General Information of the Compound
Compound ID
CP0570196
Compound Name
1-[3-[2-[(5-thiophen-3-ylpyridin-2-yl)amino]-4-[3-(trifluoromethyl)anilino]pyrimidin-5-yl]phenyl]ethanone
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Structure
Formula
C28H20F3N5OS
Molecular Weight
531.563
Canonical SMILES
CC(=O)c1cccc(c1)-c1cnc(Nc2ccc(cn2)-c2ccsc2)nc1Nc1cccc(c1)C(F)(F)F
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InChI
InChI=1S/C28H20F3N5OS/c1-17(37)18-4-2-5-19(12-18)24-15-33-27(35-25-9-8-20(14-32-25)21-10-11-38-16-21)36-26(24)34-23-7-3-6-22(13-23)28(29,30)31/h2-16H,1H3,(H2,32,33,34,35,36)
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InChIKey
ZMOZEVVIADAAHC-UHFFFAOYSA-N
Physicochemical Property
logP
7.9757
Rotatable Bonds
7
Heavy Atom Count
38
Polar Areas
79.8
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
7
Complexity
38

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 168271023
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT02790, Dipeptidyl peptidase 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000100 U-937 Homo sapiens (Human)  1
1
IC50 = 227.6 nM
   TI
   LI
   LO
   TS
CL000040 THP-1 Homo sapiens (Human)  1
1
IC50 = 307.5 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 155.7 nM