO
   TS
2
Ki = 19.95 nM
   TI
   LI
   LO
   TS
CP0648581
sodium 6-(5'-chloro-2'-isobutoxybiphenyl-2-yl)picolinate
   Show/Hide
C22H19ClNNaO3
 1
1
IC50 = 15.85 nM
   TI
   LI
   LO
   TS
CP0875503
3-(2-(2-(2-chloro-4-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H18BrClFNO3
 1
1
IC50 = 15.85 nM
   TI
   LI
   LO
   TS
CP0897819
3-(2-(5-bromo-2-(cyclopentylmethoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C24H24BrNO3
 1
1
IC50 = 15.85 nM
   TI
   LI
   LO
   TS
CP0899684
3-(2-(2-(4-(trifluoromethoxy)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C26H19BrF3NO4
 1
1
IC50 = 15.85 nM
   TI
   LI
   LO
   TS
CP0462925
4-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-N-tert-butylbenzamide
   Show/Hide
C29H27BrF2N2O2
 1
1
IC50 = 15.85 nM
   TI
   LI
   LO
   TS
CP0540240
4-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-N,N-dimethylbenzamide
   Show/Hide
C27H23BrF2N2O2
 1
1
IC50 = 15.85 nM
   TI
   LI
   LO
   TS
CP0862530
3-{2-[5-Bromo-2-(2-methyl-benzyloxy)-phenyl]-5-methyl-pyrrol-1-yl}-benzoic acid
   Show/Hide
C26H22BrNO3
 1
1
IC50 = 19.95 nM
   TI
   LI
   LO
   TS
CP0862539
3-(2-(2-(benzyloxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H21NO3
 1
1
IC50 = 19.95 nM
   TI
   LI
   LO
   TS
CP0444760
2-(5-chloro-2-phenylmethoxyphenyl)-5-methyl-1-(4-methylsulfonylphenyl)pyrrole
   Show/Hide
C25H22ClNO3S
 1
1
IC50 = 19.95 nM
   TI
   LI
   LO
   TS
CP0462927
4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzenesulfonamide
   Show/Hide
C24H21ClN2O3S
 1
1
IC50 = 19.95 nM
   TI
   LI
   LO
   TS
CP0538700
3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-N-methylbenzamide
   Show/Hide
C26H21BrF2N2O2
 1
1
IC50 = 19.95 nM
   TI
   LI
   LO
   TS
CP0920132
N-((5-(4-methoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-4-chloro-N-(2,3-dichlorophenyl)benzenesulfonamide
   Show/Hide
C23H18Cl3N3O4S
 2
1
IC50 = 19.95 nM
   TI
   LI
   LO
   TS
2
Ki = 63.1 nM
   TI
   LI
   LO
   TS
CP0932499
N-(3-chloro-2-methylphenyl)-N-((5-((4-methoxyphenylamino)methyl)-1,3,4-oxadiazol-2-yl)methyl)-4-methylbenzenesulfonamide
   Show/Hide
C25H25ClN4O4S
 2
1
IC50 = 19.95 nM
   TI
   LI
   LO
   TS
2
Ki = 79.43 nM
   TI
   LI
   LO
   TS
CP0867891
sodium 6-(5-chloro-2-(2,4-difluorobenzyloxy)benzyl)picolinate
   Show/Hide
C20H13ClF2NNaO3
 1
1
IC50 = 25.12 nM
   TI
   LI
   LO
   TS
CP0851030
3-(2-(5-bromo-2-((5-methylisoxazol-3-yl)methoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C23H19BrN2O4
 1
1
IC50 = 25.12 nM
   TI
   LI
   LO
   TS
CP0869609
3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-chloro-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C24H17Cl2NO3
 1
1
IC50 = 25.12 nM
   TI
   LI
   LO
   TS
CP0918358
3-(2-(5-chloro-2-(cyclopentylmethoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C24H24ClNO3
