General Information of the Compound
Compound ID
CP0692382
Compound Name
N-{4-[2-(6-Cyano-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-cyclohexyl}-3-(3-methanesulfonyl-phenyl)-acrylamide
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Formula
C28H34ClN3O3S
Molecular Weight
528.118
Canonical SMILES
CS(=O)(=O)c1cccc(/C=C/C(=O)N[C@H]2CC[C@H](CCN3CCc4cc(C#N)ccc4C3)CC2)c1.Cl
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InChI
InChI=1S/C28H33N3O3S.ClH/c1-35(33,34)27-4-2-3-22(18-27)8-12-28(32)30-26-10-6-21(7-11-26)13-15-31-16-14-24-17-23(19-29)5-9-25(24)20-31;/h2-5,8-9,12,17-18,21,26H,6-7,10-11,13-16,20H2,1H3,(H,30,32);1H/b12-8+;/t21-,26-;
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InChIKey
AWMRZHJPWZALJK-UCIRXCHQSA-N
Physicochemical Property
logP
4.52018
Rotatable Bonds
7
Heavy Atom Count
36
Polar Areas
90.27
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
5
Complexity
36

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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ChEMBL ID
CHEMBL2113352
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01005, D(2) dopamine receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 316.23 nM
   TI
   LI
   LO
   TS
Protein ID: PT00943, D(3) dopamine receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 5.012 nM
   TI
   LI
   LO
   TS