General Information of the Compound
Compound ID
CP0916928
Compound Name
Methyl {(S)-1-[(S)-2-(5-{6-[(2-{(S)-1-[(R)-2-(methoxycarbonylamino)-2-phenylacetyl]pyrrolidin-2-yl}-1H-imidazol-5-yl)buta-1,3-diynyl]-5-methylbiphenyl-3-yl}-1H-imidazol-2-yl)pyrrolidine-1-carbonyl]-2-methylpropyl}carbamate dihydrochloride
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Structure
Formula
C48H52Cl2N8O6
Molecular Weight
907.9
Canonical SMILES
COC(=O)N[C@H](C(=O)N1CCC[C@H]1c1ncc(-c2cc(C)c(C#CC#Cc3cnc([C@@H]4CCCN4C(=O)[C@H](NC(=O)OC)c4ccccc4)[nH]3)c(-c3ccccc3)c2)[nH]1)C(C)C.Cl.Cl
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InChI
InChI=1S/C48H50N8O6.2ClH/c1-30(2)41(53-47(59)61-4)45(57)55-24-15-23-40(55)44-50-29-38(52-44)34-26-31(3)36(37(27-34)32-16-8-6-9-17-32)21-13-12-20-35-28-49-43(51-35)39-22-14-25-56(39)46(58)42(54-48(60)62-5)33-18-10-7-11-19-33;;/h6-11,16-19,26-30,39-42H,14-15,22-25H2,1-5H3,(H,49,51)(H,50,52)(H,53,59)(H,54,60);2*1H/t39-,40-,41-,42+;;/m0../s1
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InChIKey
QTRDWBVLHZGUCW-WTMYFBLBSA-N
Physicochemical Property
logP
7.82692
Rotatable Bonds
10
Heavy Atom Count
64
Polar Areas
174.64
Hydrogen Bond Donor Count
4
Hydrogen Bond Acceptor Count
8
Complexity
64

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 126647191
ChEMBL ID
CHEMBL4763617
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00149, Nonstructural protein 5A
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000148 Huh-7 Homo sapiens (Human)  3
1
IC50 = 0.013 nM
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2
IC50 = 0.026 nM
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   TS
3
IC50 = 0.124 nM
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   LO
   TS