 1
1
IC50 = 25.12 nM
   TI
   LI
   LO
   TS
CP0920194
3-(2-(2-(benzyloxy)-5-(methylsulfonyl)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C26H23NO5S
 1
1
IC50 = 25.12 nM
   TI
   LI
   LO
   TS
CP0444759
N-benzyl-4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzamide
   Show/Hide
C32H27ClN2O2
 1
1
IC50 = 25.12 nM
   TI
   LI
   LO
   TS
CP0524536
N-benzyl-3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzamide
   Show/Hide
C32H27ClN2O2
 1
1
IC50 = 25.12 nM
   TI
   LI
   LO
   TS
CP0540241
2-[3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]phenyl]-1,1,1,3,3,3-hexafluoropropan-2-ol
   Show/Hide
C27H18BrF8NO2
 1
1
IC50 = 25.12 nM
   TI
   LI
   LO
   TS
CP0551264
5-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-2H-benzotriazole
   Show/Hide
C24H19ClN4O
 1
1
IC50 = 25.12 nM
   TI
   LI
   LO
   TS
CP0876729
N-(2-ethylphenyl)-N-((5-((4-methoxyphenoxy)methyl)-1,3,4-oxadiazol-2-yl)methyl)-4-methylbenzenesulfonamide
   Show/Hide
C26H27N3O5S
 2
1
IC50 = 25.12 nM
   TI
   LI
   LO
   TS
2
Ki = 125.89 nM
   TI
   LI
   LO
   TS
CP0867850
sodium 6-(5-chloro-2-(cyclopentylmethoxy)benzyl)picolinate
   Show/Hide
C19H19ClNNaO3
 1
1
IC50 = 31.62 nM
   TI
   LI
   LO
   TS
CP0942293
3-(2-(2-(cyclohexylmethoxy)-5-(trifluoromethyl)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C26H26F3NO3
 1
1
IC50 = 31.62 nM
   TI
   LI
   LO
   TS
CP0462929
2-(5-bromo-2-phenylmethoxyphenyl)-5-methyl-1-(4-methylsulfonylphenyl)pyrrole
   Show/Hide
C25H22BrNO3S
 1
1
IC50 = 31.62 nM
   TI
   LI
   LO
   TS
CP0876751
N-(3-chloro-2-methylphenyl)-N-((5-(4-methoxyphenylamino)-1,3,4-oxadiazol-2-yl)methyl)-4-methylbenzenesulfonamide
   Show/Hide
C24H23ClN4O4S
 2
1
IC50 = 31.62 nM
   TI
   LI
   LO
   TS
2
Ki = 79.43 nM
   TI
   LI
   LO
   TS
CP0867849
sodium 6-(5-chloro-2-(2-chlorobenzyloxy)benzyl)picolinate
   Show/Hide
C20H14Cl2NNaO3
 1
1
IC50 = 39.81 nM
   TI
   LI
   LO
   TS
CP0890928
sodium 6-(5-chloro-2-isobutoxybenzyl)picolinate
   Show/Hide
C17H17ClNNaO3
 1
1
IC50 = 39.81 nM
   TI
   LI
   LO
   TS
CP0946776
sodium 6-(5-chloro-2-(4-chlorobenzyloxy)benzyl)picolinate
   Show/Hide
C20H14Cl2NNaO3
 1
1
IC50 = 39.81 nM
   TI
   LI
   LO
   TS
CP0916323
3-(2-(2-(4-(trifluoromethyl)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C26H19BrF3NO3
 1
1
IC50 = 39.81 nM
   TI
   LI
   LO
   TS
CP0916448
3-(2-(5-bromo-2-(cyclohexylmethoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H26BrNO3
 1
1
IC50 = 39.81 nM
   TI
   LI
   LO
   TS
CP0941234
3-(2-(5-chloro-2-((tetrahydrofuran-2-yl)methoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C23H22ClNO4
 1
1
IC50 = 39.81 nM
   TI
   LI
   LO
   TS
CP0942292
3-(2-(5-chloro-2-((tetrahydro-2H-pyran-4-yl)methoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C24H24ClNO4
 1
1
IC50 = 39.81 nM
   TI
   LI
