General Information of the Compound
Compound ID
CP0576042
Compound Name
2-[7-(difluoromethyl)-5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxo-1H-isoindol-2-yl]-2-(5,5-dimethyl-6,7-dihydropyrrolo[1,2-c]imidazol-1-yl)-N-(1,3-thiazol-2-yl)acetamide
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Structure
Formula
C37H38F2N6O3S
Molecular Weight
684.813
Canonical SMILES
CC1(C)CCc2c(ncn12)C(N1Cc2c(cc(cc2C(F)F)C#Cc2ccc(CN3CCC(CO)CC3)cc2)C1=O)C(=O)Nc1nccs1
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InChI
InChI=1S/C37H38F2N6O3S/c1-37(2)12-9-30-31(41-22-45(30)37)32(34(47)42-36-40-13-16-49-36)44-20-29-27(33(38)39)17-26(18-28(29)35(44)48)8-5-23-3-6-24(7-4-23)19-43-14-10-25(21-46)11-15-43/h3-4,6-7,13,16-18,22,25,32-33,46H,9-12,14-15,19-21H2,1-2H3,(H,40,42,47)
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InChIKey
XAARYUGOCWIQON-UHFFFAOYSA-N
Physicochemical Property
logP
5.8984
Rotatable Bonds
8
Heavy Atom Count
49
Polar Areas
103.59
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
8
Complexity
49

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 168283722
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00922, Epidermal growth factor receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  2
1
IC50 = 4 nM
   TI
   LI
   LO
   TS
2
IC50 = 12 nM
   TI
   LI
   LO
   TS