General Information of the Compound
Compound ID
CP0870207
Compound Name
N-(4-methyl-5-(3-(pyridin-3-yl)-1H-indazol-6-yl)thiazol-2-yl)-2-(4-methylpiperazin-1-yl)acetamide
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Formula
C23H25N7OS
Molecular Weight
447.568
Canonical SMILES
Cc1nc(NC(=O)CN2CCN(C)CC2)sc1-c1ccc2c(-c3cccnc3)n[nH]c2c1
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InChI
InChI=1S/C23H25N7OS/c1-15-22(32-23(25-15)26-20(31)14-30-10-8-29(2)9-11-30)16-5-6-18-19(12-16)27-28-21(18)17-4-3-7-24-13-17/h3-7,12-13H,8-11,14H2,1-2H3,(H,27,28)(H,25,26,31)
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InChIKey
SQGJDOUFIABRAQ-UHFFFAOYSA-N
Physicochemical Property
logP
3.24272
Rotatable Bonds
5
Heavy Atom Count
32
Polar Areas
90.04
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
7
Complexity
32

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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ChEMBL ID
CHEMBL4798067
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00934, High affinity nerve growth factor receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  1
1
GI50 = 251 nM
   TI
   LI
   LO
   TS
Protein ID: PT00864, Vascular endothelial growth factor receptor 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  1
1
GI50 = 2630 nM
   TI
   LI
   LO
   TS