General Information of the Compound
Compound ID
CP0848763
Compound Name
4-(3,4-Difluoro-phenyl)-2-oxo-6-trifluoromethyl-1,2,3,4-tetrahydro-pyrimidine-5-carboxylic acid {3-[4-(4-fluoro-phenyl)-piperidin-1-yl]-propyl}-amide
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Structure
Formula
C26H26F6N4O2
Molecular Weight
540.508
Canonical SMILES
O=C1NC(C(F)(F)F)=C(C(=O)NCCCN2CCC(c3ccc(F)cc3)CC2)[C@@H](c2ccc(F)c(F)c2)N1
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InChI
InChI=1S/C26H26F6N4O2/c27-18-5-2-15(3-6-18)16-8-12-36(13-9-16)11-1-10-33-24(37)21-22(17-4-7-19(28)20(29)14-17)34-25(38)35-23(21)26(30,31)32/h2-7,14,16,22H,1,8-13H2,(H,33,37)(H2,34,35,38)/t22-/m1/s1
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InChIKey
JMHJPWHXTFNZBY-JOCHJYFZSA-N
Physicochemical Property
logP
4.6601
Rotatable Bonds
7
Heavy Atom Count
38
Polar Areas
73.47
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
3
Complexity
38

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 10792536
SID: 15831375
ChEMBL ID
CHEMBL90184
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01089, Alpha-1A adrenergic receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 19 nM
   TI
   LI
   LO
   TS
Protein ID: PT01007, Alpha-1B adrenergic receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000440 LM Homo sapiens (Human)  1
1
Ki = 270 nM
   TI
   LI
   LO
   TS
Protein ID: PT01004, Alpha-1D adrenergic receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 1200 nM
   TI
   LI
   LO
   TS