General Information of the Compound
Compound ID
CP0486326
Compound Name
US9353081, 3-1
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Synonyms
(+)-(R)-N-(4-(1-Methyl-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl)-5,6,7,8-tetrahydroisoquinolin-8-yl)propionamide
1428652-17-8
BDBM233806
Baxdrostat
Baxdrostat [INN]
CHEMBL4113975
CIN-107
CIN107
CS-0204056
GLXC-26998
GTPL12362
HY-132809
MS-25786
N-((8R)-5,6,7,8-Tetrahydro-4-(1,2,3,4-tetrahydro-1-methyl-2-oxo-6-quinolinyl)-8-isoquinolinyl)propanamide
N-[(8R)-4-(1-methyl-2-oxo-3,4-dihydroquinolin-6-yl)-5,6,7,8-tetrahydroisoquinolin-8-yl]propanamide
NF3P9Z8J5Y
Propanamide, N-((8R)-5,6,7,8-tetrahydro-4-(1,2,3,4-tetrahydro-1-methyl-2-oxo-6-quinolinyl)-8-isoquinolinyl)-
RO6836191
SCHEMBL14799753
UNII-NF3P9Z8J5Y
US9353081, 3-1
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Structure
Formula
C22H25N3O2
Molecular Weight
363.461
Canonical SMILES
CCC(=O)N[C@@H]1CCCc2c1cncc2-c1ccc2N(C)C(=O)CCc2c1
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InChI
InChI=1S/C22H25N3O2/c1-3-21(26)24-19-6-4-5-16-17(12-23-13-18(16)19)14-7-9-20-15(11-14)8-10-22(27)25(20)2/h7,9,11-13,19H,3-6,8,10H2,1-2H3,(H,24,26)/t19-/m1/s1
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InChIKey
VDEUDSRUMNAXJG-LJQANCHMSA-N
Physicochemical Property
logP
3.5612
Rotatable Bonds
3
Heavy Atom Count
27
Polar Areas
62.3
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
3
Complexity
27

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 71535962
SID: 163532664
ChEMBL ID
CHEMBL4113975
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT03119, Cytochrome P450 11B1, mitochondrial
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000405 G-402 Homo sapiens (Human)  1
1
EC50 = 980 nM
   TI
   LI
   LO
   TS
Protein ID: PT03120, Cytochrome P450 11B2, mitochondrial
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000405 G-402 Homo sapiens (Human)  1
1
EC50 = 14 nM
   TI
   LI
   LO
   TS
Clinical Information about the Compound
Drug 1 ( Baxdrostat )
Drug Name Baxdrostat
Company CinCor Pharma
Indication
Hypertension
Phase 2
Target(s)
Aldosterone synthase (CYP11B2)
Inhibitor