General Information of the Compound
Compound ID
CP0926481
Compound Name
(2R)-3-[[2-[[(1S)-1-(4-Fluorophenyl)ethyl]amino]-6-[(5-methyl-1H-pyrazol-3-yl)amino]pyrimidin-4-yl]amino]propane-1,2-diol
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Structure
Formula
C19H24FN7O2
Molecular Weight
401.446
Canonical SMILES
Cc1cc(Nc2cc(NC[C@@H](O)CO)nc(N[C@@H](C)c3ccc(F)cc3)n2)n[nH]1
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InChI
InChI=1S/C19H24FN7O2/c1-11-7-18(27-26-11)23-17-8-16(21-9-15(29)10-28)24-19(25-17)22-12(2)13-3-5-14(20)6-4-13/h3-8,12,15,28-29H,9-10H2,1-2H3,(H4,21,22,23,24,25,26,27)/t12-,15+/m0/s1
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InChIKey
DGMFWDCPJFKXRN-SWLSCSKDSA-N
Physicochemical Property
logP
2.32902
Rotatable Bonds
9
Heavy Atom Count
29
Polar Areas
131.01
Hydrogen Bond Donor Count
6
Hydrogen Bond Acceptor Count
8
Complexity
29

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 24949705
SID: 56247479
ChEMBL ID
CHEMBL456323
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00934, High affinity nerve growth factor receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000243 MCF-10A Homo sapiens (Human)  1
1
EC50 = 60 nM
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