General Information of the Compound
Compound ID
CP0715133
Compound Name
2-((3S,4S)-4-Amino-3-methyl-2-oxa-8-azaspiro[4.5]decan-8-yl)-5-((2-(trifluoromethyl)pyridin-3-yl)thio)pyrimidin-4(3H)-one
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Structure
Formula
C19H22F3N5O2S
Molecular Weight
441.479
Canonical SMILES
C[C@@H]1OCC2(CCN(c3ncc(Sc4cccnc4C(F)(F)F)c(=O)[nH]3)CC2)[C@@H]1N
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InChI
InChI=1S/C19H22F3N5O2S/c1-11-14(23)18(10-29-11)4-7-27(8-5-18)17-25-9-13(16(28)26-17)30-12-3-2-6-24-15(12)19(20,21)22/h2-3,6,9,11,14H,4-5,7-8,10,23H2,1H3,(H,25,26,28)/t11-,14+/m0/s1
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InChIKey
CUPNFYMVCDYJQD-SMDDNHRTSA-N
Physicochemical Property
logP
2.6675
Rotatable Bonds
3
Heavy Atom Count
30
Polar Areas
97.13
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
7
Complexity
30

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 124150540
ChEMBL ID
CHEMBL4447768
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01346, Tyrosine-protein phosphatase non-receptor type 11
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000269 KYSE-520 Homo sapiens (Human)  1
1
IC50 = 1060 nM
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