| Compound ID |
Compound Name |
Compound Formula |
|
CP0062259
|
(R)-N-(2-(1-(2-(1-benzoylpiperidin-4-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
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|
C28H33F3N4O3
|
1
|
| 1 |
IC50 = 580 nM
|
|
|
|
CP0185499
|
(R)-N-(2-(1-(2,4-dimethylbenzyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
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|
C23H26F3N3O2
|
1
|
| 1 |
IC50 = 610 nM
|
|
|
|
CP0168060
|
(R)-N-(2-(1-(2-(4-benzoylpiperazin-1-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
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|
C27H32F3N5O3
|
1
|
| 1 |
IC50 = 990 nM
|
|
|
|
CP0504524
|
(R)-N-(2-(1-(2-(1-(4-methylbenzoyl)piperidin-4-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
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|
C29H35F3N4O3
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0095368
|
(R)-N-(2-(1-(2-(4-(2-chlorobenzoyl)piperazin-1-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
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|
C27H31ClF3N5O3
|
1
|
| 1 |
IC50 = 1120 nM
|
|
|
|
CP0039053
|
(R)-N-(2-(1-(2-(1-(2-fluorobenzoyl)piperidin-4-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
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|
C28H32F4N4O3
|
1
|
| 1 |
IC50 = 1130 nM
|
|
|
|
CP0507685
|
(R)-N-(2-(1-(2-(1-(3-methylbenzoyl)piperidin-4-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
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|
C29H35F3N4O3
|
1
|
| 1 |
IC50 = 1180 nM
|
|
|
|
CP0504522
|
(1S,3R)-N-(3,5-bis(trifluoromethyl)benzyl)-1-isopropyl-3-((3S,4S)-3-methyltetrahydro-2H-pyran-4-ylamino)cyclopentanecarboxamide
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|
C24H32F6N2O2
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0062257
|
(R)-N-(2-(1-(2-(1-(2-chlorobenzoyl)piperidin-4-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
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|
C28H32ClF3N4O3
|
1
|
| 1 |
IC50 = 1310 nM
|
|
|
|
CP0095364
|
(R)-N-(2-(1-(2-(1-(2,5-difluorobenzoyl)piperidin-4-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
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|
C28H31F5N4O3
|
1
|
| 1 |
IC50 = 1410 nM
|
|
|
|
CP0504525
|
(R)-N-(2-oxo-2-(1-(2-(1-(4-propylbenzoyl)piperidin-4-yl)ethyl)pyrrolidin-3-ylamino)ethyl)-3-(trifluoromethyl)benzamide
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|
C31H39F3N4O3
|
1
|
| 1 |
IC50 = 1730 nM
|
|
|
|
CP0507684
|
(R)-N-(2-(1-(2-(1-(4-ethylbenzoyl)piperidin-4-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
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|
C30H37F3N4O3
|
1
|
| 1 |
IC50 = 1740 nM
|
|
|
|
CP0039052
|
(R)-N-(2-(1-(2-(4-(2-fluorobenzoyl)piperazin-1-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C27H31F4N5O3
|
1
|
| 1 |
IC50 = 1880 nM
|
|
|
|
CP0504523
|
(R)-N-(2-oxo-2-(1-(2-(1-(4-(trifluoromethyl)benzoyl)piperidin-4-yl)ethyl)pyrrolidin-3-ylamino)ethyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C29H32F6N4O3
|
1
|
| 1 |
IC50 = 2210 nM
|
|
|
|
CP0315692
|
(S)-1-(4-(1-(4-(1H-indol-3-yl)piperidin-1-yl)-2-hydroxyethyl)piperidin-1-yl)-3-(3,4,5-trifluorophenyl)prop-2-en-1-one
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|
C29H32F3N3O2
|
1
|
| 1 |
IC50 = 2400 nM
|
|
|
|
CP0479934
|
(R)-N-(2-(1-(2-(1-(2-methylbenzoyl)piperidin-4-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
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|
C29H35F3N4O3
|
1
|
| 1 |
IC50 = 2880 nM
|
|
|
|
CP0095877
|
(R)-N-(2-(1-(2-(4-(2,5-difluorobenzoyl)piperazin-1-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C27H30F5N5O3
|
1
|
| 1 |
IC50 = 3040 nM
|
|
|
|
CP0513999
|
(R)-N-(2-(1-(2-(1-(4-chlorobenzoyl)piperidin-4-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C28H32ClF3N4O3
|
1
|
| 1 |
IC50 = 3160 nM
|
|
|
|
CP0277402
|
(R)-N-(2-(1-(4-chlorobenzyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C21H21ClF3N3O2
|
1
|
| 1 |
IC50 = 3200 nM
|
|
|
|
CP0373123
|
(R)-N-(2-(1-(2-(4-(4-methylbenzoyl)piperazin-1-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C28H34F3N5O3
|
1
|
| 1 |
IC50 = 3460 nM
|
|
|
|
CP0479936
|
(R)-N-(2-(1-(2-(4-(3-methylbenzoyl)piperazin-1-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C28H34F3N5O3
|
1
|
| 1 |
IC50 = 3520 nM
|
|
|
|
CP0479935
|
(R)-N-(2-(1-(2-(4-(2-methylbenzoyl)piperazin-1-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C28H34F3N5O3
|
1
|
| 1 |
IC50 = 4440 nM
|
|
|
|
CP0126803
|
2-(3-isopropylureido)-N-(2-((1S,2R)-2-(4-(methylthio)benzamido)cyclohexylamino)-2-oxoethyl)-5-(trifluoromethyl)benzamide
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|
C28H34F3N5O4S
|
1
|
| 1 |
IC50 = 5100 nM
|
|
|
|
CP0521442
|
(R)-N-(2-(1-(2-(1-(4-fluorobenzoyl)piperidin-4-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C28H32F4N4O3
|
1
|
| 1 |
IC50 = 6600 nM
|
|
|
|
CP0514000
|
(R)-N-(2-(1-(2-(1-(3,4-dichlorobenzoyl)piperidin-4-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C28H31Cl2F3N4O3
|
1
|
| 1 |
IC50 = 7520 nM
|
|
|
|
CP0504526
|
(R)-N-(2-(1-(2-(1-(3-fluorobenzoyl)piperidin-4-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C28H32F4N4O3
|
1
|
| 1 |
IC50 = 8330 nM
|
|
|
|
CP0390964
|
N-[2-[[(3R)-1-[2-(4-benzoylpiperazin-1-yl)butyl]pyrrolidin-3-yl]amino]-2-oxoethyl]-3-(trifluoromethyl)benzamide
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|
C29H36F3N5O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0390965
|
N-[2-[[(3R)-1-[1-(4-benzoylpiperazin-1-yl)butan-2-yl]pyrrolidin-3-yl]amino]-2-oxoethyl]-3-(trifluoromethyl)benzamide
Show/Hide
|
C29H36F3N5O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
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CP0479937
|
N-[2-[[(3R)-1-[1-(4-benzoylpiperazin-1-yl)propan-2-yl]pyrrolidin-3-yl]amino]-2-oxoethyl]-3-(trifluoromethyl)benzamide
Show/Hide
|
C28H34F3N5O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0504527
|
(R)-N-(2-(1-(2-(4-(4-fluorobenzoyl)piperazin-1-yl)ethyl)pyrrolidin-3-ylamino)-2-oxoethyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C27H31F4N5O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0514001
|
N-[2-[[(3R)-1-[2-(4-benzoylpiperazin-1-yl)propyl]pyrrolidin-3-yl]amino]-2-oxoethyl]-3-(trifluoromethyl)benzamide
Show/Hide
|
C28H34F3N5O3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
