General Information of the Compound
Compound ID
CP0546696
Compound Name
5-(4-aminophenyl)-2-N-(5-thiophen-3-ylpyridin-2-yl)-4-N-[3-(trifluoromethyl)phenyl]pyrimidine-2,4-diamine
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Structure
Formula
C26H19F3N6S
Molecular Weight
504.541
Canonical SMILES
Nc1ccc(cc1)-c1cnc(Nc2ccc(cn2)-c2ccsc2)nc1Nc1cccc(c1)C(F)(F)F
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InChI
InChI=1S/C26H19F3N6S/c27-26(28,29)19-2-1-3-21(12-19)33-24-22(16-4-7-20(30)8-5-16)14-32-25(35-24)34-23-9-6-17(13-31-23)18-10-11-36-15-18/h1-15H,30H2,(H2,31,32,33,34,35)
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InChIKey
KMGCPKDAPLNDRR-UHFFFAOYSA-N
Physicochemical Property
logP
7.3553
Rotatable Bonds
6
Heavy Atom Count
36
Polar Areas
88.75
Hydrogen Bond Donor Count
3
Hydrogen Bond Acceptor Count
7
Complexity
36

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 168272562
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT02790, Dipeptidyl peptidase 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000040 THP-1 Homo sapiens (Human)  1
1
IC50 > 5000 nM
   TI
   LI
   LO
   TS
CL000100 U-937 Homo sapiens (Human)  1
1
IC50 > 5000 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 > 5000 nM