   LO
   TS
CP0439539
6-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-1H-indazole
   Show/Hide
C25H20ClN3O
 1
1
IC50 = 39.81 nM
   TI
   LI
   LO
   TS
CP0484290
2-[3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]phenyl]-5-methyl-1,3,4-oxadiazole
   Show/Hide
C27H20BrF2N3O2
 1
1
IC50 = 39.81 nM
   TI
   LI
   LO
   TS
CP0485320
5-[4-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]phenyl]-1H-imidazole
   Show/Hide
C27H20BrF2N3O
 1
1
IC50 = 39.81 nM
   TI
   LI
   LO
   TS
CP0510800
3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-[(1R)-1-phenylethyl]benzamide
   Show/Hide
C33H29ClN2O2
 1
1
IC50 = 39.81 nM
   TI
   LI
   LO
   TS
CP0538699
5-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-1H-indazole
   Show/Hide
C25H20ClN3O
 1
1
IC50 = 39.81 nM
   TI
   LI
   LO
   TS
CP0942621
N-(2,3-dichlorophenyl)-N-((5-(4-methoxyphenylamino)-1,3,4-oxadiazol-2-yl)methyl)-4-methylbenzenesulfonamide
   Show/Hide
C23H20Cl2N4O4S
 2
1
IC50 = 39.81 nM
   TI
   LI
   LO
   TS
2
Ki = 50.12 nM
   TI
   LI
   LO
   TS
CP0855112
3-(2-(2-(4-methoxybenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C26H22BrNO4
 1
1
IC50 = 50.12 nM
   TI
   LI
   LO
   TS
CP0916322
3-(2-(2-(3-methoxybenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C26H22BrNO4
 1
1
IC50 = 50.12 nM
   TI
   LI
   LO
   TS
CP0394640
3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-(pyridin-2-ylmethyl)benzamide
   Show/Hide
C31H26ClN3O2
 1
1
IC50 = 50.12 nM
   TI
   LI
   LO
   TS
CP0538701
4-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-N,N-diethylbenzamide
   Show/Hide
C29H27BrF2N2O2
 1
1
IC50 = 50.12 nM
   TI
   LI
   LO
   TS
CP0910970
N-((5-(4-(trifluoromethyl)benzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
   Show/Hide
C25H21ClF3N3O3S
 2
1
IC50 = 50.12 nM
   TI
   LI
   LO
   TS
2
Ki = 158.49 nM
   TI
   LI
   LO
   TS
CP0394728
7-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-4-methyl-1H-quinolin-2-one
   Show/Hide
C28H23ClN2O2
 1
1
IC50 = 63.1 nM
   TI
   LI
   LO
   TS
CP0439445
2-[3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]phenyl]-1H-benzimidazole
   Show/Hide
C31H22BrF2N3O
 1
1
IC50 = 63.1 nM
   TI
   LI
   LO
   TS
CP0439447
3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-(pyridin-3-ylmethyl)benzamide
   Show/Hide
C31H26ClN3O2
 1
1
IC50 = 63.1 nM
   TI
   LI
   LO
   TS
CP0439540
4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-(pyridin-4-ylmethyl)benzamide
   Show/Hide
C31H26ClN3O2
 1
1
IC50 = 63.1 nM
   TI
   LI
   LO
   TS
CP0484293
3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-(pyridin-4-ylmethyl)benzamide
   Show/Hide
C31H26ClN3O2
 1
1
IC50 = 63.1 nM
   TI
   LI
   LO
   TS
CP0505267
3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzamide
   Show/Hide
C25H21ClN2O2
 1
1
IC50 = 63.1 nM
   TI
