General Information of the Compound
Compound ID
CP0859051
Compound Name
N-[4-(2-[6-(4-aminopiperidino)-2-methyl-4-pyrimidinyl]amino-1,3-thiazol-5-yl)phenyl]-N'-phenylurea
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Structure
Formula
C26H28N8OS
Molecular Weight
500.632
Canonical SMILES
Cc1nc(Nc2ncc(-c3ccc(NC(=O)Nc4ccccc4)cc3)s2)cc(N2CCC(N)CC2)n1
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InChI
InChI=1S/C26H28N8OS/c1-17-29-23(15-24(30-17)34-13-11-19(27)12-14-34)33-26-28-16-22(36-26)18-7-9-21(10-8-18)32-25(35)31-20-5-3-2-4-6-20/h2-10,15-16,19H,11-14,27H2,1H3,(H2,31,32,35)(H,28,29,30,33)
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InChIKey
VFXYUDAAKURMHR-UHFFFAOYSA-N
Physicochemical Property
logP
5.22362
Rotatable Bonds
6
Heavy Atom Count
36
Polar Areas
121.09
Hydrogen Bond Donor Count
4
Hydrogen Bond Acceptor Count
8
Complexity
36

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 88876331
ChEMBL ID
CHEMBL3593284
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00980, Aurora kinase A
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000013 Sf9 Spodoptera frugiperda (Fall armyworm)  1
1
IC50 = 150 nM
   TI
   LI
   LO
   TS
Protein ID: PT01204, Receptor-type tyrosine-protein kinase FLT3
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000071 MOLM-13 Homo sapiens (Human)  1
1
GI50 = 16 nM
   TI
   LI
   LO
   TS
CL000013 Sf9 Spodoptera frugiperda (Fall armyworm)  1
1
IC50 = 73 nM
   TI
   LI
   LO
   TS
Protein ID: PT00864, Vascular endothelial growth factor receptor 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000013 Sf9 Spodoptera frugiperda (Fall armyworm)  1
1
IC50 = 53 nM
   TI
   LI
   LO
   TS