General Information of the Compound
Compound ID
CP0656008
Compound Name
ethyl 2-amino-6-n-propyl-4-(1-cyano-2-ethoxy-2-oxoethyl)-4H-chromene-3-carboxylate
    Show/Hide
Structure
Formula
C20H24N2O5
Molecular Weight
372.421
Canonical SMILES
CCCc1ccc2c(c1)C(C(C#N)C(=O)OCC)C(C(=O)OCC)=C(N)O2
    Show/Hide
InChI
InChI=1S/C20H24N2O5/c1-4-7-12-8-9-15-13(10-12)16(14(11-21)19(23)25-5-2)17(18(22)27-15)20(24)26-6-3/h8-10,14,16H,4-7,22H2,1-3H3
    Show/Hide
InChIKey
PILQZIAJJPUYDZ-UHFFFAOYSA-N
Physicochemical Property
logP
2.55138
Rotatable Bonds
7
Heavy Atom Count
27
Polar Areas
111.64
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
7
Complexity
27

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 16098790
SID: 24745398
ChEMBL ID
CHEMBL425792
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01216, Apoptosis regulator Bcl-2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000001 Jurkat Homo sapiens (Human)  1
1
GI50 = 5700 nM
   TI
   LI
   LO
   TS
Protein ID: PT01217, Bcl-2-like protein 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000001 Jurkat Homo sapiens (Human)  1
1
GI50 = 6300 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 70700 nM
Cell Viability or Cytotoxicity Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000001 Jurkat Homo sapiens (Human)  1
1
GI50 = 5200 nM
   TI
   LI
   LO
   TS