General Information of the Compound
Compound ID
CP0672452
Compound Name
2-(4-((2,4-diamino-5-methylquinazolin-6-ylamino)methyl)benzamido)pentanedioic acid
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Structure
Formula
C22H24N6O5
Molecular Weight
452.471
Canonical SMILES
Cc1c(NCc2ccc(C(=O)NC(CCC(=O)O)C(=O)O)cc2)ccc2nc(N)nc(N)c12
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InChI
InChI=1S/C22H24N6O5/c1-11-14(6-7-15-18(11)19(23)28-22(24)27-15)25-10-12-2-4-13(5-3-12)20(31)26-16(21(32)33)8-9-17(29)30/h2-7,16,25H,8-10H2,1H3,(H,26,31)(H,29,30)(H,32,33)(H4,23,24,27,28)
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InChIKey
MKOYTAPWWOTATD-UHFFFAOYSA-N
CAS
56277-34-0
Physicochemical Property
logP
1.76252
Rotatable Bonds
9
Heavy Atom Count
33
Polar Areas
193.55
Hydrogen Bond Donor Count
6
Hydrogen Bond Acceptor Count
8
Complexity
33

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 324351
ChEMBL ID
CHEMBL36866
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01651, Dihydrofolate reductase
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000341 WIL2 Homo sapiens (Human)  1
1
IC50 = 4.1 nM
   TI
   LI
   LO
   TS
Protein ID: PT01883, Thymidylate synthase
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000266 L1210 Mus musculus (Mouse)  1
1
IC50 = 150 nM
   TI
   LI
   LO
   TS