General Information of the Compound
Compound ID
CP0569186
Compound Name
2-[5-[2-(6-aminopyridin-3-yl)ethynyl]-7-fluoro-3-oxo-1H-isoindol-2-yl]-2-(6,7-dihydro-5H-pyrrolo[1,2-c]imidazol-1-yl)-N-(1,3-thiazol-2-yl)acetamide
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Structure
Formula
C26H20FN7O2S
Molecular Weight
513.558
Canonical SMILES
Nc1ccc(cn1)C#Cc1cc2C(=O)N(Cc2c(F)c1)C(C(=O)Nc1nccs1)c1ncn2CCCc12
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InChI
InChI=1S/C26H20FN7O2S/c27-19-11-16(4-3-15-5-6-21(28)30-12-15)10-17-18(19)13-34(25(17)36)23(24(35)32-26-29-7-9-37-26)22-20-2-1-8-33(20)14-31-22/h5-7,9-12,14,23H,1-2,8,13H2,(H2,28,30)(H,29,32,35)
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InChIKey
GTKRDVGWBDNWDV-UHFFFAOYSA-N
Physicochemical Property
logP
3.1377
Rotatable Bonds
4
Heavy Atom Count
37
Polar Areas
119.03
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
8
Complexity
37

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 168269395
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00922, Epidermal growth factor receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  2
1
IC50 = 116 nM
   TI
   LI
   LO
   TS
2
IC50 = 1100 nM
   TI
   LI
   LO
   TS