   LI
   LO
   TS
CP0540237
N-[3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]phenyl]acetamide
   Show/Hide
C26H23ClN2O2
 1
1
IC50 = 63.1 nM
   TI
   LI
   LO
   TS
CP0879922
N-((5-(4-methoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-4-methyl-N-(2-methyl-3-(trifluoromethyl)phenyl)benzenesulfonamide
   Show/Hide
C26H24F3N3O4S
 2
1
IC50 = 63.1 nM
   TI
   LI
   LO
   TS
2
Ki = 398.11 nM
   TI
   LI
   LO
   TS
CP0920139
N-((5-(2,6-dichlorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
   Show/Hide
C24H20Cl3N3O3S
 2
1
IC50 = 63.1 nM
   TI
   LI
   LO
   TS
2
Ki = 501.19 nM
   TI
   LI
   LO
   TS
CP0947170
N-((5-(2,4-dichlorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
   Show/Hide
C24H20Cl3N3O3S
 2
1
IC50 = 63.1 nM
   TI
   LI
   LO
   TS
2
Ki = 1000 nM
   TI
   LI
   LO
   TS
CP0867890
sodium 6-(5-chloro-2-(2-fluorobenzyloxy)benzyl)picolinate
   Show/Hide
C20H14ClFNNaO3
 1
1
IC50 = 79.43 nM
   TI
   LI
   LO
   TS
CP0928358
sodium 6-(5-chloro-2-(2,4,6-trifluorobenzyloxy)benzyl)picolinate
   Show/Hide
C20H12ClF3NNaO3
 1
1
IC50 = 79.43 nM
   TI
   LI
   LO
   TS
CP0851021
3-(2-(2-(benzyloxy)-5-bromophenyl)-5-ethyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C26H22BrNO3
 1
1
IC50 = 79.43 nM
   TI
   LI
   LO
   TS
CP0853242
3-(2-(2-(3-(difluoromethoxy)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C26H20BrF2NO4
 1
1
IC50 = 79.43 nM
   TI
   LI
   LO
   TS
CP0538703
N-[3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]phenyl]sulfonylbenzamide
   Show/Hide
C31H25ClN2O4S
 1
1
IC50 = 79.43 nM
   TI
   LI
   LO
   TS
CP0876754
N-((5-(2-chlorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
   Show/Hide
C24H21Cl2N3O3S
 2
1
IC50 = 79.43 nM
   TI
   LI
   LO
   TS
2
Ki = 398.11 nM
   TI
   LI
   LO
   TS
CP0906801
sodium 6-(5-chloro-2-(cyclohexylmethoxy)benzyl)picolinate
   Show/Hide
C20H21ClNNaO3
 1
1
IC50 = 100 nM
   TI
   LI
   LO
   TS
CP0935423
sodium 6-(5-chloro-2-(4-fluorobenzyloxy)benzyl)picolinate
   Show/Hide
C20H14ClFNNaO3
 1
1
IC50 = 100 nM
   TI
   LI
   LO
   TS
CP0862527
3-(2-(2-(3,4-dichlorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H18BrCl2NO3
 1
1
IC50 = 100 nM
   TI
   LI
   LO
   TS
CP0916446
3-(2-(2-(2-fluoro-6-(trifluoromethyl)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C26H18BrF4NO3
 1
1
IC50 = 100 nM
   TI
   LI
   LO
   TS
CP0921558
3-(2-(2-(2,4-difluorobenzyloxy)-5-chlorophenyl)-5-(trifluoromethyl)-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H15ClF5NO3
 1
1
IC50 = 100 nM
   TI
   LI
   LO
   TS
CP0922210
3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-ethyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C26H22ClNO3
 1
1
IC50 = 100 nM
   TI
   LI
   LO
   TS
CP0853249
3-(2-(5-chloro-2-(cyclohexylmethoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H26ClNO3
