General Information of the Compound
Compound ID
CP0911504
Compound Name
Methyl {(1R)-2-[(2S)-2-{5-[4-(3-fluoro-5-{2-[(2S)-1-{(2S)-2-[(methoxycarbonyl)amino]-3-methylbutanoyl}pyrrolidin-2-yl]-1H-imidazol-5-yl}biphenyl-2-yl)buta-1,3-diyn-1-yl]-1H-imidazol-2-yl}pyrrolidin-1-yl]-2-oxo-1-phenylethyl}carbamate dihydrochloride
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Structure
Formula
C47H49Cl2FN8O6
Molecular Weight
911.863
Canonical SMILES
COC(=O)N[C@H](C(=O)N1CCC[C@H]1c1ncc(-c2cc(F)c(C#CC#Cc3cnc([C@@H]4CCCN4C(=O)[C@H](NC(=O)OC)c4ccccc4)[nH]3)c(-c3ccccc3)c2)[nH]1)C(C)C.Cl.Cl
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InChI
InChI=1S/C47H47FN8O6.2ClH/c1-29(2)40(53-46(59)61-3)44(57)55-23-14-22-39(55)43-50-28-37(52-43)32-25-35(30-15-7-5-8-16-30)34(36(48)26-32)20-12-11-19-33-27-49-42(51-33)38-21-13-24-56(38)45(58)41(54-47(60)62-4)31-17-9-6-10-18-31;;/h5-10,15-18,25-29,38-41H,13-14,21-24H2,1-4H3,(H,49,51)(H,50,52)(H,53,59)(H,54,60);2*1H/t38-,39-,40-,41+;;/m0../s1
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InChIKey
MVKJKNLCTCXSJR-DYNIUFMISA-N
Physicochemical Property
logP
7.6576
Rotatable Bonds
10
Heavy Atom Count
64
Polar Areas
174.64
Hydrogen Bond Donor Count
4
Hydrogen Bond Acceptor Count
8
Complexity
64

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 126647232
ChEMBL ID
CHEMBL4782728
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00149, Nonstructural protein 5A
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000148 Huh-7 Homo sapiens (Human)  4
1
IC50 = 0.0118 nM
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2
IC50 = 0.02 nM
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3
IC50 = 0.026 nM
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4
IC50 = 0.051 nM
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