General Information of the Compound
Compound ID
CP0731719
Compound Name
(2R,3S,5R)-2-(2,5-difluorophenyl)-5-(3-(phenylsulfonyl)pyrrolo[3,4-c]pyrazol-5(1H,4H,6H)-yl)tetrahydro-2H-pyran-3-amine
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Structure
Formula
C22H22F2N4O3S
Molecular Weight
460.506
Canonical SMILES
N[C@H]1C[C@@H](N2Cc3[nH]nc(S(=O)(=O)c4ccccc4)c3C2)CO[C@@H]1c1cc(F)ccc1F
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InChI
InChI=1S/C22H22F2N4O3S/c23-13-6-7-18(24)16(8-13)21-19(25)9-14(12-31-21)28-10-17-20(11-28)26-27-22(17)32(29,30)15-4-2-1-3-5-15/h1-8,14,19,21H,9-12,25H2,(H,26,27)/t14-,19+,21-/m1/s1
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InChIKey
JLYGGWGXGVTQHE-XWRIVVANSA-N
Physicochemical Property
logP
2.6938
Rotatable Bonds
4
Heavy Atom Count
32
Polar Areas
101.31
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
6
Complexity
32

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 127035754
ChEMBL ID
CHEMBL3735843
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00989, Dipeptidyl peptidase 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000013 Sf9 Spodoptera frugiperda (Fall armyworm)  1
1
IC50 = 27000 nM
   TI
   LI
   LO
   TS
Protein ID: PT00907, Dipeptidyl peptidase 4
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000013 Sf9 Spodoptera frugiperda (Fall armyworm)  1
1
IC50 = 0.4 nM
   TI
   LI
   LO
   TS
Protein ID: PT00975, Dipeptidyl peptidase 8
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000053 COS-7 Chlorocebus aethiops (Green monkey)  1
1
IC50 = 41000 nM
   TI
   LI
   LO
   TS