 1
1
IC50 = 125.89 nM
   TI
   LI
   LO
   TS
CP0485041
3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-4-ethoxybenzoic acid
   Show/Hide
C27H24ClNO4
 1
1
IC50 = 125.89 nM
   TI
   LI
   LO
   TS
CP0400069
2-(5-chloro-2-phenylmethoxyphenyl)-5-methyl-1-(3-methylsulfonylphenyl)pyrrole
   Show/Hide
C25H22ClNO3S
 1
1
IC50 = 125.89 nM
   TI
   LI
   LO
   TS
CP0524535
3-[3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]phenyl]pyridine
   Show/Hide
C29H21BrF2N2O
 1
1
IC50 = 125.89 nM
   TI
   LI
   LO
   TS
CP0540238
2-[3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]phenyl]pyrimidine
   Show/Hide
C28H20BrF2N3O
 1
1
IC50 = 125.89 nM
   TI
   LI
   LO
   TS
CP0935660
N-((5-(4-ethoxybenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(2-ethylphenyl)-4-methylbenzenesulfonamide
   Show/Hide
C27H29N3O4S
 2
1
IC50 = 125.89 nM
   TI
   LI
   LO
   TS
2
Ki = 39.81 nM
   TI
   LI
   LO
   TS
CP0878525
sodium 6-(2-(benzyloxy)-5-chlorobenzyl)picolinate
   Show/Hide
C20H15ClNNaO3
 1
1
IC50 = 158.49 nM
   TI
   LI
   LO
   TS
CP0562588
4-chloro-3-[2-[5-chloro-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C25H17Cl2F2NO3
 1
1
IC50 = 158.49 nM
   TI
   LI
   LO
   TS
CP0439444
5-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]isoindole-1,3-dione
   Show/Hide
C26H17BrF2N2O3
 1
1
IC50 = 158.49 nM
   TI
   LI
   LO
   TS
CP0918609
N-((5-(3-chlorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
   Show/Hide
C24H21Cl2N3O3S
 2
1
IC50 = 158.49 nM
   TI
   LI
   LO
   TS
2
Ki = 1995.26 nM
   TI
   LI
   LO
   TS
CP0891913
sodium 6-(5-chloro-2-(cyclopropylmethoxy)benzyl)picolinate
   Show/Hide
C17H15ClNNaO3
 1
1
IC50 = 199.53 nM
   TI
   LI
   LO
   TS
CP0851031
3-(2-(5-bromo-2-((3,5-dimethylisoxazol-4-yl)methoxy)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C24H21BrN2O4
 1
1
IC50 = 199.53 nM
   TI
   LI
   LO
   TS
CP0918718
3-(2-(2-(4-fluorobenzyloxy)-5-chlorophenyl)-5-(trifluoromethyl)-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H16ClF4NO3
 1
1
IC50 = 199.53 nM
   TI
   LI
   LO
   TS
CP0538698
3-[3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]phenyl]-5-methyl-1,2,4-oxadiazole
   Show/Hide
C27H20BrF2N3O2
 1
1
IC50 = 199.53 nM
   TI
   LI
   LO
   TS
CP0538702
2-(5-bromo-2-phenylmethoxyphenyl)-5-methyl-1-(3-methylsulfonylphenyl)pyrrole
   Show/Hide
C25H22BrNO3S
 1
1
IC50 = 199.53 nM
   TI
   LI
   LO
   TS
CP0858980
N-((5-(4-fluorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
   Show/Hide
C24H21ClFN3O3S
 2
1
IC50 = 199.53 nM
   TI
   LI
   LO
   TS
2
Ki = 501.19 nM
   TI
   LI
   LO
   TS
CP0851029
3-(2-(2-(3-(trifluoromethyl)benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C26H19BrF3NO3
 1
1
IC50 = 251.19 nM
   TI
   LI
   LO
   TS
CP0485412
3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-4-methoxybenzoic acid
