General Information of the Compound
Compound ID
CP0468441
Compound Name
US8754075, 13
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Structure
Formula
C18H18F2N4O3
Molecular Weight
376.363
Canonical SMILES
COc1ccc(nc1)C(=O)Nc1ccc(F)c(c1)[C@@]1(C)N=C(N)OC[C@@H]1F
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InChI
InChI=1S/C18H18F2N4O3/c1-18(15(20)9-27-17(21)24-18)12-7-10(3-5-13(12)19)23-16(25)14-6-4-11(26-2)8-22-14/h3-8,15H,9H2,1-2H3,(H2,21,24)(H,23,25)/t15-,18+/m0/s1
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InChIKey
VVMUTCSDIWXUCG-MAUKXSAKSA-N
Physicochemical Property
logP
2.3798
Rotatable Bonds
4
Heavy Atom Count
27
Polar Areas
98.83
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
6
Complexity
27

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 66558690
SID: 152189119
ChEMBL ID
CHEMBL3680865
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01020, Beta-secretase 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000416 INS-1E Rattus norvegicus (Rat)  1
1
IC50 = 4 nM
   TI
   LI
   LO
   TS
Protein ID: PT01134, Beta-secretase 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000416 INS-1E Rattus norvegicus (Rat)  1
1
IC50 = 65 nM
   TI
   LI
   LO
   TS