General Information of the Compound
Compound ID
CP0553258
Compound Name
N-[3-[2-[4-amino-1-[(3R)-1-methylpyrrolidin-3-yl]pyrazolo[3,4-d]pyrimidin-3-yl]ethynyl]-4-methylphenyl]-3-(trifluoromethyl)benzamide
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Structure
Formula
C27H24F3N7O
Molecular Weight
519.531
Canonical SMILES
CN1CC[C@H](C1)n1nc(C#Cc2cc(NC(=O)c3cccc(c3)C(F)(F)F)ccc2C)c2c(N)ncnc12
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InChI
InChI=1S/C27H24F3N7O/c1-16-6-8-20(34-26(38)18-4-3-5-19(12-18)27(28,29)30)13-17(16)7-9-22-23-24(31)32-15-33-25(23)37(35-22)21-10-11-36(2)14-21/h3-6,8,12-13,15,21H,10-11,14H2,1-2H3,(H,34,38)(H2,31,32,33)/t21-/m1/s1
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InChIKey
ZNLOMIKOARFGGZ-OAQYLSRUSA-N
Physicochemical Property
logP
4.26442
Rotatable Bonds
3
Heavy Atom Count
38
Polar Areas
101.96
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
7
Complexity
38

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 122419228
ChEMBL ID
CHEMBL4783566
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00897, Potassium voltage-gated channel subfamily H member 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 680 nM
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