   Show/Hide
C26H22ClNO4
 1
1
IC50 = 251.19 nM
   TI
   LI
   LO
   TS
CP0505265
2-[3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]phenyl]pyridine
   Show/Hide
C29H21BrF2N2O
 1
1
IC50 = 251.19 nM
   TI
   LI
   LO
   TS
CP0652436
N-(4-chlorophenethyl)-2-(4-methyl-N-o-tolylphenylsulfonamido)acetamide
   Show/Hide
C24H25ClN2O3S
 1
1
IC50 = 251.19 nM
   TI
   LI
   LO
   TS
CP0434071
4-chloro-3-[2-[5-chloro-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
   Show/Hide
C25H18Cl2FNO3
 1
1
IC50 = 316.23 nM
   TI
   LI
   LO
   TS
CP0505266
3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-[(1S)-1-phenylethyl]benzamide
   Show/Hide
C33H29ClN2O2
 1
1
IC50 = 316.23 nM
   TI
   LI
   LO
   TS
CP0949627
N-((5-(3-fluorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
   Show/Hide
C24H21ClFN3O3S
 2
1
IC50 = 316.23 nM
   TI
   LI
   LO
   TS
2
Ki = 501.19 nM
   TI
   LI
   LO
   TS
CP0910942
3-[2-(4-Benzyloxy-biphenyl-3-yl)-5-methyl-pyrrol-1-yl]-benzoic acid
   Show/Hide
C31H25NO3
 1
1
IC50 = 398.11 nM
   TI
   LI
   LO
   TS
CP0920138
N-((5-(4-chlorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(2-ethylphenyl)-4-methylbenzenesulfonamide
   Show/Hide
C25H24ClN3O3S
 2
1
IC50 = 398.11 nM
   TI
   LI
   LO
   TS
2
Ki = 316.23 nM
   TI
   LI
   LO
   TS
CP0485319
1-[4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]phenyl]-1,2,4-triazole
   Show/Hide
C26H21ClN4O
 1
1
IC50 = 501.19 nM
   TI
   LI
   LO
   TS
CP0497528
2-methyl-1-(4-methylsulfonylphenyl)-5-(2-phenylmethoxyphenyl)pyrrole
   Show/Hide
C25H23NO3S
 1
1
IC50 = 501.19 nM
   TI
   LI
   LO
   TS
CP0522232
3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-N-phenylbenzamide
   Show/Hide
C31H23BrF2N2O2
 1
1
IC50 = 501.19 nM
   TI
   LI
   LO
   TS
CP0540239
3-[2-[2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzamide
   Show/Hide
C25H20F2N2O2
 1
1
IC50 = 501.19 nM
   TI
   LI
   LO
   TS
CP0876731
N-(2-ethylphenyl)-N-((5-((4-methoxyphenylamino)methyl)-1,3,4-oxadiazol-2-yl)methyl)-4-methylbenzenesulfonamide
   Show/Hide
C26H28N4O4S
 2
1
IC50 = 501.19 nM
   TI
   LI
   LO
   TS
2
Ki = 794.33 nM
   TI
   LI
   LO
   TS
CP0945695
N-((5-(2-fluorobenzyl)-1,3,4-oxadiazol-2-yl)methyl)-N-(3-chloro-2-methylphenyl)-4-methylbenzenesulfonamide
   Show/Hide
C24H21ClFN3O3S
 2
1
IC50 = 501.19 nM
   TI
   LI
   LO
   TS
2
Ki = 630.96 nM
   TI
   LI
   LO
   TS
CP0875506
3-(2-(2-(benzyloxy)-5-(thiophen-3-yl)phenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C29H23NO3S
 1
1
IC50 = 630.96 nM
   TI
   LI
   LO
   TS
CP0497524
5-[2-[2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-2H-benzotriazole
   Show/Hide
C24H18F2N4O
 1
1
IC50 = 630.96 nM
   TI
   LI
   LO
   TS
CP0862536
3-(5-(2-(benzyloxy)-5-chlorophenyl)-3-bromo-2-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H19BrClNO3
 1
1
IC50 = 794.33 nM
   TI
   LI
   LO
   TS
CP0916164
N-((5-benzyl-1,3,4-oxadiazol-2-yl)methyl)-N-(2-ethylphenyl)-4-methylbenzenesulfonamide
   Show/Hide
C25H25N3O3S
 2
1
IC50 = 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 398.11 nM
   TI
   LI
   LO
   TS
CP0427396
4-[(1S)-1-[[5-phenyl-3-[[4-(trifluoromethyl)phenyl]methyl]triazole-4-carbonyl]amino]ethyl]benzoic acid
   Show/Hide
C26H21F3N4O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0427397
4-[(1S)-1-[[5-(cyclopenten-1-yl)-3-[[4-(trifluoromethyl)phenyl]methyl]triazole-4-carbonyl]amino]ethyl]benzoic acid
   Show/Hide
C25H23F3N4O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0435681
US8686018, 107
   Show/Hide
C22H18F5N3O4
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0438577
4-[(1S)-1-[[5-phenyl-3-[2-[3-(trifluoromethyl)phenoxy]ethyl]triazole-4-carbonyl]amino]ethyl]benzoic acid
   Show/Hide
C27H23F3N4O4
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0438580
4-[(1S)-1-[[5-(furan-3-yl)-3-[[4-(trifluoromethyl)phenyl]methyl]triazole-4-carbonyl]amino]ethyl]benzoic acid
   Show/Hide
C24H19F3N4O4
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0473341
4-[(1S)-1-[[5-(5-methylthiophen-2-yl)-3-[[4-(trifluoromethyl)phenyl]methyl]triazole-4-carbonyl]amino]ethyl]benzoic acid
   Show/Hide
C25H21F3N4O3S
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0473342
4-[(1S)-1-[[5-thiophen-3-yl-3-[[4-(trifluoromethyl)phenyl]methyl]triazole-4-carbonyl]amino]ethyl]benzoic acid
   Show/Hide
C24H19F3N4O3S
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0473344
4-[(1S)-1-[[5-[(E)-prop-1-enyl]-3-[[4-(trifluoromethyl)phenyl]methyl]triazole-4-carbonyl]amino]ethyl]benzoic acid
   Show/Hide
C23H21F3N4O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0477510
4-[(1S)-1-[[5-prop-1-ynyl-3-[[4-(trifluoromethyl)phenyl]methyl]triazole-4-carbonyl]amino]ethyl]benzoic acid
   Show/Hide
C23H19F3N4O3
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0477511
4-[(1S)-1-[[3-[2-(4-fluorophenoxy)ethyl]-5-phenyltriazole-4-carbonyl]amino]ethyl]benzoic acid
   Show/Hide
C26H23FN4O4
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0853250
3-(5-(2-(benzyloxy)-5-chlorophenyl)-2-methyl-3-phenyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C31H24ClNO3
 1
1
IC50 < 1000 nM
   TI
   LI
   LO
   TS
CP0875505
3-(5-(2-(benzyloxy)-5-chlorophenyl)-3-chloro-2-methyl-1H-pyrrol-1-yl)benzoic acid
   Show/Hide
C25H19Cl2NO3
 1
1
IC50 < 1000 nM
   TI
   LI
   LO
   TS
CP0910605
2-(2-(benzyloxy)phenyl)-5-methyl-1-(3-(methylsulfonyl)phenyl)-1H-pyrrole
   Show/Hide
C25H23NO3S
 1
1
IC50 < 1000 nM
   TI
   LI
   LO
   TS
CP0882825
N-((5-(4-methoxyphenoxy)-1,3,4-oxadiazol-2-yl)methyl)-N-(2-ethylphenyl)-4-methylbenzenesulfonamide
   Show/Hide
C25H25N3O5S
 2
1
IC50 < 1000 nM
