General Information of the Compound
Compound ID
CP0480062
Compound Name
1-(4,4-difluoropiperidin-1-yl)-4-[(10R,15S)-4-methyl-1,4,12-triazatetracyclo[7.6.1.05,16.010,15]hexadeca-5,7,9(16)-trien-12-yl]butan-1-one
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Structure
Formula
C23H32F2N4O
Molecular Weight
418.532
Canonical SMILES
CN1CCN2[C@H]3CCN(CCCC(=O)N4CCC(F)(F)CC4)C[C@H]3c3cccc1c23
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InChI
InChI=1S/C23H32F2N4O/c1-26-14-15-29-19-7-11-27(16-18(19)17-4-2-5-20(26)22(17)29)10-3-6-21(30)28-12-8-23(24,25)9-13-28/h2,4-5,18-19H,3,6-16H2,1H3/t18-,19-/m0/s1
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InChIKey
YNYJUMPPJZXNLG-OALUTQOASA-N
Physicochemical Property
logP
3.1522
Rotatable Bonds
4
Heavy Atom Count
30
Polar Areas
30.03
Hydrogen Bond Donor Count
0
Hydrogen Bond Acceptor Count
4
Complexity
30

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 90655116
ChEMBL ID
CHEMBL3233408
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT00825, 5-hydroxytryptamine receptor 2A
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000065 HEK293-EBNA Homo sapiens (Human)  1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
Protein ID: PT00939, 5-hydroxytryptamine receptor 2C
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000065 HEK293-EBNA Homo sapiens (Human)  1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
Protein ID: PT00957, D(2) dopamine receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS