Brief Information of the Cell Line and Protein
Cell Line ID: CL000196 , MDA-MB-468
Synonyms
MDA-MB 468
MDA-MB468
MDAMB468
MDA-468
MDA468
MB468
MD Anderson-Metastatic Breast-468
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0419
Protein ID: PT00980 , Aurora kinase A
Gene Name AURKA
Organism Homo sapiens, Human
Protein Classification Kinase
Uniprot ID O14965
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000196  Protein ID: PT00980
 
Compound ID Compound Name Compound Formula
CP0147199
Bisanilinopyrimidine, 9c
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C20H20ClN5O2
 1
1
IC50 = 1000 nM
   TI
   LI
   LO
   TS
CP0247099
Bisanilinopyrimidine, 9e
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C18H16ClN5O
 1
1
IC50 = 1000 nM
   TI
   LI
   LO
   TS
CP0301029
Bisanilinopyrimidine, 9a
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C23H25ClN6O2
 1
1
IC50 = 1000 nM
   TI
   LI
   LO
   TS
CP0157791
Bisanilinopyrimidine, 9g
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C18H15ClN4O3
 1
1
IC50 = 3000 nM
   TI
   LI
   LO
   TS
CP0274623
Bisanilinopyrimidine, 12b
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C17H12ClFN8
 1
1
IC50 = 3000 nM
   TI
   LI
   LO
   TS
CP0704813
N4-(2-Chlorophenyl)-N2-[6-(1H-benzo[d]imidazol-2(3H)-one)]pyrimidine-2,4-diamine
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C17H13ClN6O
 1
1
IC50 = 3000 nM
   TI
   LI
   LO
   TS
CP0117152
Bisanilinopyrimidine, 12a
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C17H13ClN8
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0365386
Bisanilinopyrimidine, 12c
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C17H12ClFN8O
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0182104
Bisanilinopyrimidine inhibitor, 2
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C18H14N4O4
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0025009
Bisanilinopyrimidine, 9m
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C17H13ClFN5O
 1
1
IC50 < 300 nM
   TI
   LI
   LO
   TS
CP0103207
Bisanilinopyrimidine, 9n
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C16H13ClFN5O2S
 1
1
IC50 < 1000 nM
   TI
   LI
   LO
   TS
CP0170069
Bisanilinopyrimidine, 9d
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C17H15ClN4O2S
 1
1
IC50 < 1000 nM
   TI
   LI
   LO
   TS
CP0193836
Bisanilinopyrimidine, 9b
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C21H23ClN6O
 1
1
IC50 < 1000 nM
   TI
   LI
   LO
   TS