   TI
   LI
   LO
   TS
2
Ki = 100 nM
   TI
   LI
   LO
   TS
CP0383448
5-[2-[5-chloro-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-2-methylbenzoic acid
   Show/Hide
C26H21ClFNO3
 1
1
Ki = 1 nM
   TI
   LI
   LO
   TS
CP0035659
N-[(4-chlorophenyl)methyl]-2-(2-ethyl-N-(4-methylphenyl)sulfonylanilino)acetamide
   Show/Hide
C24H25ClN2O3S
 1
1
Ki = 10 nM
   TI
   LI
   LO
   TS
CP0484317
2-(2-ethyl-N-(4-methylphenyl)sulfonylanilino)-N-[(4-methoxyphenyl)methyl]acetamide
   Show/Hide
C25H28N2O4S
 1
1
Ki = 25.12 nM
   TI
   LI
   LO
   TS
CP0915923
N-(3,4-dimethoxybenzyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
   Show/Hide
C26H30N2O5S
 1
1
Ki = 25.12 nM
   TI
   LI
   LO
   TS
CP0897849
N-benzyl-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
   Show/Hide
C24H26N2O3S
 1
1
Ki = 63.1 nM
   TI
   LI
   LO
   TS
CP0882726
N-(3-methoxybenzyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
   Show/Hide
C25H28N2O4S
 1
1
Ki = 79.43 nM
   TI
   LI
   LO
   TS
CP0915906
N-(4-chlorobenzyl)-2-(N-(1-ethyl-1H-pyrazol-5-yl)-4-methylphenylsulfonamido)acetamide
   Show/Hide
C21H23ClN4O3S
 1
1
Ki = 158.49 nM
   TI
   LI
   LO
   TS
CP0844852
N-(4-chlorobenzyl)-2-(4-methyl-N-(2-methylpyridin-3-yl)phenylsulfonamido)acetamide
   Show/Hide
C22H22ClN3O3S
 1
1
Ki = 199.53 nM
   TI
   LI
   LO
   TS
CP0939750
N-(3-chlorobenzyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
   Show/Hide
C24H25ClN2O3S
 1
1
Ki = 251.19 nM
   TI
   LI
   LO
   TS
CP0844860
N-(4-chlorobenzyl)-2-(4-methyl-N-(1-methyl-1H-pyrazol-5-yl)phenylsulfonamido)acetamide
   Show/Hide
C20H21ClN4O3S
 1
1
Ki = 398.11 nM
   TI
   LI
   LO
   TS
CP0427199
N-(2-ethylphenyl)-N-[[5-[(4-methoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl]methyl]-4-methylbenzenesulfonamide
   Show/Hide
C26H27N3O4S
 1
1
Ki = 630.96 nM
   TI
   LI
   LO
   TS
CP0942223
N-(4-chlorobenzyl)-2-(4-methyl-N-(3-methylpyridin-2-yl)phenylsulfonamido)acetamide
   Show/Hide
C22H22ClN3O3S
 1
1
Ki = 794.33 nM
   TI
   LI
   LO
   TS
CP0895712
N-(4-chlorobenzyl)-2-(4-methyl-N-(6-methylpyridin-3-yl)phenylsulfonamido)acetamide
   Show/Hide
C22H22ClN3O3S
 1
1
Ki < 1000 nM
   TI
   LI
   LO
   TS
CP0902805
N-(4-chlorobenzyl)-2-(4-methyl-N-(6-methylpyridin-2-yl)phenylsulfonamido)acetamide
   Show/Hide
C22H22ClN3O3S
 1
1
Ki < 1000 nM
   TI
   LI
   LO
   TS
CP0915907
N-(4-chlorobenzyl)-2-(4-methyl-N-(pyridin-2-yl)phenylsulfonamido)acetamide
   Show/Hide
C21H20ClN3O3S
 1
1
Ki < 1000 nM
   TI
   LI
   LO
   TS
CP0918668
N-(4-chlorobenzyl)-2-(4-methyl-N-(pyridin-3-yl)phenylsulfonamido)acetamide
   Show/Hide
C21H20ClN3O3S
 1
1
Ki < 1000 nM
   TI
   LI
   LO
   TS
CP0918673
N-(4-chlorobenzyl)-2-(4-methyl-N-(5-methylpyridin-2-yl)phenylsulfonamido)acetamide
   Show/Hide
C22H22ClN3O3S
 1
1
Ki < 1000 nM
   TI
   LI
   LO
   TS