General Information of the Compound
Compound ID
CP0500801
Compound Name
5-[2-(4-chlorophenyl)-2-oxoethyl]sulfanyl-3-methyl-7-(2-methylpropyl)-1-propylpyrimido[4,5-d]pyrimidine-2,4-dione
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Structure
Formula
C22H25ClN4O3S
Molecular Weight
460.987
Canonical SMILES
CCCn1c2nc(CC(C)C)nc(SCC(=O)c3ccc(Cl)cc3)c2c(=O)n(C)c1=O
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InChI
InChI=1S/C22H25ClN4O3S/c1-5-10-27-19-18(21(29)26(4)22(27)30)20(25-17(24-19)11-13(2)3)31-12-16(28)14-6-8-15(23)9-7-14/h6-9,13H,5,10-12H2,1-4H3
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InChIKey
ZFNQZVBBVIGUGE-UHFFFAOYSA-N
Physicochemical Property
logP
3.7271
Rotatable Bonds
8
Heavy Atom Count
31
Polar Areas
86.85
Hydrogen Bond Donor Count
0
Hydrogen Bond Acceptor Count
8
Complexity
31

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 17559143
ChEMBL ID
CHEMBL2326942
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01305, 3',5'-cyclic-AMP phosphodiesterase 4B
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000012 Sf21 Spodoptera frugiperda (Fall armyworm)  1
1
IC50 = 26000 nM
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   LI
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   TS
Protein ID: PT00212, Phosphodiesterase
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000012 Sf21 Spodoptera frugiperda (Fall armyworm)  1
1
IC50 = 10000 nM
   TI
   LI
   LO
   TS