General Information of the Compound
Compound ID
CP0790987
Compound Name
5-[2-Fluoro-4-(trifluoromethyl)phenyl]bicyclo[3.1.0]hex-2-yl}-(3-{[4-methyl-5-(4-methyl-1,3-oxazol-5-yl)-4H-1,2,4-triazol-3-yl]-thio}propyl)amine
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Structure
Formula
C23H26ClF4N5OS
Molecular Weight
532.007
Canonical SMILES
Cc1ncoc1-c1nnc(SCCCN[C@@H]2CC3C[C@]3(c3ccc(C(F)(F)F)cc3F)C2)n1C.Cl
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InChI
InChI=1S/C23H25F4N5OS.ClH/c1-13-19(33-12-29-13)20-30-31-21(32(20)2)34-7-3-6-28-16-8-15-10-22(15,11-16)17-5-4-14(9-18(17)24)23(25,26)27;/h4-5,9,12,15-16,28H,3,6-8,10-11H2,1-2H3;1H/t15?,16-,22+;/m1./s1
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InChIKey
ZQWGORNKXZEBSY-RFRLNANNSA-N
Physicochemical Property
logP
5.55032
Rotatable Bonds
8
Heavy Atom Count
35
Polar Areas
68.77
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
7
Complexity
35

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 52945022
ChEMBL ID
CHEMBL1258269
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01005, D(2) dopamine receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki > 3162.28 nM
   TI
   LI
   LO
   TS
Protein ID: PT00943, D(3) dopamine receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 31.62 nM
   TI
   LI
   LO
   TS