| Compound ID |
Compound Name |
Compound Formula |
|
CP0239863
|
2-[(3-chlorophenyl)methoxy]-4-(1-hydroxy-3,4-dihydro-2,1-benzoxaborinin-3-yl)benzenecarboximidamide;hydrochloride
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|
C22H21BCl2N2O3
|
1
|
| 1 |
IC50 = 63.1 nM
|
|
|
|
CP0384876
|
ethyl 4-[(2R)-3-(3-carbamimidoylphenyl)-2-[[2,4,6-tri(propan-2-yl)phenyl]sulfonylamino]propanoyl]piperazine-1-carboxylate
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|
C32H47N5O5S
|
1
|
| 1 |
IC50 = 285 nM
|
|
|
|
CP0067298
|
(E,E)-2,7-Bis(4-amidinobenzylidine)cycloheptan-1-one
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|
C23H24N4O
|
1
|
| 1 |
IC50 = 484 nM
|
|
|
|
CP0548645
|
2-benzyl-N-(4-carbamimidoylphenyl)-3-[(4-methylphenyl)sulfonylamino]propanamide
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|
C24H26N4O3S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0326107
|
1-[(2S)-3-(3-carbamimidoylphenyl)-2-(naphthalen-2-ylsulfonylamino)propanoyl]-N-(thiophen-2-ylmethyl)piperidine-3-carboxamide
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|
C31H33N5O4S2
|
2
|
| 1 |
IC50 = 2430 nM
|
|
|
| 2 |
IC50 = 6000 nM
|
|
|
|
CP0521053
|
N-(4-carbamimidoylphenyl)-2-[(4-methylphenyl)sulfonylamino]hexanamide
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|
C20H26N4O3S
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0064994
|
(2R)-N-(4-carbamimidoylphenyl)-2-cyclohexyl-2-[(4-methylphenyl)sulfonylamino]acetamide
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|
C22H28N4O3S
|
2
|
| 1 |
IC50 = 4400 nM
|
|
|
| 2 |
IC50 > 10000 nM
|
|
|
|
CP0521056
|
(2R)-N-(4-carbamimidoylphenyl)-2-cyclohexyl-2-[[4-(trifluoromethyl)phenyl]sulfonylamino]acetamide
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|
C22H25F3N4O3S
|
1
|
| 1 |
IC50 = 4700 nM
|
|
|
|
CP0354488
|
4-(1-hydroxy-8-methyl-3,4-dihydro-2,1-benzoxaborinin-3-yl)-2-(pyridin-3-ylmethoxy)benzenecarboximidamide;hydrochloride
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|
C22H23BClN3O3
|
1
|
| 1 |
IC50 = 5011.87 nM
|
|
|
|
CP0558973
|
N-(4-carbamimidoylphenyl)-1-(4-methylphenyl)sulfonylpyrrolidine-2-carboxamide
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|
C19H22N4O3S
|
1
|
| 1 |
IC50 = 5300 nM
|
|
|
|
CP0521796
|
N-(4-carbamimidoylphenyl)-3-methyl-2-[(4-methylphenyl)sulfonylamino]butanamide
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|
C19H24N4O3S
|
1
|
| 1 |
IC50 = 7200 nM
|
|
|
|
CP0164331
|
4-[(3R)-1-hydroxy-7-(trifluoromethyl)-3,4-dihydro-2,1-benzoxaborinin-3-yl]-2-(pyridin-3-ylmethoxy)benzenecarboximidamide;hydrochloride
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|
C22H20BClF3N3O3
|
1
|
| 1 |
IC50 = 7943.28 nM
|
|
|
|
CP0513705
|
N-(4-carbamimidoyl-2-fluorophenyl)-2-[(4-methylphenyl)sulfonylamino]hexanamide
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|
C20H25FN4O3S
|
1
|
| 1 |
IC50 = 8000 nM
