General Information of the Compound
Compound ID
CP0545265
Compound Name
N-[4-[[2-[2-(1,1-difluoroethyl)-4-fluorophenyl]-6H-thieno[2,3-e]indazol-3-yl]oxy]-2-methoxyphenyl]-1-(3-fluoropropyl)azetidin-3-amine
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Structure
Formula
C30H28F4N4O2S
Molecular Weight
584.639
Canonical SMILES
COc1cc(Oc2c(sc3c2ccc2[nH]ncc32)-c2ccc(F)cc2C(C)(F)F)ccc1NC1CN(CCCF)C1
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InChI
InChI=1S/C30H28F4N4O2S/c1-30(33,34)23-12-17(32)4-6-20(23)29-27(21-7-9-24-22(14-35-37-24)28(21)41-29)40-19-5-8-25(26(13-19)39-2)36-18-15-38(16-18)11-3-10-31/h4-9,12-14,18,36H,3,10-11,15-16H2,1-2H3,(H,35,37)
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InChIKey
WRJNMJDNMBEZFL-UHFFFAOYSA-N
Physicochemical Property
logP
7.952
Rotatable Bonds
10
Heavy Atom Count
41
Polar Areas
62.41
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
6
Complexity
41

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 168274413
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00886, Estrogen receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000083 MCF-7 Homo sapiens (Human)  1
1
EC50 = 1.1 nM
   TI
   LI
   LO
   TS
CL001042 HEK293/Gal4 Homo sapiens (Human)  1
1
IC50 = 0.6 nM
   TI
   LI
   LO
   TS
Protein ID: PT00897, Potassium voltage-gated channel subfamily H member 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 11500 nM
   TI
   LI
   LO
   TS