| Compound ID |
Compound Name |
Compound Formula |
|
CP0387547
|
(S)-4-(2,5-difluorophenyl)-N-methyl-N-(1-methylpiperidin-4-yl)-2-phenyl-2H-pyrrole-1(5H)-carboxamide
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|
C24H27F2N3O
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0452185
|
(2S)-4-(2,5-difluorophenyl)-N-(1-(2-fluoroethyl)piperidin-4-yl)-2-(hydroxymethyl)-N-methyl-2-phenyl-2,5-dihydro-1H-pyrrole-1-carboxamide
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|
C26H30F3N3O2
|
1
|
| 1 |
IC50 = 13800 nM
|
|
|
|
CP0495651
|
(2S)-4-(2,5-Difluorophenyl)-2-(hydroxymethyl)-N-methyl-N-(1-methylpiperidin-4-yl)-2-phenyl-2,5-dihydro-1H-pyrrole-1-carboxamide
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|
C25H29F2N3O2
|
1
|
| 1 |
IC50 = 14600 nM
|
|
|
|
CP0468453
|
(2S)-N-(1-cyclopropylpiperidin-4-yl)-4-(2,5-difluorophenyl)-2-(hydroxymethyl)-N-methyl-2-phenyl-2,5-dihydro-1H-pyrrole-1-carboxamide
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|
C27H31F2N3O2
|
1
|
| 1 |
IC50 = 15200 nM
|
|
|
|
CP0277177
|
(S)-2-((R)-3-amino-4,4-difluorobutyl)-4-(2,5-difluorophenyl)-N,N-dimethyl-2-phenyl-2H-pyrrole-1(5H)-carboxamide
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|
C23H25F4N3O
|
1
|
| 1 |
IC50 = 15900 nM
|
|
|
|
CP0440516
|
(S)-4-(2,5-difluorophenyl)-2-(hydroxymethyl)-N-methyl-2-phenyl-N-(piperidin-4-yl)-2,5dihydro-1H-pyrrole-1-carboxamide
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|
C24H27F2N3O2
|
1
|
| 1 |
IC50 = 19200 nM
|
|
|
|
CP0201232
|
(2S)-4-(2,5-difluorophenyl)-N-[(3R,4S)-3-fluoro-1-methylpiperidin-4-yl]-2-(hydroxymethyl)-N-methyl-2-phenyl-2,5-dihydro-1H-pyrrole-1-carboxamide
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|
C25H28F3N3O2
|
1
|
| 1 |
IC50 = 20500 nM
|
|
|
|
CP0480241
|
(S)-4-(2,5-difluorophenyl)-N-((3S,4S)-3-fluoro-1-methylpiperidin-4-yl)-2-(hydroxymethyl)-N-methyl-2-phenyl-2H-pyrrole-1(5H)-carboxamide
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|
C25H28F3N3O2
|
1
|
| 1 |
IC50 = 36900 nM
|
|
|