|
|
|
|
CP0216665
|
3-(3-Carbamimidoyl-phenyl)-2-[2-(toluene-4-sulfonylamino)-acetylamino]-propionic acid methyl ester
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|
C20H24N4O5S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0417006
|
N-(4-carbamimidoylphenyl)-2-[(4-methylphenyl)sulfonylamino]-4-phenylbutanamide
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|
C24H26N4O3S
|
2
|
| 1 |
IC50 > 10000 nM
|
|
|
| 2 |
IC50 = 26000 nM
|
|
|
|
CP0513704
|
N-(4-carbamimidoylphenyl)-4-methyl-2-[(4-methylphenyl)sulfonylamino]pentanamide
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|
C20H26N4O3S
|
1
|
| 1 |
IC50 = 11000 nM
|
|
|
|
CP0485679
|
(2R)-N-(4-carbamimidoylphenyl)-2-cyclohexyl-2-[(4-methoxyphenyl)sulfonylamino]acetamide
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|
C22H28N4O4S
|
1
|
| 1 |
IC50 = 12000 nM
|
|
|
|
CP0438055
|
4-[1-hydroxy-7-(trifluoromethyl)-3,4-dihydro-2,1-benzoxaborinin-3-yl]-2-(pyridin-3-ylmethoxy)benzenecarboximidamide;hydrochloride
Show/Hide
|
C22H20BClF3N3O3
|
1
|
| 1 |
IC50 = 12589.25 nM
|
|
|
|
CP0099151
|
(2R)-N-(4-carbamimidoylphenyl)-2-cyclohexyl-2-[(4-fluorophenyl)sulfonylamino]acetamide
Show/Hide
|
C21H25FN4O3S
|
1
|
| 1 |
IC50 > 14000 nM
|
|
|
|
CP0558969
|
N-(4-carbamimidoylphenyl)-3-cyclopentyl-2-[(4-methylphenyl)sulfonylamino]propanamide
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|
C22H28N4O3S
|
1
|
| 1 |
IC50 = 16000 nM
|
|
|
|
CP0549822
|
(2R)-N-(4-carbamimidoylphenyl)-2-[(4-chlorophenyl)sulfonylamino]-2-cyclohexylacetamide
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|
C21H25ClN4O3S
|
1
|
| 1 |
IC50 = 18000 nM
|
|
|
|
CP0558972
|
N-(4-carbamimidoylphenyl)-2-[(4-methylphenyl)sulfonylamino]-2-(oxan-4-yl)acetamide
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|
C21H26N4O4S
|
1
|
| 1 |
IC50 > 19000 nM
|
|
|
|
CP0560431
|
N-(3-carbamimidoylphenyl)-2-[(4-methylphenyl)sulfonylamino]hexanamide
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|
C20H26N4O3S
|
1
|
| 1 |
IC50 = 19000 nM
|
|
|
|
CP0549821
|
(2R)-2-(benzenesulfonamido)-N-(4-carbamimidoylphenyl)-2-cyclohexylacetamide
Show/Hide
|
C21H26N4O3S
|
1
|
| 1 |
IC50 = 22000 nM
|
|
|
|
CP0558971
|
N-(4-carbamimidoylphenyl)-4-methyl-2-[methyl-(4-methylphenyl)sulfonylamino]pentanamide
Show/Hide
|
C21H28N4O3S
|
1
|
| 1 |
IC50 = 24000 nM
|
|
|
|
CP0521055
|
N-[(1R)-2-(4-carbamimidoylanilino)-1-cyclohexyl-2-oxoethyl]-4-methylbenzamide
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|
C23H28N4O2
|
1
|
| 1 |
IC50 = 24500 nM
|
|
|
|
CP0485687
|
(2R)-N-(4-carbamimidoylphenyl)-2-cyclohexyl-2-[(4-methylphenyl)carbamoylamino]acetamide
Show/Hide
|
C23H29N5O2
|
1
|
| 1 |
IC50 = 43000 nM
|
|
|
|
CP0250361
|
2-[(2-chlorophenyl)methoxy]-4-(1-hydroxy-3,4-dihydro-2,1-benzoxaborinin-3-yl)benzenecarboximidamide;hydrochloride
Show/Hide
|
C22H21BCl2N2O3
|
1
|
| 1 |
IC50 = 50118.72 nM
|
|
|
|
