General Information of the Compound
Compound ID
CP0801129
Compound Name
SID862358
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Structure
Formula
C23H24ClN5O2
Molecular Weight
437.931
Canonical SMILES
CC(=O)N1CCN(c2ccc(Nc3nc(C)nc4c3oc3ccccc34)cc2)CC1.Cl
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InChI
InChI=1S/C23H23N5O2.ClH/c1-15-24-21-19-5-3-4-6-20(19)30-22(21)23(25-15)26-17-7-9-18(10-8-17)28-13-11-27(12-14-28)16(2)29;/h3-10H,11-14H2,1-2H3,(H,24,25,26);1H
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InChIKey
KQEWWCQMRGIPKN-UHFFFAOYSA-N
Physicochemical Property
logP
4.51832
Rotatable Bonds
3
Heavy Atom Count
31
Polar Areas
74.5
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
6
Complexity
31

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 6603377
ChEMBL ID
CHEMBL1419089
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT02805, CREB-binding protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Potency = 31622.8 nM
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