CP0360969
|
4-(1-hydroxy-3,4-dihydro-2,1-benzoxaborinin-3-yl)-2-(pyridin-3-ylmethoxy)benzenecarboximidamide;hydrochloride
Show/Hide
|
C21H21BClN3O3
|
1
|
| 1 |
IC50 = 50118.72 nM
|
|
|
|
CP0537151
|
N-(4-bromophenyl)-2-[(4-methylphenyl)sulfonylamino]hexanamide
Show/Hide
|
C19H23BrN2O3S
|
1
|
| 1 |
IC50 = 58000 nM
|
|
|
|
CP0548644
|
N-(4-carbamimidoylphenyl)-2-[(4-methylphenyl)sulfonylamino]-2-phenylacetamide
Show/Hide
|
C22H22N4O3S
|
1
|
| 1 |
IC50 = 60000 nM
|
|
|
|
CP0521054
|
N-(4-carbamimidoylphenyl)-2-cyclopentyl-2-[(4-methylphenyl)sulfonylamino]acetamide
Show/Hide
|
C21H26N4O3S
|
1
|
| 1 |
IC50 = 64000 nM
|
|
|
|
CP0558970
|
N-(4-carbamimidoylphenyl)-3-cyclohexyl-3-[(4-methylphenyl)sulfonylamino]propanamide
Show/Hide
|
C23H30N4O3S
|
1
|
| 1 |
IC50 = 68000 nM
|
|
|
|
CP0239864
|
4-[(1-hydroxy-3H-2,1-benzoxaborol-3-yl)methyl]-2-(pyridin-3-ylmethoxy)benzenecarboximidamide;hydrochloride
Show/Hide
|
C21H21BClN3O3
|
1
|
| 1 |
IC50 = 79432.82 nM
|
|
|
|
CP0354490
|
4-(6-chloro-7-fluoro-1-hydroxy-3,4-dihydro-2,1-benzoxaborinin-3-yl)-2-(pyridin-3-ylmethoxy)benzenecarboximidamide;hydrochloride
Show/Hide
|
C21H19BCl2FN3O3
|
1
|
| 1 |
IC50 = 79432.82 nM
|
|
|
|
CP0477255
|
4-[(6-fluoro-1-hydroxy-3H-2,1-benzoxaborol-3-yl)methyl]-2-(pyridin-3-ylmethoxy)benzenecarboximidamide;hydrochloride
Show/Hide
|
C21H20BClFN3O3
|
1
|
| 1 |
IC50 = 79432.82 nM
|
|
|
|
CP0063723
|
4-[(5-phenyl-1H-imidazol-2-yl)methylamino]-2-(pyridin-3-ylmethoxy)benzenecarboximidamide
Show/Hide
|
C23H22N6O
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0239865
|
4-[(1-hydroxy-5-methoxy-3H-2,1-benzoxaborol-3-yl)methyl]-2-(pyridin-3-ylmethoxy)benzenecarboximidamide;hydrochloride
Show/Hide
|
C22H23BClN3O4
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0340135
|
4-[[1-hydroxy-6-(trifluoromethyl)-3H-2,1-benzoxaborol-3-yl]methyl]-2-(pyridin-3-ylmethoxy)benzenecarboximidamide;hydrochloride
Show/Hide
|
C22H20BClF3N3O3
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0340136
|
4-[(5-fluoro-1-hydroxy-3H-2,1-benzoxaborol-3-yl)methyl]-2-(pyridin-3-ylmethoxy)benzenecarboximidamide;hydrochloride
Show/Hide
|
C21H20BClFN3O3
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0360970
|
4-[(1-hydroxy-5-methyl-3H-2,1-benzoxaborol-3-yl)methyl]-2-(pyridin-3-ylmethoxy)benzenecarboximidamide;hydrochloride
Show/Hide
|
C22H23BClN3O3
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0360971
|
4-[(3S)-1-hydroxy-7-(trifluoromethyl)-3,4-dihydro-2,1-benzoxaborinin-3-yl]-2-(pyridin-3-ylmethoxy)benzenecarboximidamide;hydrochloride
Show/Hide
|
C22H20BClF3N3O3
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
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CP0477254
|
4-(7-fluoro-1-hydroxy-3,4-dihydro-2,1-benzoxaborinin-3-yl)-2-(pyridin-3-ylmethoxy)benzenecarboximidamide;hydrochloride
Show/Hide
|
C21H20BClFN3O3
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
